Free Fatty Acid Receptors(游离脂肪酸受体)

FFAR1 (GPR40) is a G protein-coupled receptor for medium and long chain saturated and unsaturated fatty acids. It plays a role in glucose homeostasis, insulin secretion and bone homeostasis etc.

Cat.No. 产品名称 Information
GC50662 DL 175 Potent and selective GPR84 biased agonist (EC50 = 33 nM)
GC50578 AZ 1729 AZ 1729 是一种有效的游离脂肪酸 2 受体 (FFA2) 激活剂，可作为直接变构激动剂和正变构调节剂。
GC50333 AMG 837 hemicalcium salt An FFAR1 (GPR40) partial
GC50313 ZQ 16 Selective GPR84 agonist
GC50293 CATPB CATPB 是一种有效的选择性游离脂肪酸受体 2 (FFA2R/GPR43) 拮抗剂。
GC16176 GSK 137647 A selective GPR120 agonist
GC17753 AH 7614 A selective FFAR4 antagonist
GC17149 4-CMTB A positive allosteric modulator of FFAR2/GPR43
GC11467 AS 2034178 AS 2034178 是一种特异性的口服活性 GPR40 激动剂，具有葡萄糖依赖性胰岛素分泌增强作用。
GC10373 MEDICA 16 A GPR40 agonist and GPR120 partial agonist
GC10922 TUG 424 A selective FFAR1 (GPR40) agonist
GC11434 GSK1292263 An agonist of GPR119
GC16555 TAK-875 A selective FFAR1 (GPR40) agonist
GC12401 GW9508 An agonist of GPR40
GC16054 TUG-770 An agonist of FFA1/GPR40
GC14027 GW-1100 A selective GPR40 antagonist