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Metabolism(代谢)

  1. Cat.No. 产品名称 Information
  2. GC91791 Cholic Acid 3-sulfate (potassium salt)

    3-Sulfocholate,3-Sulfocholic Acid

    Cholic acid 3-sulfate is a metabolite of the primary bile acid cholic acid .
  3. GC91783 FA16 FA16 is a ferroptosis inducer and an inhibitor of the system xc- cystine/glutamate transporter.
  4. GC91775 h-e5'NT Inhibitor 5C

    Human Ecto-5'-nucleotidase Inhibitor 5C

    h-e5'NT Inhibitor 5C is an inhibitor of ecto-5'-nucleotidase, also known as CD73 (IC50s = 0.37 and 1.66 µM for the human and rat enzymes, respectively).
  5. GC91773 18-hydroxy Oleoyl Leucine-d7 18-hydroxy Oleoyl leucine-d7 is intended for use as an internal standard for the quantification of 18-hydroxy oleoyl leucine by GC- or LC-MS.
  6. GC91768 GSK205 (hydrobromide) GSK205 is an inhibitor of transient receptor potential vanilloid 4 (TRPV4) and transient receptor potential ankyrin 1 (TRPA1; IC50s = 4.19 and 5.56 µM, respectively, for the rat channels).
  7. GC91767 ENPP3 Inhibitor 5J ENPP3 inhibitor 5J is an inhibitor of ectonucleotide pyrophosphatase/phosphodiesterase family member 1 (ENPP1) and ENPP3 (IC50s = 0.59 and 0.62 µM, respectively, for the human enzymes).
  8. GC91761 ABBV-CLS-484 (hydrochloride)

    Osunprotafib

    ABBV-CLS-484 is a dual inhibitor of protein tyrosine phosphatase 1N (PTP1N) and PTP2N (IC50s = 2.5 and 1.8 nM, respectively).
  9. GC91705 Etomidate-d5

    (+)-Etomidate-d5,d-Etomidate-d5,(R)-Etomidate-d5

    Etomidate-d5 is intended for use as an internal standard for the quantification of etomidate by GC- or LC-MS.
  10. GC91691 viFSP1

    Versatile Inhibitor of Ferroptosis Suppressor Protein 1,Versatile Inhibitor of FSP1

    viFSP1 is a species-independent inhibitor of ferroptosis suppressor protein 1 (FSP1; IC50s = 34 and 83 nM for the human and mouse enzymes, respectively).
  11. GC91690 TASP0277308 TASP0277308 is a sphingosine-1-phosphate receptor 1 (S1P1) antagonist (IC50 = 4.2 nM).
  12. GC91667 NSC 44625

    Bendroflumethiazide Impurity A,2,4-Disulfamyl-5-trifluoromethylaniline

    NSC 44625 is an inhibitor of carbonic anhydrase II (CAII; Ki = 63 nM for the human enzyme).
  13. GC91641 4-Hydroxy-1-(2-phenylethyl)piperidine 4-Hydroxy-1-(2-phenylethyl)piperidine is a building block that has been used in the synthesis of ligands of the muscarinic acetylcholine receptor (mAChR) or sigma non-opioid intracellular receptor 1 (σ1 receptor).
  14. GC91623 Ferroptosis Inducer 24 Ferroptosis inducer 24 is an inducer of ferroptosis.
  15. GC91613 FerroLOXIN-1 FerroLOXIN-1 is an inhibitor of the 15-lipoxygenase-2 (15-LO-2) and phosphatidylethanolamine-binding protein 1 (PEBP1) catalytic complex.
  16. GC91598 GPX4 16

    Glutathione Peroxidase 4 16

    GPX4 16 is an inhibitor of glutathione peroxidase 4 (GPX4).
  17. GC91548 Rosuvastatin EP Impurity A (calcium salt) Rosuvastatin EP impurity A is a potential impurity in commercial preparations of the HMG-CoA reductase inhibitor rosuvastatin.
  18. GC91547 Tanzawaic Acid B

    (+)-Tanzawaic Acid B

    Tanzawaic acid B is a fungal metabolite that has been found in Penicillium and has diverse biological activities.
  19. GC91543 (E/Z)-Droloxifene

    3-Hydroxytamoxifen

    (E/Z)-Droloxifene is a mixture of (E)-droloxifene, a selective estrogen receptor modulator (SERM), and (Z)-droloxifene.
  20. GC91499 Voriconazole-d3 N-oxide Voriconazole-d3 N-oxide is intended for use as an internal standard for the quantification of voriconazole N-oxide by GC- or LC-MS.
  21. GC91492 Propiverine N-oxide Propiverine N-oxide is an active metabolite of the muscarinic acetylcholine receptor antagonist propiverine .
  22. GC91489 Chondroitin Sulfate A (sodium salt)

    Chondroitin-4-sulfate,CSA

    Chondroitin sulfate A (CSA) is a glycosaminoglycan.
  23. GC91486 D-(+)-Ribonic Acid γ-lactone

    NSC 1031

    D-(+)-Ribonic acid γ-lactone is an oxidized derivative of ribose and a synthetic material.
  24. GC26431 Pentacosafluorotridecanoic Acid

    全氟十三烷酸,PFTrDA

    Perfluorotridecanoic Acid (Perfluorinated Compound (PFC)) is a perfluorinated alkyl acid (PFAA) and a possible organic pollutant.

  25. GC72637 Hexadecanoate-13C16 potassium Hexadecanoate-13C16 potassium是13C标记的十六烷酸钠。
  26. GC72527 S-(-)-Warfarin
  27. GC72482 Theodrenaline hydrochloride Theodrenaline hydrochloride是一种心脏兴奋剂,也与Cafedrine一起作为降压药。
  28. GC72481 Naveglitazar Naveglitazar(LY519818)是一种非噻唑烷二酮过氧化物酶体增殖物激活受体(PPAR)α-γ双γ显性激动剂,在动物模型中显示出降低血糖的潜力。
  29. GC72438 Osocimab Osocimab (BAY 1213790),抗fxia抗体(Ki=2.4 nM;EC50 = 0.2海里)。
  30. GC72222 Survodutide Survodutide(BI 456906)是一种强效的选择性胰高血糖素受体/GLP-1受体(GCGR/GLP-1R)双重激动剂,在CHO-K1细胞中的EC50分别为0.52 nM和0.33 nM。
  31. GC72096 Bamadutide Bamadutide(SAR425899)是一种强效的双胰高血糖素样肽-1受体/胰高血糖激素受体激动剂。
  32. GC72078 Azadiradione Azadiradione是在印度印楝中发现的一种生物活性类柠檬素。
  33. GC72068 Batatasin IV Batatasin IV是一种具有抗炎活性的LTA4H抑制剂。
  34. GC72026 Sclareol glycol Sclareol glycol是氨溴化酶的前体。
  35. GC71865 Palmitic acid-13C2 Palmitic acid-13C2是13C标记的棕榈酸。
  36. GC71863 Palmitic acid-13C16 sodium Palmitic acid-13C16 sodium是13C标记的棕榈酸钠。
  37. GC71840 L-Cystine-34S2 L-Cystine-34S2是34S标记的L-胱氨酸。
  38. GC71839 L-Cystine-d4 L-Cystine-d4是氘标记的L-胱氨酸。
  39. GC71837 L-Glutamine-13C5,15N2,d5 L-Glutamine-13C5,15N2,d5是氘、13C-和15-标记的L-谷氨酰胺。
  40. GC71789 ZY-1 ZY-1是ZY-2的控制分子。
  41. GC71730 L-Glutathione reduced-13C2,15N L-Glutathione reduced-13C2,15N13C和15N标记的L-谷胱甘肽是否减少。
  42. GC71605 Doxofylline-d6 Doxofylline-d6是氘标记的多索茶碱。
  43. GC71583 Dechloro Rivaroxaban Dechloro Rivaroxaban是一种高度选择性、口服活性的Xa因子抑制剂。
  44. GC71580 Otamixaban hydrochloride Otamixaban hydrochloride是一种强效、选择性、速效、竞争性和可逆的fXa抑制剂(Ki=0.5 nM),可有效抑制游离和凝血酶原酶结合的fXa。
  45. GC71535 Fuzapladib Fuzapladib(IS-741)是一种口服活性白细胞功能相关抗原1型(LFA-1)活化抑制剂,是一种白细胞粘附分子。
  46. GC71531 Ciraparantag acetate Ciraparantag acetate是凝血酶和Xa因子抑制剂。
  47. GC71502 CA/MAO-B-IN-1 CA/MAO-B-IN-1(化合物78)是人脑碳酸酐酶(CA)和单胺氧化酶-B(MAO-B)的双重抑制剂,IC50分别为8.8和7.0 nM。
  48. GC71498 Carbonic anhydrase inhibitor 16 Carbonic anhydrase inhibitor 16(化合物1)是一种登革热蛋白酶抑制剂,对碳酸酐酶hCA I和hCA II具有抑制活性(Ki:28.5 nM,2.2 nM)。
  49. GC71411 Dasatinib analog-1 Dasatinib analog-1(化合物5826)抑制CYP3A4的活性,Ki值为5.4μM。
  50. GC71393 Opevesostat Opevesostat是一种胆固醇侧链裂解酶(CYP11A1)抑制剂。
  51. GC71367 PPARγ-IN-2 PPARγ-IN-2(化合物5a)是PPARγ抑制剂。

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