GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(40)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(450)
- Acetylcholine(19)
- Adenosine Deaminase(9)
- Adenosine Receptor(122)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(367)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(98)
- Bombesin Receptors(22)
- Bradykinin Receptors(26)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(90)
- Calcimimetic Agent(2)
- CaSR(19)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(65)
- Chemokine Receptors(25)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(63)
- CysLT1 receptor(1)
- Endothelin Receptor(44)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(18)
- GIP Receptor(5)
- Glucagon Receptor(59)
- Glucocorticoid Receptor(78)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(3)
- GPR119(10)
- GPR120(9)
- GPR35(7)
- GPR44(1)
- GPR55(8)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(52)
- LPA Receptor(12)
- LPL Receptor(52)
- mGluR (100)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(44)
- Melatonin Receptors(21)
- Motilin Receptor(6)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(17)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(38)
- Oxytocin Receptors(20)
- P2Y Receptor(51)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(155)
- Protease-Activated Receptors(10)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(32)
- Sigma Receptor(52)
- Vasopressin Receptor(28)
- 17,20-lyase(4)
- Ras(100)
- Urotensin-II Receptor(11)
- VIP Receptors(6)
- EBI2/GPR183(5)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(4)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(4)
- CRFR(21)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(23)
- GPR139(2)
- mAChR(164)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(67)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(18)
- GRK(1)
- Cat.No. 产品名称 Information
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GC26069
WAY-639889
WAY-639889 is a bioactive compound relative to neuropeptide Y-5.
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GC26027
V-0219
V-0219 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R), can be used for obesity-associated diabetes research.
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GC26016
TSHR antagonist S37
TSHR antagonist S37 is a selective and competitive antagonist of the thyrotropin receptor (TSHR).
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GC26002
Trazodone
Trazodone (AF-1161) is a 5-HT 2A/2C receptor antagonist that is used as an antidepressant for treating major depressive disorder and anxiety disorders.
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GC25898
SB 200646
SB 200646 (SB 200646A) is a potent, selective and oral-active antagonist of 5-HT2B/2C over 5-HT2A receptor with 50 fold selectivity. The pKi for rat 5-HT2C receptor, rat 5-HT2B receptor and rat 5-HT2A receptor are 6.9, 7.5 and 5.2, respectively. SB 200646 has electrophysiological and anxiolytic properties in vivo.
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GC25786
Propafenone
Propafenone (SA-79) is an orally active sodium channel blocking agent and a beta-adrenoceptor (β-adrenergic receptor) antagonist. Propafenone offers a broad spectrum of activity in the treatment of cardiac arrhythmias.
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GC25756
Pirenperone
Pirenperone (R-47456, R-50656), a quinazoline derivative, is a selective antagonist of SR-2A (5-HT2 serotonin receptor) when employed in low doses. Pirenperone behaves like a typical neuroleptic when used in higher doses (greater than 0.1 mg/kg).
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GC25728
PF-4136309
PF-4136309 (INCB8761, PF-04136309) is a potent, selective, and orally bioavailable CCR2 antagonist with an IC50 of 5.2 nM for human CCR2.
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GC25663
Nebivolol
Nebivolol (Bystolic,R 065824) is a β1 receptor blocker with nitric oxide-potentiating vasodilatory effect used in treatment of hypertension and also for left ventricular failure.
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GC25618
Maropitant citrate
Maropitant citrate is a novel neurokinin type-1 (NK1) receptor antagonist with anti-inflammatory and analgesic properties
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GC25569
Lerisetron
Lerisetron (F 0930, F 0930RS) is a 5-HT3 receptor antagonist with IC50 of 0.81μM.
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GC25563
Lasmiditan succinate
Lasmiditan succinate (COL-144, LY573144) is a novel, centrally acting, highly selective 5-HT(1F) receptor agonist (Ki=2.21 nM) without vasoconstrictor activity.
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GC25484
Guanabenz
Guanabenz (GBZ, GA, Wytensin, Wy-8678,BR-750) is an orally active central alpha 2-adrenoceptor (α2 adrenergic receptor) agonist with antihypertensive action.
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GC25434
Frovatriptan Succinate
Frovatriptan Succinate(SB 209509 Succinate,VML 251 Succinate) is the succinate salt form of frovatriptan, a synthetic triptan with serotonin (5-HT) receptor agonist activity especially for the 5-HT1B/1D receptors.
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GC25412
Fenoterol
Fenoterol (Phenoterol) is a β2 adrenoreceptor agonist with bronchodilator activity.
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GC25385
Esmolol
Esmolol is a cardioselective beta1 receptor blocker with rapid onset, a very short duration of action, and no significant intrinsic sympathomimetic or membrane stabilising activity at therapeutic dosages.
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GC25259
Cisapride hydrate
Cisapride (Propulsid, Alimix, Propulsin, Enteropride, Kinestase) acts directly as a selective serotonin 5-HT4 receptor agonist with IC50 of 0.483 μM. And It also acts indirectly as a parasympathomimetic.
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GC25253
Cinitapride Hydrogen Tartrate
Cinitapride Hydrogen Tartrate is a gastroprokinetic agent that acts as an agonist of the 5-HT1 and 5-HT4 receptors and as an antagonist of the 5-HT2 receptors
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GC25197
Carvedilol EP IMpurity E
Carvedilol is a nonselective beta blocker/alpha-1 blocker and used in management of congestive heart failure (CHF).
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GC25140
Bisoprolol
Bisoprolol is a cardioselective β1-adrenergic blocking agent used for secondary prevention of myocardial infarction (MI), heart failure, angina pectoris and mild to moderate hypertension.
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GC25120
Balixafortide (POL6326)
Balixafortide (POL6326) is an orally bioavailable peptidic CXC chemokine receptor 4 (CXCR4) antagonist
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GC25051
Alloxazine
Alloxazine (Isoalloxazine) is an A2 receptor antagonist, which is approximately 10-fold more selective for the A2B receptor than for the A2A receptor.
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GC25046
Albiglutide Fragment
Albiglutide fragment is one copy of a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36).
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GC67989
(S)-Mirtazapine
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GC67982
Treprostinil palmitil
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GC67979
MK-6884
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GC67977
Lubabegron
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GC67974
L-Glutamine-15N2
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GC67972
S-777469
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GC67957
Orexin A (human, rat, mouse) (acetate)
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GC67937
(R)-Mirtazapine
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GC67929
Orexin 2 Receptor Agonist 2
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GC67923
Renzapride
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GC67897
CCR8 antagonist 2
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GC67893
Sigma-LIGAND-1 hydrochloride
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GC67882
VU6028418
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GC67869
RPT193
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GC67795
P2Y2R/GPR17 antagonist 1
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GC67788
CCR6 antagonist 1
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GC67786
THX-B
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GC67768
TRV055 hydrochloride
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GC67726
ONO-8711 dicyclohexylamine
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GC67715
Upidosin
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GC67702
Abanoquil
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GC67692
Bufuralol
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GC67691
Midaglizole
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GC67683
Romifidine
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GC67681
(αR,8aS)-GSK1614343
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GC67620
Methacholine bromide
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GC66678
2-(3-Trifluoromethylphenyl)glycine hydrochloride