AMPAR
AMPAR is an glutamate ionotropic α-amino-3-hydroxy- 5-methylisoxazole-4-propionic acid receptor that mediates fast excitatory synaptic transmission in the central nervous system.
Products for AMPAR
- Cat.No. 产品名称 Information
- GC50582 TAT-GluA2 3Y TAT-GluA2 3Y 是一种干扰肽,通过破坏 AMPAR 的内吞作用来阻断谷氨酸能突触的长期抑制 (LTD)。
- GC50428 UoS 12258 A positive allosteric modulator of AMPA receptors
- GC50111 CX 614 Positive allosteric modulator of AMPA receptors
- GC45989 JNJ-55511118 A negative modulator of AMPA receptors containing TARP-γ8
- GC12742 CP-465022 (maleate) An AMPA receptor antagonist
- GC12703 Philanthotoxin 74 An AMPA receptor antagonist
- GC13032 (RS)-AMPA hydrobromide AMPAR agonist
- GC14480 CNQX disodium salt A non-NMDA glutamate receptor antagonist
- GC13482 NBQX disodium salt An AMPA/kainate glutamate receptor antagonist
- GC17213 (S)-AMPA (S)-AMPA (L-AMPA) 是 AMPA 的活性 S-对映异构体,是一种有效的选择性 AMPA 受体激动剂。
- GC16011 L-Quisqualic acid A natural analog of glutamate
- GC13290 CMPDA A positive allosteric modulator of GluA2
- GC13684 S 18986 A positive allosteric modulator of AMPA receptors
- GC13007 PEPA A positive allosteric modulator of AMPA receptors
- GC10275 DNQX disodium salt A non-NMDA glutamate receptor antagonist
- GC13235 IEM 1925 dihydrobromide AMPA receptor antagonist
- GC11259 GYKI 47261 dihydrochloride AMPA receptor antagonist, non-competitive and selective
- GC14495 CX 546 CX 546 是第一代选择性苯甲酰胺型正 AMPAR 调节剂。
- GC12589 CP 465022 hydrochloride AMPA receptor antagonist, non-competitive and selective
- GC16909 YM 90K hydrochloride An AMPA receptor antagonist
- GC14842 GYKI 53655 hydrochloride GYKI 53655 (LY300168) hydrochloride 是一种 α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid (AMPA) 拮抗剂。
- GC16300 ZK 200775 ZK 200775 (ZK200775) 是一种高度选择性的 AMPA/红藻氨酸拮抗剂,对 NMDA 几乎没有活性; Ki 值分别为 3.2 nM、100 nM 和 8.5 μ;M 分别针对 quisqualate、红藻氨酸和 NMDA。
- GC11397 UBP 282 UBP 282 是一种有效的、选择性的和竞争性的 AMPA 和红藻氨酸受体拮抗剂。
- GC15012 Cl-HIBO Cl-HIBO 是一种高度亚型选择性的 GluR1/2 激动剂(EC50 分别为 4.7 和 1.7 μM)。
- GC14140 IEM 1460 An open channel blocker of calcium permeable glutamate receptors
- GC17313 (S)-CPW 399 AMPA agonist,subtype-selective,weakly desensitizing
- GC11301 GYKI 52466 dihydrochloride GYKI 52466 dihydrochloride 是一种具有口服活性、高选择性和非竞争性的 AMPA/红藻氨酸受体拮抗剂,IC50 值分别为 7.5 和 11μM。
- GC17928 IDRA 21 IDRA 21 是 AMPA 受体的阳性和口服活性调节剂。
- GC18079 CFM-2 CFM-2 是一种有效且选择性的非竞争性 AMPAR 拮抗剂。
- GC12863 1-BCP A positive allosteric modulator of AMPA receptors
- GC13728 SYM 2206 SYM 2206 是一种有效的非竞争性 AMPA 受体拮抗剂,IC50 为 1.6 μM。
- GC12207 Cyclothiazide A potentiator of AMPA receptors
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GC14156
NBQX
NBQX is a highly selective and competitive AMPA receptor antagonist.
- GC11889 (S)-(-)-5-Fluorowillardiine (S)-(-)-5-Fluorowillardiine 是一种有效且特异性的 AMPAR 激动剂。
- GC11799 CNQX CNQX是一种有效的竞争性AMPA /海藻酸酯受体(AMPA/kainate receptor)拮抗剂,IC50 分别为0.3µM和1.5µM。.
- GC13631 (RS)-AMPA (RS)-AMPA ((±)-AMPA) 是一种谷氨酸类似物和一种有效的选择性兴奋性神经递质 L-谷氨酸激动剂。
- GC14492 PF 4778574 PF 4778574 是 AMPA 受体的正向变构调节剂,在不同细胞中的 EC50 为 45 至 919 nM。
- GC14372 Pep2m, myristoylated Pep2m, myristoylated (Myr-Pep2m) 是一种细胞渗透性肽。
- GC12999 Pep1-AGL Analog of Pep1-TGL
- GC17103 Pep1-TGL Peptide containing the 'TGL' motif that corresponds to the C-terminus of GluR1 subunit
- GC11244 pep2-AVKI Inhibitor peptide that selectively disrupts binding of the GluR2 subunit(at the C-terminal PDZ site) to PICK1
- GC10669 pep2-EVKI 选择性破坏 GluR2 亚基(在 C 末端 PDZ 位点)与 PICK1 结合的抑制肽
- GC16112 pep2-SVKE Inactive control peptide analog of pep2-SVKI
- GC10272 pep2-SVKI Inhibitor peptide corresponding to last 10 amino acids of the C-terminus of the GluR2 subunit
- GC10551 pep4c Inactive control peptide analog of pep2m
- GC17069 pep2m GluR2亚基C端与N-乙基马来酰亚胺敏感融合蛋白相互作用的肽抑制剂
- GC14579 NPEC-caged-(S)-AMPA AMPA receptor agonist
- GC13349 Naspm trihydrochloride A synthetic analog of Joro spider toxin
- GC11598 Diazoxide An activator of SUR1/Kir6.2
- GC11071 (R)-AMPA inactive enantiomer of AMPA