OX Receptor(OX 受体)
OX receptor (orexin receptor) is a G-protein coupled receptor that is involved in the regulation of feeding behaviour.
- Cat.No. 产品名称 Information
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GC67957
Orexin A (human, rat, mouse) (acetate)
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GC67929
Orexin 2 Receptor Agonist 2
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GC65550
Danavorexton
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GC65382
Orexin receptor antagonist 5
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GC64826
Vornorexant
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GC64021
Orexin B, rat, mouse TFA
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GC63415
JNJ-54717793
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GC61770
Orexin receptor antagonist 2
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GC50559
YNT 185
YNT 185 是一种非肽、选择性食欲素 2 型受体 (OX2R) 激动剂,对于 OX2R 和 OX1R,EC50 分别为 0.028 和 2.75 μ;M。
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GC50142
ACT 462206
ACT 462206 是一种口服有效的 Orexin 1/Orexin 2 双重受体拮抗剂,IC50 分别为 60 nM (Orexin 1) 和 11 nM (Orexin 2)。
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GC38352
Orexin A (human, rat, mouse) (TFA)
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GC37623
Seltorexant
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GC36812
Orexin B, human TFA
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GC30941
Nemorexant (ACT-541468)
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GC30832
GSK1059865
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GC30829
IPSU
An orexin receptor 2 antagonist
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GC19323
SB-649868
A dual orexin receptor antagonist
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GC19272
Orexin 2 Receptor Agonist
An orexin 2 receptor agonist
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GC19250
MK-3697
An orexin receptor 2 antagonist
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GC19249
MK-1064
An orexin 2 receptor antagonist
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GC19220
Lemborexant
Lemborexant (E2006) is an oral active diorexin receptor antagonist (DORA) and has been approved by the US Food and Drug Administration for the treatment of insomnia.
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GC12242
MK 6096
A dual orexin receptor antagonist
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GC16336
ACT 335827
ACT 335827 是一种选择性、口服活性、脑渗透性食欲素 1 型受体拮抗剂。
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GC13741
EMPA
An OX2R receptor antagonist
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GC14809
JNJ 10397049
An oxrexin 2 receptor antagonist
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GC10549
TCS OX2 29
A selective orexin receptor 2 antagonist
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GC11818
OXA (17-33)
OXA (17-33) 是一种有效的选择性 orexin-1 受体 (OX1) 激动剂。
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GC17992
[Ala11,D-Leu15]-Orexin B
[Ala11,D-Leu15]-Orexin B 是一种有效的选择性orexin-2 受体 (OX2) 激动剂。
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GC16745
Orexin B (mouse)
Orexin B (mouse) (Rat orexin B) 是 Orexin 受体的内源性激动剂,对 OX1 和 OX2 的 Kis 分别为 420 和 36 nM。
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GC14887
Orexin B (human)
Orexin B (human) 是 Orexin 受体的内源性激动剂,对 OX1 和 OX2 的 Kis 分别为 420 和 36 nM。
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GC15034
SB-334867 free base
An orexin 1 receptor antagonist
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GC15317
SB408124
A potent orexin 1 receptor antagonist
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GC17807
TCS 1102
A dual orexin receptor antagonist
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GC13539
SB-334867
An orexin 1 receptor antagonist
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GC10050
Almorexant hydrochloride
An orexin 1 and orexin 2 receptor antagonist
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GC10717
Almorexant
Almorexant (ACT 078573) 是一种具有口服活性、强效和竞争性的双重食欲素受体拮抗剂,Kd 值分别为 1.3 nM (OX1) 和 0.17 nM (OX2)。
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GC15534
SB-674042
A potent and selective orexin 1 receptor antagonist
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GC16540
SB-408124 Hydrochloride
A potent orexin 1 receptor antagonist