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Home >> Signaling Pathways >> GPCR/G protein >> Cannabinoid Receptor

Cannabinoid Receptor(大麻素受体)

The cannabinoid receptor (CB1 and CB2) is a member of G-protein coupled receptor which plays a significant role in physiologic processes such as cognitive and immune functions.

Products for  Cannabinoid Receptor

  1. Cat.No. 产品名称 Information
  2. GC17116 Hemopressin (rat)

    血红蛋白Α1链HEMOPRESSIN(RAT)

     Hemopressin (rat) 是一种衍生自血红蛋白 α1 链的九肽，最初是从大鼠脑匀浆中分离出来的。
  3. GC13660 JD5037 JD5037 是一种有效的 CB1R 拮抗剂，IC50 为 1.5 nM。
  4. GC16644 JTE 907

    N-(1,3-苯并二氧戊环-5-基甲基)-1,2-二氢-7-甲氧基-2-氧代-8-(戊氧基)-3-喹啉甲酰胺

     A selective CB2 receptor inverse agonist
  5. GC18496 Leelamine (hydrochloride)

    脱氢松香胺盐酸盐

     An inhibitor of pyruvate dehydrogenase kinase
  6. GC50273 LEI 101 hydrochloride Potent and selective CB2 partial agonist; orally biovailable
  7. GC12538 LH 21 Weak CB1 antagonist
  8. GC13318 LY 320135

    [6-甲氧基-2-(4-甲氧基苯基)苯并[B]呋喃-3-基](4-氰基苯基)甲酮

     A selective CB1 receptor antagonist
  9. GC19231 LY2828360 A selective CB2 receptor agonist
  10. GC12420 MAFP

    Methyl Arachidonyl Fluorophosphonate

     An inhibitor of MAGL, FAAH, cPLA2, and iPLA2
  11. GC18866 MCHB-1

    NMethylcyclohexyl benzimidazole analog 1

     A CB2 receptor agonist
  12. GC91240 Methyl γ-Linolenyl Fluorophosphonate

    MγLnFP

    一种磷脂酶抑制剂
  13. GC15788 MJ 15 A potent CB1 receptor antagonist
  14. GC11453 ML-191

    CCG-152883,CID-23612552

     An antagonist of GPR55
  15. GC14626 MM-22

    biotinylated anandamide analog acts as a probe for visualizing the accumulation and intracellular trafficking of anandamide
  16. GC71262 Monlunabant Monlunabant ((S)-MRI-1891)是一种固体分散化合物，也是大麻素CB1受体抑制剂。
  17. GC70724 MRL-650 MRL-650（CB1反向激动剂1）是CB1受体的高效、口服活性和特异性反向激动剂，CB1和CB2受体的IC50分别为7.5 nM和4100 nM。
  18. GC14750 N-Arachidonylglycine

    N-Arachidonyl Glycine, NAGly

     A metabolite of anandamide with analgesic activity
  19. GC31536 N-Oleoyl glycine

    A putative substrate for peptidyl glycine α-amidating enzyme
  20. GC18041 NESS 0327 A potent CB1 receptor antagonist
  21. GC13267 NIDA 41020 A CB1 receptor antagonist
  22. GC69562 Nimacimab

    RYI-018

     Nimacimab (RYI-018) 是一种靶向 CB1 受体 的负变构调节单克隆抗体。Nimacimab 可用于代谢性疾病研究。
  23. GC17699 O-1821

    Cannabidiorcin, Cannabidiorcol, Cannabidiorocol, CBD-C1, CBDO

     An analog of O-1918, a selective antagonist of a non-CB1/CB2 receptor
  24. GC13847 O-1918

    1,3-二甲氧基-5-甲基-2-[(1R,6R)-3-甲基-6-(1-甲基乙烯基)-2-环己烯-1-基]苯

     A selective antagonist of abnormal cannabidiol-mediated effects
  25. GC14042 Oleamide

    油酸酰胺

     An amide of oleic acid and agonist of CB1 receptors
  26. GC30966 Olivetol

    橄榄醇

     An Analytical Reference Standard
  27. GC30504 Olorinab (APD 371)

    APD 371

    Olorinab (APD 371) (APD 371) 是一种高效、选择性和完全有效的 2 型大麻素受体 (CB2) 激动剂，对 hCB2 的 EC50 为 6.2 nM。
  28. GC10664 Org 27569

    ORG275695-氯-3-乙基-N-[2-[4-(1-哌啶基)苯基]乙基-1H-吲哚-2-甲酰胺

     Org 27569 是一种有效的 CB1 受体变构调节剂，可增加激动剂的结合，但阻断激动剂诱导的 CB1 信号传导。
  29. GC10843 Otenabant

    奥替那班,CP 945598;CP-945598;CP945598

     Otenabant 是一种有效的选择性大麻素受体 CB1 拮抗剂，Ki 为 0.7 nM，对人 CB2 受体的选择性高 10,000 倍。
  30. GC47866 Palmitoyl Ethanolamide-d5

    Palmidrold5, PEA15,15,16,16,16d5

     A neuropeptide with diverse biological activities
  31. GC16548 Palmitoylisopropylamide

    PIA

     FAAH inhibitor
  32. GC16171 PF 514273 CB1 receptor antagonist
  33. GC70955 PGN36 PGN36（化合物18）是一种选择性大麻素CB2受体（CB2R）拮抗剂，Ki为0.09µM。
  34. GC50387 PM 226 PM 226 是一种选择性大麻素 CB2R 激动剂 (Ki (CB2R)\u003d13 nM; EC50 (CB2R)\u003d39 nM; Ki (CB1R) \u003e40 μM;)，在体外和体内具有神经保护特性。
  35. GC12920 Pregnenolone

    孕烯醇酮; 3β-Hydroxy-5-pregnen-20-one

     A natural steroid hormone
  36. GC36963 Pregnenolone monosulfate

    3β-Hydroxy-5-pregnen-20-one monosulfate

     Pregnenolone monosulfate 是大麻素 CB1 受体的特异性抑制剂。
  37. GC44680 Pregnenolone sulfate (sodium salt)

    3β-Hydroxy-5-pregnen-20-one monosulfate sodium

     Pregnenolone sulfate (sodium salt)是一种孕烯醇酮的神经活性代谢产物，对氨基丁酸A型受体（GABAAR）的IC50值为26±2μmol/L，对不含γ亚基的GABAAR的IC50值为18±3μmol/L。
  38. GC65106 Pregnenolone-d4-1

    妊娠烯醇酮-D4,3β-Hydroxy-5-pregnen-20-one-d4-1

     Pregnenolone-d4-1 (3β-Hydroxy-5-pregnen-20-one-d4-1) 是一种氘代标记的 Pregnenolone。Pregnenolone (3β-Hydroxy-5-pregnen-20-one) 是一种功能强大的神经甾体，是包括甾体酮在内的各种甾体激素的主要前体。Pregnenolone 是大麻素 CB1 受体的信号传导特异性抑制剂，抑制由 CB1 受体介导的四氢大麻酚 (THC) 的作用。Pregnenolone 可以保护大脑免受大麻中毒。Pregnenolone 也是一种 TRPM3 通道激活剂，也可以弱激活 TRPM1 通道。
  39. GC50435 PSB CB5

    CID-85469571

     A GPR18 antagonist
  40. GC74008 PSB-KK1415 PSB-KK1415是人类孤儿G蛋白偶联受体GPR18的选择性激动剂，EC50为19.1nM。
  41. GC41087 PSB-SB1202 A CB1 and CB2 receptor agonist
  42. GC50143 PSNCBAM-1

    1-(4-氯苯基)-3-[3-[6-(吡咯烷-1-基)吡啶-2-基]苯基]脲

     A CB1 receptor antagonist
  43. GC14177 R-1 Methanandamide Phosphate

    R-1MAP,(R)-(+)-Arachidonyl-1'-Hydroxy-2'-Propylamide Phosphate

     A water soluble prodrug AEA analog
  44. GC13190 R-Palmitoyl-(1-methyl) Ethanolamide

    R-1 PMA

     A synthetic analog of palmitoyl ethanolamide
  45. GC17259 Rimonabant

    利莫那班; SR141716

     A potent and selective CB1 receptor antagonist
  46. GC16466 Rimonabant hydrochloride

    盐酸利莫那班; SR 141716A Hydrochloride

     A potent and selective CB1 receptor antagonist
  47. GC63617 RTICBM-189 RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.
  48. GC66413 RVD-Hpα TFA RVD-Hpα TFA is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist. RVD-Hpα TFA increases intracellular Ca2+ levels in cells expressing CB1 receptors in vitro. RVD-Hpα TFA also high affinity CB2 positive allosteric modulator (Ki=50 nM).
  49. GC13605 S-1 Methanandamide

    (S)-(−)-Arachidonyl-1'-Hydroxy-2'-Propylamide

     A CB1 receptor ligand
  50. GC12868 S-2 Methanandamide

    (S)-(+)-Arachidonyl-2'-Hydroxy-1'-Propylamide

     A potent CB1 receptor agonist
  51. GC67972 S-777469 S-777469 是一种选择性，具有口服活性的大麻素 2 型受体 (CB2) 激动剂，Ki 为 36 nM。S-777469 以剂量依赖性方式显著抑制化合物 48/80 诱导的小鼠抓挠行为。S-777469 通过 CB2 兴奋抑制瘙痒信号的传递，从而产生止痒作用。

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