Sigma Receptor(Sigma受体)
Sigma receptors are non-opioid receptors that interacted with psychostimulants such as cocaine and methamphetamine. It is associated with central nervous systems diseases, cancer and neuropathic pain etc.
- Cat.No. 产品名称 Information
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GC67893
Sigma-LIGAND-1 hydrochloride
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GC65450
CT1812
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GC65178
KB-5492 free base
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GC63801
CM398
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GC62960
EST73502 hydrochloride
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GC62959
EST64454 hydrochloride
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GC62708
σ1 Receptor antagonist-1
WQ 1 is a high affinity and selective σ1 receptor antagonist with pKi values of 10.85, 6.53 and 5.80 at σ1, σ2 receptors and dopamine transporter (DAT), displaying σ1/σ2 selectivity ratio of 20893.
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GC61926
Panamesine
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GC61889
OPC-14523 hydrochloride
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GC61838
Pentoxyverine
Pentoxyverine Citrate (Carbetapentane) is an antitussive (cough suppressant) commonly used for cough associated with illnesses like common cold.
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GC61822
DuP 734
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GC60216
KB-5492 anhydrous
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GC50048
(+/-)-PPCC oxalate
Selective sigma (σ) agonist (σ1> σ2)
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GC38721
(Rac)-E1R
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GC38714
(2S,3S)-E1R
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GC38713
(2R,3S)-E1R
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GC38712
(2R,3R)-E1R
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GC38048
Sigma-1 receptor antagonist 3
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GC38039
Sigma-1 receptor antagonist 2
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GC38038
Sigma-1 receptor antagonist 1
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GC35923
E1R
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GC33697
Cutamesine (SA4503)
Cutamesine (SA4503) (SA4503; AGY-94806) 是一种选择性 sigma 1 受体 (⌃1R) 激动剂;对 (+)-[3H]喷他佐辛标记的 sigma 1 受体亚型具有高亲和力(IC50= 17.4±;1.9 nM);对 sigma 2 受体的亲和力降低 100 倍。
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GC32821
Noscapine ((S,R)-Noscapine)
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GC31294
Sigma-LIGAND-1
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GC30956
Dimemorfan phosphate
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GC30206
Roluperidone (CYR-101)
A dual antagonist of 5-HT2A and σ2 receptors
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GC19032
AVex-73 hydrochloride
AVex-73 hydrochloride 是一种 Sigma-1 Receptor 激动剂,IC50 为 860 nM。
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GC17088
SA 4503 dihydrochloride
A selective σ1 receptor agonist
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GC18146
(+)-Igmesine hydrochloride
σ1 receptor ligand
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GC13796
BMY 14802 hydrochloride
BMY 14802 hydrochloride (BMY-14802-1) 是一种选择性和口服活性的 sigma 受体拮抗剂,IC50 为 112 nM。
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GC17380
Metaphit
Acylator of PCP and σ-receptors
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GC17721
IPAG
IPAG 是一种有效的 sigma-1 受体拮抗剂,pKi 为 4.3。 IPAG 诱导细胞凋亡。
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GC12490
L-693,403 maleate
High affinity σ ligand
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GC14249
UNC 0642
A G9a histone methyltransferase inhibitor
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GC15144
(±)-PPCC oxalate
sigma (σ) receptor ligand
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GC16004
NE 100 hydrochloride
A potent σ1 receptor antagonist
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GC16473
TC 1
σ1 receptor ligand
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GC11187
PD 144418 oxalate
PD 144418 oxalate 是一种高亲和力、有效和选择性的 sigma 1 (σ1) 受体配体(σ1 和 σ2 的 Ki 值分别为 0.08 nM 和 1377 nM)。
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GC17392
PB 28 dihydrochloride
A σ receptor ligand with anticancer and antiviral activities
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GC10795
Rimcazole dihydrochloride
Rimcazole (BW 234U) dihydrochloride 是一种咔唑衍生物,部分用作 sigma (σ) 受体拮抗剂。
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GC17301
(+)-SK&F 10047 hydrochloride
原型 σ1 受体激动剂
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GC15374
BD 1047 dihydrobromide
A selective antagonist of σ1 receptors
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GC15838
BD 1063 dihydrochloride
An antagonist of σ1 receptors
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GC17723
4-IBP
A σ1 receptor ligand
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GC13357
4-PPBP maleate
4-PPBP maleate 是一种有效的 σ 1 受体配体和激动剂。
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GC14960
PRE-084 hydrochloride
An Analytical Reference Standard
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GC16595
BD 1008 dihydrobromide
An Analytical Reference Standard
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GC16598
DTG
A σ receptor ligand
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GC13911
S1RA hydrochloride
A σ1 receptor antagonist
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GC10407
S1RA
A σ1 receptor antagonist