Proton Pump(质子泵)
Proton pump is a protein complex that transport the H+ ion across the membranes of lysosomes and vacuoles to generate an electrical and chemical gradient that provide energy for ATP synthesis from ADP.
- Cat.No. 产品名称 Information
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GC69839
(R)-Tegoprazan
(R)-Tegoprazan ((R)-CJ-12420; example 3) 是一种苯并咪唑衍生物,是一种有效的胃 H+/K+-ATP 酶抑制剂,对犬肾 Na+/K+-ATPase 的 IC50 为 98 nM。(R)-Tegoprazan 具有胃肠道疾病研究的潜力。
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GC25386
Ethacrynate Sodium
Ethacrynate Sodium (ethacrynic acid sodium) is the sodium salt form of ethacrynic acid, which inhibits symport of sodium, potassium, and chloride primarily in the ascending limb of Henle, but also in the proximal and distal tubules.
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GC65377
Abeprazan hydrochloride
Abeprazan (DWP14012) hydrochloride 是一种钾竞争性酸 (potassium-competitive acid) 阻滞剂。Abeprazan hydrochloride 通过可逆的钾竞争性离子结合抑制 H+,K+- ATPase,而无需酸激活。Abeprazan hydrochloride 是一种潜在的质子泵抑制剂,用于研究与酸相关的疾病。
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GC64070
Omeprazole-d3-1
An internal standard for the quantification of omeprazole
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GC63954
KM91104
KM 91104 is a cell-permeable inhibitor of V-ATPase that specifically targets the interaction between V-ATPase subunit a3 and subunit B2.
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GC63687
Rabeprazole-d4
An internal standard for the quantification of rabeprazole
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GC63472
Zastaprazan
Zastaprazan 是一种 proton pump 抑制剂 (WO2018008929)。Zastaprazan 可用于胃肠道炎症或胃酸相关疾病的研究。
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GC63335
Omeprazole-13CD3
Omeprazole-13CD3 (H 16868-13CD3) 是一种 13C 标记和氘代标记 Omeprazole。Omeprazole (H 16868) 是一种质子泵 (proton pump) 抑制剂 (PPI),有潜力用于胃肠道疾病的研究。Omeprazole 竞争性抑制 CYP2C19 活性,Ki 为 2 到 6 μM。Omeprazole 还抑制革兰氏阳性菌和革兰氏阴性菌生长。Omeprazole 是中性鞘磷脂酶 (N-SMase) 的抑制剂(外泌体抑制剂)。
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GC62885
Caloxin 2A1 TFA
Caloxin 2A1 TFA 是一种细胞外质膜 Ca2+-ATPase (PMCA) 肽抑制剂。Caloxin 2A1 TFA 不影响基础 Mg2+-ATPase 或 Na+-K+-ATPase。
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GC62823
Abeprazan
Abeprazan (DWP14012) 是一种钾竞争性酸 (potassium-competitive acid) 阻滞剂。Abeprazan 通过可逆的钾竞争性离子结合抑制 H+,K+- ATPase,而无需酸激活。Abeprazan 是一种潜在的质子泵抑制剂,用于研究与酸相关的疾病。
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GC61863
Verucopeptin
Verucopeptin 是一种有效的 HIF-1 (IC50=0.22 µM) 抑制剂,可以降低 HIF-1 靶基因的表达和 HIF-1α 的蛋白水平。通过直接靶向 v-ATPase ATP6V1G 亚基 (但不靶向 ATP1V1B2 或 ATP6V1D),Verucopeptin 强烈抑制 v-ATPase 活性。Verucopeptin 对耐药性癌细胞表现出抗肿瘤活性,常用作癌症相关研究。
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GC47537
Lansoprazole-d4
An internal standard for the quantification of lansoprazole
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GC61155
Omeprazole sodium
An irreversible inhibitor of the gastric proton pump
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GC60975
Lansoprazole Sulfide D4
LansoprazoleSulfideD4是LansoprazoleSulfide的氘代物。LansoprazoleSulfide是质子泵抑制剂Lansoprazole的活性代谢产物。LansoprazoleSulfide是一种口服活性抗结核药,细胞内的IC50值为0.59µM,肉汤中的IC50值为0.46µM。
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GC60929
Ilaprazole sodium
A gastric proton pump inhibitor
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GC60530
5-Hydroxylansoprazole
5-Hydroxylansoprazole(AG1908)是血浆中Lansoprazole的活性代谢产物。Lansoprazole由CYP2C19代谢形成5-Hydroxylansoprazole。Lansoprazole是一种胃质子泵(proton-pump)抑制剂,可有效研究各种消化系统疾病。
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GC39734
Diphyllin
A lignan with diverse biological activities
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GC39429
Rabeprazole Sulfide
An active metabolite of rabeprazole
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GC37920
Vonoprazan
A selective and reversible proton pump inhibitor
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GC37756
Tenatoprazole sodium
A proton pump inhibitor
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GC36848
Pantoprazole sodium hydrate
A proton pump inhibitor
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GC36847
Pantoprazole sodium
A proton pump inhibitor
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GC36806
Omeprazole D3
An internal standard for the quantification of omeprazole
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GC36009
Esomeprazole magnesium salt
An H+/K+-ATPase inhibitor
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GC35982
EN6
An activator of autophagy
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GC33575
Esomeprazole potassium salt ((S)-Omeprazole potassium)
An H+/K+-ATPase inhibitor
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GC32924
Linaprazan (AZD0865)
An H+/K+-ATPase inhibitor
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GC32250
Chebulinic acid
An ellagitannin with diverse biological activities
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GC31987
S3337
S3337是一种H+,K+-ATPase抑制剂。
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GC31969
Pumaprazole (BY-841)
Pumaprazole (BY-841) 是一种可逆的质子泵拮抗剂。
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GC31566
Tegoprazan
A proton pump inhibitor
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GC31466
Picoprazole
Picoprazole是一种特异性的H+/K+-ATPase抑制剂,IC50为3.1±0.4μM。
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GC31426
Bamaquimast (F 10126)
Bamaquimast (F 10126) (F 10126; L 0042) 是一种有效的平喘药。
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GC31347
Ilaprazole (IY-81149)
A gastric proton pump inhibitor
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GC30418
SKF96067
SKF96067是一种可逆的H+/K+-ATPase抑制剂。
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GC30130
Soraprazan (BYK61359)
Soraprazan (BYK61359) (BYK61359) 是一种选择性的、可逆的 K 竞争性 H,K-ATPase 抑制剂 (Ki=6.4 nM),在胃腺中的 IC50 为 0.19 μM。
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GC15334
N2-Methyl-L-arginine
Selective L-arginine uptake inhibitor
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GC11151
SCH 28080
An inhibitor of H+/K+-ATPases
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GC16516
BCH
An inhibitor of LAT1
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GC12718
Pantoprazole
A proton pump inhibitor
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GC16645
Rabeprazole
雷贝拉唑 (LY307640) 是第二代质子泵抑制剂 (PPI),可不可逆地灭活胃 H+/K+-ATPase。
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GC15670
Rabeprazole sodium
A proton pump inhibitor
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GC14313
Esomeprazole Magnesium
A form of esomeprazole in complex with magnesium
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GC16453
Zinc Pyrithione
A coordination complex of zinc and pyrithione
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GC16622
Dexlansoprazole
A proton pump inhibitor
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GC10599
Esomeprazole Sodium
An H+/K+-ATPase inhibitor
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GC12112
Lansoprazole sodium
Proton pump inhibitor
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GC17519
Concanamycin A
A plecomacrolide antibiotic
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GC17597
Bafilomycin A1
A fungal metabolite with diverse biological activities
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GC15418
TAK-438
A selective and reversible proton pump inhibitor