Glucocorticoid Receptor(糖皮质激素受体)
Glucocorticoid receptor is a neuroendocrine integration that functions as a major component of endocrine influence - specifically the stress response - upon the brain.
- Cat.No. 产品名称 Information
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GC68316
Loteprednol Etabonate-d5
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GC65370
ORIC-101
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GC65345
BI 653048
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GC64949
AZD5423
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GC64466
Dexamethasone-d5
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GC64330
Dazucorilant
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GC63872
Dagrocorat hydrochloride
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GC63739
Deflazacort-D5
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GC63738
Deflazacort-D7
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GC63737
21-Desacetyldeflazacort-D5
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GC62663
Glucocorticoid receptor agonist-1
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GC61850
Medroxyprogesterone acetate D3
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GC61536
Beclomethasone 17-propionate
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GC60914
Hydrocortisone hemisuccinate
Hydrocortisone hemisuccinate (A-hydrocort, Hydrocortisone 21-hemisuccinate), a physiological glucocorticoid with anti-inflammatory properties, is an inhibitor of proinflammatory cytokine with IC50 of 6.7 μM and 21.4 μM for Interleukin-6 (IL-6) and IL-3, respectively.
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GC60467
21-Acetoxypregna-1,4,9(11),16-tetraene-3,20-dione
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GC39564
Vamorolone
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GC39363
Cortodoxone
Cortodoxone (11-Deoxycortisol, cortexolone, 11-Desoxycortisol, 17α,21-dihydroxyprogesterone), also known as 11-Deoxycortisol, is a glucocorticoid steroid hormone.
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GC39362
Clobetasone butyrate
Clobetasone butyrate is a new corticosteroid that is often employed topically as a treatment for a variety of conditions such as eczema, psoriasis, various forms of dermatitis, and also for certain ophthalmologic conditions.
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GC39222
Fluticasone furoate
A synthetic glucocorticoid
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GC45994
Hydrocortisone Acetate
A synthetic corticosteroid
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GC38573
Dexamethasone palmitate
地塞米松棕榈酸酯 (DXP) 是地塞米松的前药。
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GC36962
Prednisone acetate
Prednisone acetate (Betapar, Cortan, Deltasone, Fernisone, Meticorten, Prednisone 21-acetate) is a glucocorticoid steroid that can be used as a glucocorticoid receptor agonist with anti-inflammatory and immunomodulating properties.
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GC36961
Prednisolone Tebutate
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GC36809
OP-3633
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GC36269
Hydrocortisone phosphate
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GC36268
Hydrocortisone cypionate
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GC35843
Desisobutyryl-ciclesonide
A glucocorticoid receptor agonist and the active metabolite of ciclesonide
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GC35503
Betamethasone hydrochloride
A synthetic corticosteroid
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GC35502
Betamethasone acibutate
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GC35485
Beclometasone dipropionate
Beclometasone二丙酸盐是糖皮质素激动剂,为beclometasone游离形式的原药。
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GC35002
(S)-Mapracorat
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GC34965
(20S)-Protopanaxatriol
An active ginsenoside metabolite
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GC44678
Prednisolone Phosphate (sodium salt)
A prodrug form of prednisolone
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GC42782
Amcinonide
A synthetic corticosteroid
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GC42587
6α-Methylprednisolone 21-hemisuccinate
A prodrug form of methylprednisolone
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GC40775
Dexamethasone
A synthetic glucocorticoid
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GC40771
Fluorometholone
A synthetic glucocorticoid
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GC33868
Triamcinolone Benetonide
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GC33856
Beclometasone (Beclomethasone)
A glucocorticoid
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GC33839
Cortisone (17-Hydroxy-11-dehydrocorticosterone)
A precursor and metabolite of cortisol
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GC32654
Relacorilant (CORT 125134)
Relacorilant (CORT125134) is a potent, selective and orally bioavailable glucocorticoid receptor antagonist, with a Ki of 7.2 nM in HepG2 TAT assay, and also shows Kis of 12, 81.2, 210 nM for rat, human and monkey glucocorticoid receptor in cell-based assay, respectively.
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GC32585
AZD2906
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GC32405
AL 082D06 (D06)
A non-steroidal glucocorticoid receptor antagonist
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GC31936
GW-870086
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GC31929
Amebucort
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GC31894
AZD9567
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GC31885
Fosdagrocorat (PF-04171327)
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GC31844
Dagrocorat (PF-00251802)
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GC31747
Flunisolide
A fluorinated corticosteroid receptor agonist
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GC31658
Dexamethasone phosphate disodium (Dexamethasone 21-phosphate disodium salt)
A glucocorticoid