Glucagon Receptor(胰高血糖素受体)
Glucagon receptor is a member of the class B G-protein coupled family of receptors and is activated by glucagon, resulting in activation of adenylate cyclase and increased levels of intracellular cAMP.
- Cat.No. 产品名称 Information
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GC26027
V-0219
V-0219 is an orally active, positive allosteric modulator (PAM) of the glucagon-like peptide-1 receptor (GLP-1R), can be used for obesity-associated diabetes research.
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GC25046
Albiglutide Fragment
Albiglutide fragment is one copy of a 30-amino-acid sequence of modified human GLP-1 (fragment 7-36).
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GC62753
[Des-His1,Glu9]-Glucagon amide TFA
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GC61545
GLP-1(28-36)amide
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GC61540
GLP-1(32-36)amide
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GC60877
GLP-2(3-33)
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GC60876
GLP-1(7-36), amide TFA
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GC60829
Exendin-3/4 (59-86)
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GC39364
Cotadutide acetate
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GC39323
{Val1}-Exendin-3/4
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GC38832
PF-06882961
Danuglipron (PF-06882961), a non-peptide agonist, activates the canonical G protein signaling activity only in the Glucagon-like peptide-1 (GLP-1) receptor with Trp33ECD.
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GC38495
Secretin (33-59), rat TFA
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GC38133
Tirzepatide (TFA)
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GC38132
Tirzepatide hydrochloride
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GC37929
VU0453379
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GC36753
NNC-0640
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GC36152
Glucagon-like peptide 1 (1-37), human (TFA)
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GC36150
Glucagon-Like Peptide (GLP) I (7-36), amide, human
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GC36148
GLP-1R Antagonist 1
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GC36147
GLP-1 receptor agonist 2
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GC43761
GLP-1 (1-37) (human, rat, mouse, bovine) (trifluoroacetate salt)
An incretin hormone
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GC43644
Exendin-4 (acetate)
A GLP-1R agonist
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GC34904
GLP-1(7-37) acetate
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GC34840
Tirzepatide
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GP21258
Glucagon (1-29), bovine, human, porcine
胰高血糖素是一种由 29 个氨基酸组成的肽,由胰腺 α 细胞分泌,以响应低血糖水平。
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GC34328
Semaglutide TFA
Semaglutide (Rybelsus, Ozempic, NN9535, OG217SC, NNC 0113-0217), a long-acting glucagon-like peptide 1 (GLP-1) analogue, is a GLP-1 receptor agonist with the potential for the treatment of type 2 diabetes mellitus (T2DM).
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GC34249
KQMEEEAVRLFIEWLKNGGPSSGAPPPS
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GC34246
FTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS
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GC34245
GTFTSDVSKQMEEEAVRLFIEWLKNGGPSSGAPPPS
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GC34244
GLP-1 moiety from Dulaglutide
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GC33759
GLP-1(7-36) Acetate (Human GLP-1-(7-36)-amide Acetate)
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GC33757
Glucagon (Porcine glucagon)
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GC31436
HAEGTFTSD
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GC31416
HAEGTFTSDVS
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GC31404
Semaglutide
A GLP-1R agonist
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GC31379
GRA Ex-25
GRAEx-25是一种glucagon受体的抑制剂,抑制大鼠和人的glucagon受体,IC50值分别为56和55nM。
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GC31363
GLP-1 receptor agonist 1
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GC31360
Taspoglutide (ITM077)
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GC31343
LGD-6972
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GC31334
Lixisenatide
Lixisenatide (Lyxumia, Adlyxin, ZP10A peptide, AVE0010) is a once-daily short-acting glucagon-like peptide-1 (GLP-1) receptor agonist (GLP-1RA) with an IC50 of 1.4 nM for the human GLP-1 receptor in receptor binding studies.
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GC31322
Adomeglivant (LY2409021)
An allosteric antagonist of the glucagon receptor
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GC30254
HAEGTFT
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GC30058
GLP-1(7-37)
An incretin hormone
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GC19170
Glucagon receptor antagonists-4
A GCGR antagonist
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GC10311
Liraglutide
A potent agonist of the GLP-1 receptor
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GC10075
Methylprednisolone Sodium Succinate
A prodrug form of methylprednisolone
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GC16232
BETP
A positive allosteric modulator of GLP-1R
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GC17298
L-168,049
L-168,049 是一种有效的、选择性的、具有口服活性的非竞争性胰高血糖素受体拮抗剂,对人、鼠和犬胰高血糖素受体的 IC50 分别为 3.7 nM、63 nM 和 60 nM。
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GC13743
GLP-1 (9-36) amide
GLP-1 (9-36) amide 是胰高血糖素样肽 1-(7-36) 酰胺的主要代谢物,由二肽基肽酶 4 (DPP-4) 形成。
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GC13075
GLP-2 (rat)
A gut peptide hormone antagonist of GLP-2R