Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(54)
- ATPase(70)
- Calcium Channel(289)
- Cannabinoid Transporters(6)
- CFTR(33)
- Chloride Channels(12)
- GABA Receptor(206)
- Glucose Transporters(8)
- Glutamate (EAAT) Transporters(18)
- Glycine Receptors(2)
- GlyT(17)
- GTPase(20)
- ICB(1)
- MCT2(2)
- Monoamine transporter(12)
- Monocarboxylate Transporters(10)
- Multidrug Transporters(4)
- Na+/Ca2+ Exchanger(15)
- NKCC(7)
- NMDA Receptor(74)
- Nucleoside Transporters(4)
- Pannexin-1(2)
- P2X purinergic receptor(61)
- P-gp(10)
- Proton Pump(52)
- Potassium Channel(258)
- Sodium Channel(170)
- TRP Channel(138)
- TRPV1(10)
- URAT1(5)
- Other Channel Modulators(9)
- MCT(3)
- Kainate Receptors(11)
- Ionophore(3)
- sodium-hydrogen exchanger(3)
- Chloride Channel(23)
- CRAC Channel(13)
- EAAT2(5)
- HCN Channel(4)
- Na+/HCO3- Cotransporter(1)
- Na+/K+ ATPase(28)
- P-glycoprotein(47)
- iGluR(140)
- nAChR(85)
- VDAC(2)
- Aquaporins(1)
- Piezo Channels(1)
- GlyR(1)
- Cat.No. 产品名称 Information
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GC26033
Veratrine
Veratridine (Cevadine, Cevadin, Cevadene), a steroidal alkaloid found in plants of the lily family, is a voltage-gated sodium channel activator. Veratridine induces anxiogenic-like behaviors in rats.
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GC26029
Valbenazine tosylate
Valbenazine tosylate (NBI-98854) is the tosylate salt of valbenazine, a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).
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GC25991
tetrathiomolybdate
Tetrathiomolybdate (TM) is used in the clinic for the treatment of Wilson's disease by inducing dimerization of the metal-binding domain of the cellular copper efflux protein ATP7B (WLN4) through a unique sulfur-bridged Mo2S6O2 cluster.
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GC25936
SLC13A5-IN-1
SLC13A5-IN-1 is a selective inhibitor of sodium-citrate co-transporter (SLC13A5/NaCT). It completely blocks the uptake of 14 C-citrate and has the potential for the treatment of metabolic and/or cardiovascular diseases.
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GC25812
Quinidine sulfate
Quinidine (Chinidin, Pitayine, β-quinine, (+)-quinidine) acts as a blocker of voltage-gated sodium channels, also an antimuscarinic and antimalarial.
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GC25566
L-DAB HBR
L-DAB HBR (L-Dab Hydrobromide, L-2,4-Diaminobutyric acid hydrobromide) is an inhibitor of GABA (Gamma-aminobutyric acid) transaminase with IC50 of >500 μM
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GC25558
Lanthanum(III) chloride heptahydrate
Lanthanum(III) chloride is the inorganic compound used in biochemical research to block the activity of divalent cation channels, mainly calcium channels.
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GC25531
Isonipecotic acid
Isonipecotic acid (4-Piperidinecarboxylic acid, 4-Carboxypiperidine, Hexahydroisonicotinic acid) is a heterocyclic compound that mainly acts as a GABAA receptor partial agonist.
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GC25405
Evodine
Evodine, a natural product extracted from Evodiae fructus (EF), is a biomarker for quality assessment of EF in the Chinese Pharmacopoeia. Evodine is a potent P-gp inhibitor.
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GC25386
Ethacrynate Sodium
Ethacrynate Sodium (ethacrynic acid sodium) is the sodium salt form of ethacrynic acid, which inhibits symport of sodium, potassium, and chloride primarily in the ascending limb of Henle, but also in the proximal and distal tubules.
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GC25345
Deudextromethorphan (AVP-786)
Deudextromethorphan (AVP-786) is an active N-methyl-D-aspartate (NMDA) receptor antagonist.
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GC25174
Brucine sulfate heptahydrate
Brucine is an alkaloid that acts as an antagonist at glycine receptors and paralyzes inhibitory neurons.
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GC25134
Benzocaine hydrochloride
Benzocaine hydrochloride (Ethyl 4-aminobenzoate, Ethyl p-aminobenzoate) is a surface anesthetic that acts by preventing transmission of impulses along nerve fibers and at nerve endings.
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GC67996
TPA-023B
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GC67949
GNE-0439
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GC67939
CFTR corrector 4
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GC67925
Crinecerfont hydrochloride
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GC67924
Dihydrocapsiate
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GC67922
Zelquistinel
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GC67920
WS-898
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GC67895
EVT-401
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GC67871
SSR504734
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GC67799
PF-05198007
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GC67789
SRI-37240
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GC67784
ML-SI3
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GC67767
(R)-Olacaftor
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GC67747
Dalazatide TFA
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GC67739
D-erythro-Sphingosine hydrochloride
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GC52503
FTase Inhibitor II (trifluoroacetate salt)
A potent, selective inhibitor of farnesyltransferase
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GC52466
ICR-1 (potassium salt)
A cell-impermeable fluorescent calcium indicator
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GC52465
ICR-1 AM
A cell-permeable fluorescent calcium indicator
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GC52250
Mevalonate (lithium salt)
An intermediate in the mevalonate pathway
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GC66843
L-Homocysteic acid
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GC66836
Dimethyl L-glutamate
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GC66470
SW157765
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GC66436
FEMA 4809
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GC66419
(R)-Lercanidipine-d3 hydrochloride
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GC66255
(E)-3,4,5-Trimethoxycinnamic acid
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GC66240
Lei-Dab7 TFA
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GC66073
Flupyradifurone
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GC66038
PF-06649298
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GC66016
Evifacotrep
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GC65999
piCRAC-1
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GC65959
CaV1.3 antagonist-1
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GC65954
Plazinemdor
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GC65940
Zandatrigine
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GC65611
AMG 333
A TRPM8 antagonist
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GC65593
6-Benzoylheteratisine
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GC65536
TRPV4 agonist-1
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GC65531
Hardwickiic acid