Cannabinoid Receptor(大麻素受体)
The cannabinoid receptor (CB1 and CB2) is a member of G-protein coupled receptor which plays a significant role in physiologic processes such as cognitive and immune functions.
- Cat.No. 产品名称 Information
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GC10907
(±)-SLV 319
A selective antagonist of CB1
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GC10028
(R)-SLV 319
The inactive enantiomer of SLV 319
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GC63410
(Rac)-MRI-1867
(Rac)-MRI-1867 ((Rac)-MRI-1867, Compound 6b) 是一种大麻素受体 1 型 (CB1R)/iNOS 拮抗剂,对 CB1R 的 Ki 为 5.7 nM。
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GC10753
(S)-SLV 319
A selective antagonist of CB1
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GC16403
2-Arachidonoyl Glycerol
Endogenous CB1 and CB2 receptor agonist
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GC16196
2-Palmitoylglycerol
An endogenous fatty acid ester
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GC17100
4-Quinolone-3-Carboxamide CB2 Ligand
An Analytical Reference Standard
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GC15850
4-Quinolone-3-Carboxamide Furan CB2 Agonist
Selective CB2 agonist
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GC16480
AM 281
A CB1 receptor antagonist/inverse agonist
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GC62835
AM-6538
AM6538 是一种长效、高亲和力、伪不可逆的 cannabinoid (CB) 拮抗剂。AM6538 是利莫那班的结构类似物。AM6538可有效评价大麻素完全和部分激动剂的表观疗效。AM6538 可能在未来需要暂时减少大麻素受体可用性的研究中有用。
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GC15414
AM1241
A CB2 receptor agonist and inverse agonist
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GC15717
AM251
A CB1 receptor antagonist
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GC15093
AM4113
A CB1 receptor neutral antagonist
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GC10147
AM630
An inverse agonist at CB2 and partial agonist at CB1 receptors
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GC14661
AM6545
A peripherally restricted CB1 receptor antagonist
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GC35339
Anandamide
An endogenous cannabinoid
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GC18435
Arachidonoyl 2'-Chloroethylamide
A potent and selective CB1 receptor agonist
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GC16826
Arachidonoyl amide
An AEA analog with similar biological activity
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GC18097
Arachidonoyl Serinol
A CB1 receptor agonist
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GC11849
Arachidonyl serotonin
An inhibitor of FAAH
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GC10205
Arvanil
A structural analog of capsaicin with analgesic activity
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GC14115
AVE-1625
A potent CB1 receptor antagonist
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GC62855
AZD1940
AZD1940 是一种具有口服活性,高亲和力的大麻素 CB1/CB2 受体激动剂,对 CB1R 和 CB2R 的 pKi 值分别为 7.93 和 9.06,并具有强大的镇痛作用。
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GC61778
BAY 38-7271
BAY38-7271是一个选择性、高效的大麻素受体CB1/CB2激动剂,对人重组CB1和CB2作用的Ki值分别为1.85nM和5.96nM。BAY38-7271具有很强的神经保护特性。
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GC19060
Bay 59-3074
A partial agonist of CB1 and CB2 receptors
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GC11376
BML-190
A CB2 receptor inverse agonist
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GC66030
CB1 agonist 1
CB1 agonist 1 (compound 22) 是 CB1 的激动剂。CB1 agonist 1 与 CB1 受体的亲和力的 pIC50 值为 5.7。CB1 agonist 1可以用于大脑失调的研究。
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GC31306
CB1 antagonist 1
CB1antagonist1是CB1receptor的拮抗剂,可用于代谢综合征、肥胖、神经炎性疾病、认知障碍和精神病、胃肠功能紊乱和心血管疾病的研究。
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GC30935
CB1-IN-1
CB1-IN-1是一种新型外周大麻素-1受体(CB1R)拮抗剂,作用于CB1R(EC50=3nM)和CB2R,Ki值分别为0.3nM和21nM。
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GC33756
CB2R-IN-1
CB2R-IN-1是一种有效的cannabinoidCB2受体反向激动剂,Ki为0.9nM。
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GC18110
COR 170
COR 170 (11u) 是一种选择性 CB2 反向激动剂,它是一种 4-喹诺酮-3-羧酸衍生物,对 CB2 受体的 Ki 值为 3.8 nM。
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GC17205
CP-945598 HCl
A selective CB1 receptor antagonist
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GC50579
Ec2la
Ec2la 是一种口服活性大麻素 2 型受体 (CB2Rs) 正变构调节剂。
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GC11760
GW842166X
A CB2 receptor agonist
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GC17133
Hemopressin (human, mouse)
Hemopressin 是一种衍生自血红蛋白 α1 链的九肽,最初是从大鼠脑匀浆中分离出来的。
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GC17116
Hemopressin (rat)
Hemopressin (rat) 是一种衍生自血红蛋白 α1 链的九肽,最初是从大鼠脑匀浆中分离出来的。
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GC13660
JD5037
JD5037 是一种有效的 CB1R 拮抗剂,IC50 为 1.5 nM。
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GC16644
JTE 907
A selective CB2 receptor inverse agonist
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GC18496
Leelamine (hydrochloride)
An inhibitor of pyruvate dehydrogenase kinase
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GC50273
LEI 101 hydrochloride
Potent and selective CB2 partial agonist; orally biovailable
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GC12538
LH 21
Weak CB1 antagonist
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GC13318
LY 320135
A selective CB1 receptor antagonist
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GC19231
LY2828360
A selective CB2 receptor agonist
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GC12420
MAFP
An inhibitor of MAGL, FAAH, cPLA2, and iPLA2
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GC15788
MJ 15
A potent CB1 receptor antagonist
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GC11453
ML-191
An antagonist of GPR55
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GC14626
MM-22
biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamide
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GC14750
N-Arachidonylglycine
A metabolite of anandamide with analgesic activity
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GC31536
N-Oleoyl glycine
A putative substrate for peptidyl glycine α-
amidating enzyme -
GC18041
NESS 0327
A potent CB1 receptor antagonist