GPR55(G蛋白偶联受体55)
GPR55 is a lysophosphatidylinositols and cannabinoids receptor. It is involved in various signaling cascade and plays a role in neuropathic/inflammatory pain, cancer and metabolic regulation etc.
Products for GPR55
- Cat.No. 产品名称 Information
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                     GC73616 
					
						
							GPR55 agonist 4							
                            									            
                    GPR55 agonist 4(化合物28)是GPR55激动剂(EC50:131nM,hGPR55和rGPR55为1.41nM)。           
					
					 
 
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                     GC69771 
					
						
							PSB-SB-487							
                            									            
                    PSB-SB-487 是一种有效的 GPR55 拮抗剂与 CB2 激动剂,对 GPR55 的 IC50 为 0.113 µM,对人 CB2 的 Ki 为 0.292 µM。PSB-SB-487 可用于研究糖尿病、帕金森病、神经性疼痛以及癌症。           
					
					 
 
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                     GC35694 
					
						
							CID 16020046							
                                                           
4-[4,6-二氢-4-(3-羟基苯基)-3-(4-甲基苯基)-6-氧代吡咯并[3,4-C]吡唑-5(1H)-基]苯甲酸
A selective GPR55 inverse agonist
 
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                     GC35339 
					
						
							Anandamide							
                                                           
花生四烯酸乙醇胺
Anandamide是一种来源于含花生四烯酸膜脂的内源性大麻素,通过结合并激活CB1和CB2大麻素受体以及香草素瞬时受体电位通道1(TRPV1)受体发挥作用。
 
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                     GC44217 
					
						
							ML-184							
                                                           
CID2440433
A synthetic agonist of GPR55
 
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                     GC14026 
					
						
							ML-193							
                                                           
CID-1261822
A selective GPR55 antagonist
 
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                     GC16103 
					
						
							Oleylethanolamide							
                                                           
油酰单乙醇胺,N-Oleoylethanolamide; Oleamide MEA; Oleic acid monoethanolamide
An endogenous, potent agonist for PPARα
 
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                     GC17777 
					
						
							Palmitoylethanolamide							
                                                           
十六酰胺乙醇,Palmidrol; Loramine P 256
An endogenous cannabinoid
 
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                     GC13513 
					
						
							O-1602							
                                                           
Abn-CBDO, Abnormal Cannabidiorcin, Abnormal Cannabidiorcinol, Abnormal Cannabiorcodiol
An agonist of GPR55
 
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                     GC12728 
					
						
							Abn-CBD							
                                                           
AbnCBD, ortho-Cannabidiol, o-CBD
An Analytical Reference Standard