Endothelin Receptor(内皮素受体)
Endothelin receptors are members of rhodopsin-like g-protein coupled receptor (GPCRA) with 4 types (ETA, ETB1, ETB2 and ETC), which mediate various physiological processes including vasoconstriction, vasodilation, and neurotransmission etc.
- Cat.No. 产品名称 Information
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GC64457
Endothelin 1 (swine, human) (TFA)
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GC63837
Ro 46-8443
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GC61118
Nebentan potassium
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GC60544
A-192621
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GC60266
Nebentan free base
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GC60094
BQ-3020 TFA
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GC50247
A 127722
Highly potent, selective ETA antagonist; orally bioavailable
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GC45723
Macitentan-d4
An internal standard for the quantification of macitentan
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GC38641
IRL-1620 TFA
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GC37644
Sitaxsentan
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GC36525
Macitentan n-butyl analogue
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GC35811
Darusentan
An ETA receptor antagonist
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GC35546
BQ-788
A peptide ETB receptor antagonist
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GC35426
Atrial Natriuretic Peptide (ANP) (1-28), rat TFA
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GC35424
Atrasentan
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GC34031
PD-159020
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GC34025
Atrial Natriuretic Peptide (ANP) (1-28), human, porcine Acetate
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GC34023
Atrial Natriuretic Peptide (ANP) (1-28), human, porcine
An atrial natriuretic peptide
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GC32556
ZD-1611
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GC32548
Aminaftone (Aminaftone)
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GC32528
Ro 46-2005
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GC32479
Sparsentan (RE-021)
A dual antagonist of AT1 and ETA
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GC30942
Tezosentan (RO 610612)
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GC30937
IRL-1620
A peptide ETB receptor agonist
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GC30577
Endothelin Mordulator 1
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GC30485
Endothelin 1 swine, human
Endothelin 1 (swine, human) is a 21aa peptide vasoconstrictor and agonist of endothelin (ET) receptors ETA and ETB (IC50s = 0.15 and 0.12 nM, respectively).
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GC18501
Kendomycin
A cytotoxic macrolide
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GC11314
Atrial natriuretic factor (1-28) (rat)
Atrial natriuretic factor (1-28) (rat) 是大鼠体内 ANP 的主要循环形式,以浓度依赖性方式有效抑制血管紧张素 II (Ang II) 刺激的 endothelin-1 分泌。
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GC13175
Sarafotoxin S6a
Sarafotoxin S6a 是一种 sarafotoxin 类似物,是一种内皮素受体激动剂,具有与 Endothelin-3 相似的 ETA/ETB 选择性特征。
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GC14678
Sarafotoxin S6b
Sarafotoxin S6b 是一种血管收缩肽和非选择性内皮素受体激动剂。
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GC13924
Endothelin 3 (human, rat)
A peptide vasoconstrictor
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GC15246
IRL-2500
IRL-2500 是一种有效的内皮素受体拮抗剂。
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GC15887
BQ-123
A peptide ETA receptor antagonist
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GC12231
Sulfisoxazole
An antibiotic and endothelin receptor antagonist
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GC11465
Bosentan Hydrate
An antagonist of endothelin receptors
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GC16269
Bosentan
An antagonist of endothelin receptors
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GC17184
Ambrisentan
An ETA receptor antagonist
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GC17769
Sitaxentan sodium
A potent ETA receptor antagonist
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GC13236
ACT-132577
A dual ETA and ETB receptor antagonist and an active metabolite of macitentan
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GC15916
BQ-788 sodium salt
A peptide ETB receptor antagonist
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GC17785
Macitentan
A dual ETA/ETB receptor antagonist
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GC16862
Zibotentan (ZD4054)
A selective ETA receptor antagonist
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GC11405
Avosentan
Avosentan (Ro 67-0565; SPP-301) 是一种有效的选择性内皮素受体 (ETA 受体) 拮抗剂。
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GC11783
Atrasentan hydrochloride
Atrasentan hydrochloride (ABT-627 hydrochloride) 是一种选择性内皮素 A 受体拮抗剂,对 ETA 的 IC50 为 0.0551 nM。