Monoamine transporter(单胺转运蛋白)

Monoamine transporters are a family of plasma membrane transporter that regulates the reuptake of neurotransmitters into nerve terminals. It divided into DAT (dopamine transporter), NET (norepinephrine transporter) and SERT (serotonin transporter).

Cat.No. 产品名称 Information
GC69565 Nisoxetine Nisoxetine 是一种有效的和选择性的去甲肾上腺素转运蛋白 (NET) 抑制剂，Kd 值为 0.76 nM。Nisoxetine 是一种抗抑郁试剂和局部麻药，它可以阻断电压门控性钠通道。
GC26029 Valbenazine tosylate Valbenazine tosylate (NBI-98854) is the tosylate salt of valbenazine, a vesicular monoamine transporter 2 (VMAT2) inhibitor with a Ki value of 150 nM while displaying no significant binding to VAMT1(Ki<10 μM).
GC50649 FFN 200 dihydrochloride Selective fluorescent VMAT2 substrate
GC37820 Trans (2,3)-Dihydrotetrabenazine Trans (2,3)-Dihydrotetrabenazine，是抗精神病药物Tetrabenazine的体内代谢物，能够抑制囊泡单胺转运体 2 (VMAT2)。
GC37768 Tetrabenazine Racemate Tetrabenazine (Racemate)是一个有选择性和可逆转的VMAT-2抑制剂。
GC36705 NBI-98782
NBI-98782(alpha-dihydrotetrabenazine)是囊泡单胺转运体（VMAT2）抑制剂，Ki为0.97nM。
GC40180 Tetrabenazine-d6 An internal standard for the quantification of tetrabenazine
GC31060 Radafaxine hydrochloride (GW-353162A)
An active metabolite of bupropion
GC30994 Vanilpyruvic acid (Vanylpyruvic acid) 香草丙酮酸 (Vanylpyruvic acid) 是儿茶酚胺代谢物和香草乳酸的前体。
GC19370 Valbenazine An inhibitor of VMAT2
GC13672 Tetrabenazine
An inhibitor of VMAT2
GC14792 Reserpine hydrochloride Irreversible inhibitor of VMAT1 and VMAT2
GN10779 Reserpine Irreversible inhibitor of VMAT1 and VMAT2