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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

  1. Cat.No. 产品名称 Information
  2. GC18496 Leelamine (hydrochloride)

    脱氢松香胺盐酸盐

     An inhibitor of pyruvate dehydrogenase kinase
  3. GC18472 Elinogrel

    5-氯-N-[[[4-[6-氟-1,4-二氢-7-(甲基氨基)-2,4-二氧代-3(2H)-喹唑啉基]苯基]氨基]羰基]-2-噻吩磺酰胺,PRT060128

     A reversible P2Y12 antagonist
  4. GC18458 Terrein

    土曲霉酮

     A fungal metabolite with diverse biological activities
  5. GC18435 Arachidonoyl 2'-Chloroethylamide

    ACEA, 2'-chloro-AEA

     A potent and selective CB1 receptor agonist
  6. GC18412 VU0409551

    VU 0409551

     A positive allosteric modulator of mGluR5
  7. GC18348 Ceralifimod

    ONO-4641

     An agonist of S1P1 and S1P5 receptors
  8. GC18327 Todralazine (hydrochloride)

    盐酸托屈嗪,Ecarazine hydrochloride

     A β2-adrenergic receptor antagonist
  9. GC18318 CAY10441

    RO1138452

     An IP receptor antagonist
  10. GC18255 Xanomeline (oxalate)

    诺美林草酸盐,LY246708 oxalate

     Potent agonist of muscarinic receptors
  11. GC18244 Eltoprazine (hydrochloride)

    1-(2,3-二氢苯并[B][1,4]二氧杂芑-5-基)哌嗪,DU 28853 hydrochloride

     A partial agonist of 5-HT1A, 5-HT1B, and 5-HT2B receptors
  12. GC18216 ML314 An NTS1 agonist
  13. GC18202 Temocaprilat

    替莫普利

     An ACE inhibitor
  14. GC18152 AZ-3451

    (S)-2-(6-溴苯并[D][1,3]二氧杂环戊烯-5-基)-N-(4-氰基苯基)-1-(1-环己基乙基)-1H-苯并[D]咪唑-5-甲酰胺

     A PAR2 antagonist
  15. GC10311 Liraglutide

    利拉鲁肽

     利拉鲁肽是一种高效、长效的 GLP-1 受体激动剂 (EC50 = 61 pM)，其氨基酸序列与人 GLP-1 有 97% 的同一性 .用 PA/LPS 处理的肝细胞中的活细胞数量显着减少，利拉鲁肽以浓度依赖性方式逆转细胞活力的下降。
  16. GC16403 2-Arachidonoyl Glycerol

    2-花生酰基甘油乙腈溶液,2-AG

    Endogenous CB1 and CB2 receptor agonist
  17. GC16539 Butaprost

    布他前列素

     A selective agonist for the EP2 receptors
  18. GC17888 Metipranolol

    美替洛尔

     A β-AR antagonist
  19. GC12238 Oxomemazine

    双氧异丁嗪

     Oxomemazine 是一种基于吩噻嗪的组胺 H1 受体阻滞剂，具有明显的抗毒蕈碱特性。
  20. GC13844 p-iodo-Clonidine (hydrochloride) An α2-adrenergic receptor partial agonist
  21. GC14211 ONO-8130 A selective, orally bioavailable EP1 antagonist
  22. GC14300 GPR120 Compound A

    GPR120 cpdA

     A selective GPR120/FFAR4 agonist
  23. GC13180 Carazolol

    卡拉洛尔; (±)-Carazolol; DL-Carazolol; Suacron

     A β-AR ligand
  24. GC10283 γ-Linolenic Acid

    γ-亚麻酸 ;Gamma-Linolenic acid

     γ-Linolenic Acid是一种来源于琉璃苣油的口服ω-6多不饱和脂肪酸，可作为β-分泌酶（BACE1）的特异性抑制剂，IC50值为7.6×10−5mol/L，Ki值为3.5×10−5mol/L。
  25. GC14939 REV 5901 An antagonist of cysteinyl-leukotriene receptors
  26. GC12868 S-2 Methanandamide

    (S)-(+)-Arachidonyl-2'-Hydroxy-1'-Propylamide

     A potent CB1 receptor agonist
  27. GC13605 S-1 Methanandamide

    (S)-(−)-Arachidonyl-1'-Hydroxy-2'-Propylamide

     A CB1 receptor ligand
  28. GC17736 Anisodamine

    山莨菪碱; 6-Hydroxyhyoscyamine

     Anisodamine (6-Hydroxyhyoscyamine) 是一种颠茄生物碱，是一种非亚型选择性毒蕈碱，也是一种烟碱型胆碱受体拮抗剂。
  29. GC17488 Trimipramine (maleate)

    三甲丙咪嗪马来酸盐

     A tricyclic antidepressant
  30. GC11667 VU0483605 A selective mGlu1 PAM
  31. GC11668 ML-031

    CID-2113511

     A S1P2 agonist
  32. GC18132 U-44069

    9,11-dideoxy-9α,11α-epoxymethano PGF2α,9,11-dideoxy-9α,11α-epoxymethano Prostaglandin F2α,9,11-epoxymethano Prostaglandin H2

     A TP receptor agonist
  33. GC15365 N-Acetylserotonin

    N-乙酰-5-羟色胺,N-Acetyl-5-hydroxytryptamine,NAS

     N-Acetylserotonin是褪黑素生物合成中的一个化学中间体，以昼夜节律的方式激活酪氨酸激酶受体B（TrkB）。
  34. GC11350 6-OAU

    GTPL5846

     An agonist for GPR84
  35. GC11966 O-Phospho-D-Serine

    D-O-Phosphoserine,D-Serine-O-Phosphate,D-SOP

    weak agonist of the metabotropic glutamate receptor mGluR4
  36. GC12620 Calindol (hydrochloride) A calcimimetic and CaSR agonist
  37. GC12823 (R,S)-Atenolol

    阿替洛尔; (RS)-Atenolol

     A β1-AR antagonist
  38. GC16930 Adenosine Kinase Inhibitor (hydrate)

    ABT-702

     Blocks the action of adenosine kinase
  39. GC18041 NESS 0327 A potent CB1 receptor antagonist
  40. GC15327 Tetrahydromagnolol

    二丙基联苯二醇,Magnolignan

     An agonist of CB1 and CB2 and antagonist of GPR55
  41. GC15528 (±)trans-2,5-bis-(3,4,5-Trimethoxyphenyl)-1,3-dioxolane

    trans-BTP Dioxolane

     A PAF receptor antagonist
  42. GC11584 Butenoyl PAF A PAF analog
  43. GC13732 TG4-155 A brain penetrant EP2 antagonist
  44. GC14445 2-Ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridine

    咪唑并二甲基吡啶

     An angiotensin II receptor antagonist
  45. GC10020 γ-Linolenic Acid methyl ester

    r-亚麻酸甲酯,Methyl GLA,Methyl γ-Linolenate

     A dietary ω-6 PUFA
  46. GC12671 Angiotensin Fragment 1-7 (acetate) A type 1 angiotensin II receptor agonist
  47. GC14940 5-Methoxytryptamine

    5-甲氧基色胺
  48. GC13597 Pyrrolidino PAF C-16 A potent analog of PAF C-16
  49. GC13752 Hexanolamino PAF C-16 A PAF analog
  50. GC18125 DC260126 An FFAR1 (GPR40) antagonist
  51. GC17224 AH 23848 (calcium salt) Dual antagonist of TP and EP4 receptors

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