Home >> Signaling Pathways >> GPCR/G protein >> Glucocorticoid Receptor

Glucocorticoid Receptor(糖皮质激素受体)

Glucocorticoid receptor is a neuroendocrine integration that functions as a major component of endocrine influence - specifically the stress response - upon the brain.

  1. Cat.No. 产品名称 Information
  2. GC68316 Loteprednol Etabonate-d5
  3. GC65370 ORIC-101
  4. GC65345 BI 653048
  5. GC64949 AZD5423
  6. GC64466 Dexamethasone-d5
  7. GC64330 Dazucorilant
  8. GC63872 Dagrocorat hydrochloride
  9. GC63739 Deflazacort-D5
  10. GC63738 Deflazacort-D7
  11. GC63737 21-Desacetyldeflazacort-D5
  12. GC62663 Glucocorticoid receptor agonist-1
  13. GC61850 Medroxyprogesterone acetate D3
  14. GC61536 Beclomethasone 17-propionate
  15. GC60914 Hydrocortisone hemisuccinate Hydrocortisone hemisuccinate (A-hydrocort, Hydrocortisone 21-hemisuccinate), a physiological glucocorticoid with anti-inflammatory properties, is an inhibitor of proinflammatory cytokine with IC50 of 6.7 μM and 21.4 μM for Interleukin-6 (IL-6) and IL-3, respectively.
  16. GC60467 21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione
  17. GC39564 Vamorolone
  18. GC39363 Cortodoxone Cortodoxone (11-Deoxycortisol, cortexolone, 11-Desoxycortisol, 17α,21-dihydroxyprogesterone), also known as 11-Deoxycortisol, is a glucocorticoid steroid hormone.
  19. GC39362 Clobetasone butyrate Clobetasone butyrate is a new corticosteroid that is often employed topically as a treatment for a variety of conditions such as eczema, psoriasis, various forms of dermatitis, and also for certain ophthalmologic conditions.
  20. GC39222 Fluticasone furoate A synthetic glucocorticoid
  21. GC45994 Hydrocortisone Acetate A synthetic corticosteroid
  22. GC38573 Dexamethasone palmitate 地塞米松棕榈酸酯 (DXP) 是地塞米松的前药。
  23. GC36962 Prednisone acetate Prednisone acetate (Betapar, Cortan, Deltasone, Fernisone, Meticorten, Prednisone 21-acetate) is a glucocorticoid steroid that can be used as a glucocorticoid receptor agonist with anti-inflammatory and immunomodulating properties.
  24. GC36961 Prednisolone Tebutate
  25. GC36809 OP-3633
  26. GC36269 Hydrocortisone phosphate
  27. GC36268 Hydrocortisone cypionate
  28. GC35843 Desisobutyryl-ciclesonide A glucocorticoid receptor agonist and the active metabolite of ciclesonide
  29. GC35503 Betamethasone hydrochloride A synthetic corticosteroid
  30. GC35502 Betamethasone acibutate
  31. GC35485 Beclometasone dipropionate Beclometasone二丙酸盐是糖皮质素激动剂,为beclometasone游离形式的原药。
  32. GC35002 (S)-Mapracorat
  33. GC34965 (20S)-Protopanaxatriol An active ginsenoside metabolite
  34. GC44678 Prednisolone Phosphate (sodium salt) A prodrug form of prednisolone
  35. GC42782 Amcinonide A synthetic corticosteroid
  36. GC42587 6α-Methylprednisolone 21-hemisuccinate A prodrug form of methylprednisolone
  37. GC40775 Dexamethasone A synthetic glucocorticoid
  38. GC40771 Fluorometholone A synthetic glucocorticoid
  39. GC33868 Triamcinolone Benetonide
  40. GC33856 Beclometasone (Beclomethasone) A glucocorticoid
  41. GC33839 Cortisone (17-Hydroxy-11-dehydrocorticosterone) A precursor and metabolite of cortisol
  42. GC32654 Relacorilant (CORT 125134) Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.
  43. GC32585 AZD2906
  44. GC32405 AL 082D06 (D06) A non-steroidal glucocorticoid receptor antagonist
  45. GC31936 GW-870086
  46. GC31929 Amebucort
  47. GC31894 AZD9567
  48. GC31885 Fosdagrocorat (PF-04171327)
  49. GC31844 Dagrocorat (PF-00251802)
  50. GC31747 Flunisolide A fluorinated corticosteroid receptor agonist
  51. GC31658 Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt)

    A glucocorticoid

Items 1 to 50 of 81 total

per page
  1. 1
  2. 2

Set Descending Direction