Cannabinoid Receptor(大麻素受体)
The cannabinoid receptor (CB1 and CB2) is a member of G-protein coupled receptor which plays a significant role in physiologic processes such as cognitive and immune functions.
Products for Cannabinoid Receptor
- Cat.No. 产品名称 Information
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GC10907
(±)-SLV 319
(±)-SLV319; (±)-BMS-646256
A selective antagonist of CB1 -
GC10028
(R)-SLV 319
The inactive enantiomer of SLV 319
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GC63410
(Rac)-MRI-1867
(Rac)-MRI-1867
(Rac)-MRI-1867 ((Rac)-MRI-1867, Compound 6b) 是一种大麻素受体 1 型 (CB1R)/iNOS 拮抗剂,对 CB1R 的 Ki 为 5.7 nM。 -
GC10753
(S)-SLV 319
伊必那班,Ibipinabant|BMS 646256|JD 5001
A selective antagonist of CB1 -
GC16403
2-Arachidonoyl Glycerol
2-花生酰基甘油乙腈溶液,2-AG
Endogenous CB1 and CB2 receptor agonist
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GC16196
2-Palmitoylglycerol
2-(1,3-二羟基丙-2-基)十六酸复合物1,3-二羟基丙-2-基棕榈酸酯(1:1),2-Palm-Gl
An endogenous fatty acid ester -
GC17100
4-Quinolone-3-Carboxamide CB2 Ligand
4Q3C CB2 Ligand
An Analytical Reference Standard -
GC15850
4-Quinolone-3-Carboxamide Furan CB2 Agonist
4Q3C CB2 Agonist
Selective CB2 agonist -
GC16480
AM 281
1-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-吗啉-1H-吡唑-3-甲酰胺
A CB1 receptor antagonist/inverse agonist -
GC62835
AM-6538
AM6538 是一种长效、高亲和力、伪不可逆的 cannabinoid (CB) 拮抗剂。AM6538 是利莫那班的结构类似物。AM6538可有效评价大麻素完全和部分激动剂的表观疗效。AM6538 可能在未来需要暂时减少大麻素受体可用性的研究中有用。
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GC15414
AM1241
A CB2 receptor agonist and inverse agonist
-
GC15717
AM251
1-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-(哌啶-1-基)-1H-吡唑-3-甲酰胺
AM251是一种 1 型大麻素受体 (CB1) 拮抗剂,IC50为8nM,同时也是G蛋白偶联受体55 (GPR55) 激动剂,其EC50为39nM。 -
GC15093
AM4113
AM4113
A CB1 receptor neutral antagonist -
GC10147
AM630
[6-碘-2-甲基-1-[2-(4-吗啉基)乙基]-1H-吲哚-3-基](4-甲氧基苯基)甲酮,AM 630;AM-630
An inverse agonist at CB2 and partial agonist at CB1 receptors -
GC14661
AM6545
A peripherally restricted CB1 receptor antagonist
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GC35339
Anandamide
花生四烯酸乙醇胺
An endogenous cannabinoid -
GC18435
Arachidonoyl 2'-Chloroethylamide
ACEA, 2'-chloro-AEA
A potent and selective CB1 receptor agonist -
GC16826
Arachidonoyl amide
Arachidonamide,Arachidonic Acid amide
An AEA analog with similar biological activity -
GC18097
Arachidonoyl Serinol
A CB1 receptor agonist
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GC11849
Arachidonyl serotonin
Arachidonyl serotonin; AA-5-HT
An inhibitor of FAAH -
GC10205
Arvanil
N-Vanillylarachidonamide
A structural analog of capsaicin with analgesic activity -
GC14115
AVE-1625
屈那班,Drinabant
A potent CB1 receptor antagonist -
GC62855
AZD1940
AZD1940 是一种具有口服活性,高亲和力的大麻素 CB1/CB2 受体激动剂,对 CB1R 和 CB2R 的 pKi 值分别为 7.93 和 9.06,并具有强大的镇痛作用。
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GC61778
BAY 38-7271
BAY38-7271是一个选择性、高效的大麻素受体CB1/CB2激动剂,对人重组CB1和CB2作用的Ki值分别为1.85nM和5.96nM。BAY38-7271具有很强的神经保护特性。
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GC19060
Bay 59-3074
A partial agonist of CB1 and CB2 receptors
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GC11376
BML-190
吲哚美辛吗啉代酰胺; Indomethacin morpholinylamide; IMMA
A CB2 receptor inverse agonist -
GC66030
CB1 agonist 1
CB1 agonist 1 (compound 22) 是 CB1 的激动剂。CB1 agonist 1 与 CB1 受体的亲和力的 pIC50 值为 5.7。CB1 agonist 1可以用于大脑失调的研究。
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GC31306
CB1 antagonist 1
CB1antagonist1是CB1receptor的拮抗剂,可用于代谢综合征、肥胖、神经炎性疾病、认知障碍和精神病、胃肠功能紊乱和心血管疾病的研究。
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GC30935
CB1-IN-1
1-(2,4-二氯苯基)-N-1-哌啶基-4-[[(1-吡咯烷基磺酰基)氨基]甲基]-5-[5-[2-[4-(三氟甲基)苯基]乙炔基]-2-噻吩基]-1H-吡唑-3-甲酰胺,BPRCB1184
CB1-IN-1是一种新型外周大麻素-1受体(CB1R)拮抗剂,作用于CB1R(EC50=3nM)和CB2R,Ki值分别为0.3nM和21nM。 -
GC33756
CB2R-IN-1
CB2R-IN-1是一种有效的cannabinoidCB2受体反向激动剂,Ki为0.9nM。
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GC18110
COR 170
COR 170 (11u) 是一种选择性 CB2 反向激动剂,它是一种 4-喹诺酮-3-羧酸衍生物,对 CB2 受体的 Ki 值为 3.8 nM。
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GC17205
CP-945598 HCl
CP 945598 Hydrochloride
A selective CB1 receptor antagonist -
GC50579
Ec2la
Ec2la 是一种口服活性大麻素 2 型受体 (CB2Rs) 正变构调节剂。
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GC11760
GW842166X
2-(2,4-二氯苯基氨基)-4-三氟甲基嘧啶-5-羧酸[(四氢吡喃-4-基)甲基]酰胺
A CB2 receptor agonist -
GC17133
Hemopressin (human, mouse)
Hemopressin 是一种衍生自血红蛋白 α1 链的九肽,最初是从大鼠脑匀浆中分离出来的。
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GC17116
Hemopressin (rat)
血红蛋白Α1链HEMOPRESSIN(RAT)
Hemopressin (rat) 是一种衍生自血红蛋白 α1 链的九肽,最初是从大鼠脑匀浆中分离出来的。 -
GC13660
JD5037
JD5037 是一种有效的 CB1R 拮抗剂,IC50 为 1.5 nM。
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GC16644
JTE 907
N-(1,3-苯并二氧戊环-5-基甲基)-1,2-二氢-7-甲氧基-2-氧代-8-(戊氧基)-3-喹啉甲酰胺
A selective CB2 receptor inverse agonist -
GC18496
Leelamine (hydrochloride)
脱氢松香胺盐酸盐
An inhibitor of pyruvate dehydrogenase kinase -
GC50273
LEI 101 hydrochloride
Potent and selective CB2 partial agonist; orally biovailable
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GC12538
LH 21
Weak CB1 antagonist
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GC13318
LY 320135
[6-甲氧基-2-(4-甲氧基苯基)苯并[B]呋喃-3-基](4-氰基苯基)甲酮
A selective CB1 receptor antagonist -
GC19231
LY2828360
A selective CB2 receptor agonist
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GC12420
MAFP
Methyl Arachidonyl Fluorophosphonate
An inhibitor of MAGL, FAAH, cPLA2, and iPLA2 -
GC15788
MJ 15
A potent CB1 receptor antagonist
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GC11453
ML-191
CCG-152883,CID-23612552
An antagonist of GPR55 -
GC14626
MM-22
biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamide
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GC14750
N-Arachidonylglycine
N-Arachidonyl Glycine, NAGly
A metabolite of anandamide with analgesic activity -
GC31536
N-Oleoyl glycine
A putative substrate for peptidyl glycine α-
amidating enzyme -
GC18041
NESS 0327
A potent CB1 receptor antagonist