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Home >> Signaling Pathways >> GPCR/G protein >> Vasopressin Receptor

Vasopressin Receptor(血管加压素受体)

Vasopressin receptors are G-protein coupled receptors that mediate coagulation factor release, platelet aggregation, vasoconstriction, release of antidiuresis and ACTH release etc.

  1. Cat.No. 产品名称 Information
  2. GC66678 2-(3-Trifluoromethylphenyl)glycine hydrochloride
  3. GC65415 Felypressin acetate
  4. GC61959 D[LEU4,LYS8]-VP TFA
  5. GC39849 Atosiban acetate An oxytocin receptor antagonist
  6. GC39830 Terlipressin acetate A prodrug form of lysipressin
  7. GC50376 SSR 149415 强效选择性加压素 V1B 拮抗剂
  8. GC50246 TASP 0390325 TASP 0390325 是一种高亲和力和口服活性精氨酸加压素受体 1B（V1B 受体）拮抗剂，具有抗抑郁和抗焦虑活性。
  9. GC38948 SRX246
  10. GA20808 Big Endothelin-1 (1-39), porcine Big Endothelin-1 (1-39)，猪是 endothelin-1 的前体。
  11. GA20807 Big Endothelin-1 (1-38), human A peptide precursor of endothelin-1
  12. GA20084 (Deamino-Cys¹,β-cyclohexyl-Ala⁴,Arg⁸)-Vasopressin Studies revealed that this specific vasopressin agonist exhibited a nanomolar affinity for V-1b receptors from various mammalian species (bovine, human, rat). It exhibited high V-1b/V-1a and V-1b/oxytocin selectivity for rat, human, and bovine receptors. Furthermore, it showed a high V-1b/V-2 specificity for both bovine and human vasopressin receptors. Therefore, d(Cha?)-AVP is a promising tool for research of V-1b receptor structure-function relationships.
  13. GC44247 Mozavaptan (hydrochloride) A vasopressin V2 receptor antagonist
  14. GC32463 Terlipressin A prodrug form of lysipressin
  15. GC32453 Lixivaptan (VPA-985) A nonpeptide vasopressin V2 receptor antagonist
  16. GC31475 WAY-151932 (VNA-932)
  17. GC30890 RG7713 (RO5028442) A vasopressin V1a receptor antagonist
  18. GC30764 Argipressin (Vasopressin) Argipressin (Vasopressin) (Arg8-vasopressin) 与 V1、V2、V3-血管精氨酸加压素受体结合，在 A7r5 大鼠主动脉平滑肌细胞中对 V1 的 Kd 值为 1.31 nM。
  19. GC10622 OPC 21268 A nonpeptide antagonist of vasopressin V1 receptors
  20. GC15154 d[Leu4,Lys8]-VP D[LEU4,LYS8]-VP 是血管加压素 V1b 受体的选择性激动剂，对大鼠、人和小鼠 V1b 受体的 Kis 值分别为 0.16 nM、0.52 nM 和 0.1.38 nM。
  21. GC16591 d[Cha4]-AVP d[Cha4]-AVP 是一种有效的选择性加压素 (AVP) V1b 受体激动剂，对人 V1b 受体的 Ki 值为 1.2 nM。
  22. GC11991 L-371,257 L-371,257 是一种口服生物可利用的、非血脑屏障渗透剂、选择性和竞争性催产素受体 (pA2=8.4) 拮抗剂，对催产素受体 (Ki=19 nM) 和加压素 V1a 受体 (Ki=3.7) 具有高亲和力nM)。
  23. GC12462 SR 49059 A vasopressin receptor V1a antagonist
  24. GC12194 Atosiban An oxytocin receptor antagonist
  25. GC14880 Mozavaptan Mozavaptan (OPC-31260) 是一种苯并氮杂类衍生物，是一种有效的、选择性的、竞争性的、具有口服活性的加压素 V2 受体拮抗剂，IC50 为 14 nM。
  26. GC15575 Tolvaptan A vasopressin V2 receptor antagonist
  27. GC12627 Conivaptan HCl A vasopressin V1A and V2 receptor antagonist
  28. GC11265 Desmopressin Acetate 精氨酸加压素的合成类似物
  29. GC12303 Desmopressin A vasopressin receptor agonist

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