GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(482)
- Acetylcholine(28)
- Adenosine Deaminase(9)
- Adenosine Receptor(130)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(407)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(111)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(118)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(80)
- Chemokine Receptors(23)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(77)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(96)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(12)
- LPL Receptor(59)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(54)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(23)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(47)
- Oxytocin Receptors(22)
- P2Y Receptor(60)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(170)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(58)
- Vasopressin Receptor(33)
- 17,20-lyase(4)
- Ras(138)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(183)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(26)
- GRK(1)
- GCGR(2)
- GLP Receptor(2)
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
- Cat.No. 产品名称 Information
-
GC15023
Telmisattan
替米沙坦; BIBR 277
Selective angiotensin II receptor antagonist -
GC11819
Strontium Ranelate
雷尼酸锶; Distrontium renelate; S12911
An antiosteoporotic agent -
GC15719
Silodosin
西洛多辛; KAD 3213; KMD 3213
A potent α1A-adrenoceptor antagonist -
GC10460
Rizatriptan Benzoate
苯甲酸利扎曲坦,MK 462
A 5-HT1B and 5-HT1D receptor agonist -
GC12986
Risperidone
利培酮; R 64 766
An atypical antipsychotic -
GC14113
Oxybutynin
奥昔布宁
An antagonist of muscarinic acetylcholine receptors -
GC17498
L-Glutamine
L-谷氨酰胺; L-Glutamic acid 5-amide
A conditionally essential amino acid -
GC11590
Istradefylline(KW-6002)
伊曲茶碱; KW-6002
Istradefylline(KW-6002)是一种腺苷A2A受体拮抗剂。Istradefylline通过选择性拮抗腺苷A2A受体并调节基底神经节的间接通路来改善帕金森病患者的运动功能障碍。Istradefylline主要用于治疗帕金森病。 -
GC11434
GSK1292263
An agonist of GPR119
-
GC16526
Atropine
阿托品; Tropine tropate; DL-Hyoscyamine
A non-selective muscarinic acetylcholine receptor antagonist -
GC16555
TAK-875
TAK 875;TAK875
A selective FFAR1 (GPR40) agonist -
GC15090
Maraviroc
马拉维若,UK-427857; Selzentry; Celsentri
马拉韦罗作为第一款CCR5拮抗剂已被批准用于治疗HIV感染,对hERG离子通道的IC50>10μM。
-
GC12470
ZCL278
A selective Cdc42 inhibitor
-
GC16788
PRX-08066 Maleic acid
5-HT2B receptor antagonist,potent and selective
-
GC14437
Vortioxetine (Lu AA21004) HBr
盐酸沃替西汀; Lu AA21004 hydrobromide
A multimodal serotonergic agent -
GC17785
Macitentan
马西替坦; ACT-064992
A dual ETA/ETB receptor antagonist -
GC16150
VU 0364439
N-[3-氯-4-[[(2-氯苯基)氨基]磺酰基]苯基]-2-吡啶甲酰胺
A positive allosteric modulator of mGluR4 -
GC14745
Plerixafor (AMD3100)
普乐沙福; AMD 3100; JM3100; SID791
Plerixafor(AMD3100) 是 CXCR4 和 CXCL12 介导的趋化作用的小分子抑制剂,IC50 值分别为 44 nM 和 5.7 nM 。 -
GC12401
GW9508
An agonist of GPR40
-
GC10069
NSC 23766 trihydrochloride
Inhibitor of Rac1
-
GC17205
CP-945598 HCl
CP 945598 Hydrochloride
A selective CB1 receptor antagonist -
GC10467
Irbesartan
厄贝沙坦; SR-47436; BMS-186295
An AT1 receptor antagonist
-
GC15414
AM1241
A CB2 receptor agonist and inverse agonist
-
GC16862
Zibotentan (ZD4054)
齐泊腾坦,ZD4054
A selective ETA receptor antagonist -
GC15463
Iloperidone
伊潘立酮; HP 873
An atypical antipsychotic -
GC11521
Ziprasidone HCl
盐酸齐拉西酮; CP-88059 hydrochloride
An atypical antipsychotic -
GC18006
Sumatriptan Succinate
舒马普坦琥珀酸盐; GR 43175
An agonist of 5-HT1B and 5-HT1D receptors -
GC15964
Clopidogrel hydrogen sulfate
硫酸氢氯吡格雷; (S)-(+)-Clopidogrel bisulfate; (S)-(+)-Clopidogrel hydrogen sulfate
A prodrug form of a P2Y12 antagonist -
GC10121
Tianeptine sodium
噻奈普汀钠
An atypical antidepressant -
GC13730
Alfuzosin HCl
盐酸阿夫唑嗪; SL 77499-10
α1-Adrenergic receptor antagonist -
GC10911
Venlafaxine hydrochloride
盐酸文拉法辛; Wy 45030 hydrochloride
An Analytical Reference Material -
GC13389
Tranilast
曲尼司特; MK-341; SB 252218
An antiallergic agent -
GC16978
Candesartan
坎地沙坦; CV 11974
An AT1 receptor antagonist -
GC18072
Prazosin HCl
哌唑嗪盐酸盐
An α1-adrenergic receptor antagonist -
GC11814
Ondansetron HCl
盐酸昂丹司琼; GR 38032 hydrochloride; SN 307 hydrochloride
A Certified Reference Material -
GC11374
Ki16425
Debio 0719
Ki16425是溶血磷脂酸受体 LPA1 和 LPA3 的拮抗剂,Ki 值分别为 0.25 和 0.36μM。Ki16425 可降低 LPA 诱导的 p42/p44 MAPK 的活化,阻断 LPA 诱导的是相关蛋白(YAP)和含 WW 结构域的转录调节蛋白 1(TAZ)的去磷酸化,从而抑制 Hippo 信号通路。 -
GC15200
Aprepitant
阿瑞匹坦; MK-0869; MK-869; L-754030
An antiemetic and NK1 antagonist -
GC15053
Ramelteon
雷美替胺; TAK-375
A melatonin receptor agonist -
GC10509
Cladribine
克拉屈滨; 2-Chloro-2′-deoxyadenosine; CldAdo; 2CdA
A nucleoside analog and prodrug form of 2-CdATP -
GC17464
Prasugrel
普拉格雷; PCR 4099
A prodrug form of R-99224 -
GC15025
Fluvoxamine maleate
氟伏沙明马来酸盐; DU-23000 maleate
A selective serotonin reuptake inhibitor -
GC11709
Fluoxetine HCl
盐酸氟西汀; LY 110140
An Analytical Reference Material -
GC10257
Losartan Potassium (DuP 753)
氯沙坦钾; DuP-753 potassium
A potent, synthetic AT1 receptor antagonist -
GC13443
Doxazosin Mesylate
甲磺酸多沙唑嗪; UK 33274 mesylate
An α1-AR antagonist -
GC11824
Asenapine
阿塞那平; Org 5222
An atypical antipsychotic -
GC15618
Melatonin
褪黑素; N-Acetyl-5-methoxytryptamine
An indoleamine neurohormone that entrains circadian rhythms
-
GC17779
Levetiracetam
左乙拉西坦; UCB L059
An antiepileptic compound -
GC17536
Mosapride Citrate
莫沙必利柠檬酸盐; TAK-370 citrate; AS-4370 citrate
A 5-HT4 receptor agonist -
GC16029
Granisetron HCl
盐酸格拉司琼; BRL 43694A
A 5-HT3 receptor antagonist with antiemetic activity -
GC14860
Oncrasin 1
1-(4-氯苄基)-1H-吲哚-3-甲醛
An anticancer agent