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P2Y Receptor

P2Y Receptor is a family of purinergic G protein-coupled receptors, stimulated by nucleotides.

  1. Cat.No. Product Name Information
  2. GC41668 (±)-Clopidogrel (hydrochloride) Clopidogrel is an antithrombic compound whose active metabolite is a selective, irreversible antagonist of the platelet purinergic P2Y12 receptor (IC50 = 100 nM).
  3. GC60016 2-Methylthioadenosine diphosphate trisodium 2-Methylthioadenosinediphosphatetrisodium(2-Methylthio-ADPtrisodium)是一种有效的嘌呤能P2Y受体激动剂,对人P2Y13、小鼠P2Y13和人P2Y12的EC50分别为19、6.2和5nM。2-Methylthioadenosinediphosphatetrisodium对人P2Y1和大鼠P2Y6的pEC50分别为8.29和5.75。2-Methylthioadenosinediphosphatetrisodium诱导血小板聚集和形态改变,并抑制前列腺素E1作用下血小板内环腺苷酸的积累。
  4. GC14753 2-ThioUTP tetrasodium salt P2Y2 agonist
  5. GC13588 5-OMe-UDP trisodium salt Potent P2Y6 agonist
  6. GC50081 AR-C 118925XX

    Selective and competitive P2Y2 antagonist

  7. GC12914 AR-C 66096 tetrasodium salt P2Y12 antagonist,potent and selective
  8. GC14956 AZD1283 Potent P2Y12 antagonist
  9. GC19081 BPTU BPTU is a novel P2Y1 allosteric antagonist.
  10. GC43137 Cangrelor (sodium salt) Cangrelor is an ATP analog that inhibits platelet aggregation (IC50 = 0.4 nM).
  11. GC35710 Clopidogrel Clopidogrel 是一种以 P2Y12 受体为靶点的、具有口服活性 的血小板抑制剂。Clopidogrel 可用于抑制冠状动脉疾病、周围血管疾病和脑血管疾病中的血凝块。
  12. GC15964 Clopidogrel hydrogen sulfate P2Y12 receptor antagonist
  13. GC35711 Clopidogrel thiolactone Clopidogrel thiolactone是一种P2Y12受体抑制剂, 是一种有效的抗血小板药物。
  14. GC31664 Diquafosol tetrasodium (INS365) Diquafosoltetrasodium是一种P2Y2受体激动剂,可刺激眼睛表面的液体和粘蛋白分泌,用于干眼病的局部治疗。
  15. GC10124 DMNPE-caged ATP diammonium salt DMNPE-caged ATP
  16. GC18472 Elinogrel Elinogrel is a reversible antagonist of the platelet purinergic P2Y12 receptor (Ki = 23 nM) that inhibits platelet aggregation in a human platelet-rich plasma (hPRP) assay (IC50 = 2.81 nM).
  17. GC11311 MRS 2179 tetrasodium salt competitive antagonist at P2Y1 receptors
  18. GC15590 MRS 2211 P2Y13 receptor antagonist
  19. GC12723 MRS 2279 Selective, high affinity competitive antagonist of the P2Y1 receptor
  20. GC14852 MRS 2365 Highly potent, selective P2Y1 receptor agonist
  21. GC17476 MRS 2500 tetraammonium salt Highly potent and selective antagonist of the platelet P2Y1 receptor

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