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Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

  1. Cat.No. 产品名称 Information
  2. GC15023 Telmisattan

    替米沙坦; BIBR 277

     Selective angiotensin II receptor antagonist
  3. GC11819 Strontium Ranelate

    雷尼酸锶; Distrontium renelate; S12911

     An antiosteoporotic agent
  4. GC15719 Silodosin

    西洛多辛; KAD 3213; KMD 3213

     A potent α1A-adrenoceptor antagonist
  5. GC10460 Rizatriptan Benzoate

    苯甲酸利扎曲坦,MK 462

     A 5-HT1B and 5-HT1D receptor agonist
  6. GC12986 Risperidone

    利培酮; R 64 766

     An atypical antipsychotic
  7. GC14113 Oxybutynin

    奥昔布宁

     An antagonist of muscarinic acetylcholine receptors
  8. GC17498 L-Glutamine

    L-谷氨酰胺; L-Glutamic acid 5-amide

     A conditionally essential amino acid
  9. GC11590 Istradefylline(KW-6002)

    伊曲茶碱; KW-6002

     Istradefylline(KW-6002)是一种腺苷A2A受体拮抗剂。Istradefylline通过选择性拮抗腺苷A2A受体并调节基底神经节的间接通路来改善帕金森病患者的运动功能障碍。Istradefylline主要用于治疗帕金森病。
  10. GC11434 GSK1292263 An agonist of GPR119
  11. GC16526 Atropine

    阿托品; Tropine tropate; DL-Hyoscyamine

     A non-selective muscarinic acetylcholine receptor antagonist
  12. GC16555 TAK-875

    TAK 875;TAK875

     A selective FFAR1 (GPR40) agonist
  13. GC15090 Maraviroc

    马拉维若,UK-427857; Selzentry; Celsentri

    马拉韦罗作为第一款CCR5拮抗剂已被批准用于治疗HIV感染，对hERG离子通道的IC50＞10μM。
  14. GC12470 ZCL278 A selective Cdc42 inhibitor
  15. GC16788 PRX-08066 Maleic acid 5-HT2B receptor antagonist,potent and selective
  16. GC14437 Vortioxetine (Lu AA21004) HBr

    盐酸沃替西汀; Lu AA21004 hydrobromide

     A multimodal serotonergic agent
  17. GC17785 Macitentan

    马西替坦; ACT-064992

     A dual ETA/ETB receptor antagonist
  18. GC16150 VU 0364439

    N-[3-氯-4-[[(2-氯苯基)氨基]磺酰基]苯基]-2-吡啶甲酰胺

     A positive allosteric modulator of mGluR4
  19. GC14745 Plerixafor (AMD3100)

    普乐沙福; AMD 3100; JM3100; SID791

     Plerixafor(AMD3100) 是 CXCR4 和 CXCL12 介导的趋化作用的小分子抑制剂，IC50 值分别为 44 nM 和 5.7 nM 。
  20. GC12401 GW9508 An agonist of GPR40
  21. GC10069 NSC 23766 trihydrochloride Inhibitor of Rac1
  22. GC17205 CP-945598 HCl

    CP 945598 Hydrochloride

     A selective CB1 receptor antagonist
  23. GC10467 Irbesartan

    厄贝沙坦; SR-47436; BMS-186295

    An AT1 receptor antagonist
  24. GC15414 AM1241 A CB2 receptor agonist and inverse agonist
  25. GC16862 Zibotentan (ZD4054)

    齐泊腾坦,ZD4054

     A selective ETA receptor antagonist
  26. GC15463 Iloperidone

    伊潘立酮; HP 873

     An atypical antipsychotic
  27. GC11521 Ziprasidone HCl

    盐酸齐拉西酮; CP-88059 hydrochloride

     An atypical antipsychotic
  28. GC18006 Sumatriptan Succinate

    舒马普坦琥珀酸盐; GR 43175

     An agonist of 5-HT1B and 5-HT1D receptors
  29. GC15964 Clopidogrel hydrogen sulfate

    硫酸氢氯吡格雷; (S)-(+)-Clopidogrel bisulfate; (S)-(+)-Clopidogrel hydrogen sulfate

     A prodrug form of a P2Y12 antagonist
  30. GC10121 Tianeptine sodium

    噻奈普汀钠

     An atypical antidepressant
  31. GC13730 Alfuzosin HCl

    盐酸阿夫唑嗪; SL 77499-10

     α1-Adrenergic receptor antagonist
  32. GC10911 Venlafaxine hydrochloride

    盐酸文拉法辛; Wy 45030 hydrochloride

     An Analytical Reference Material
  33. GC13389 Tranilast

    曲尼司特; MK-341; SB 252218

     An antiallergic agent
  34. GC16978 Candesartan

    坎地沙坦; CV 11974

     An AT1 receptor antagonist
  35. GC18072 Prazosin HCl

    哌唑嗪盐酸盐

     An α1-adrenergic receptor antagonist
  36. GC11814 Ondansetron HCl

    盐酸昂丹司琼; GR 38032 hydrochloride; SN 307 hydrochloride

     A Certified Reference Material
  37. GC11374 Ki16425

    Debio 0719

     Ki16425是溶血磷脂酸受体 LPA1 和 LPA3 的拮抗剂，Ki 值分别为 0.25 和 0.36μM。Ki16425 可降低 LPA 诱导的 p42/p44 MAPK 的活化，阻断 LPA 诱导的是相关蛋白（YAP）和含 WW 结构域的转录调节蛋白 1（TAZ）的去磷酸化，从而抑制 Hippo 信号通路。
  38. GC15200 Aprepitant

    阿瑞匹坦; MK-0869; MK-869; L-754030

     An antiemetic and NK1 antagonist
  39. GC15053 Ramelteon

    雷美替胺; TAK-375

     A melatonin receptor agonist
  40. GC10509 Cladribine

    克拉屈滨; 2-Chloro-2′-deoxyadenosine; CldAdo; 2CdA

     A nucleoside analog and prodrug form of 2-CdATP
  41. GC17464 Prasugrel

    普拉格雷; PCR 4099

     A prodrug form of R-99224
  42. GC15025 Fluvoxamine maleate

    氟伏沙明马来酸盐; DU-23000 maleate

     A selective serotonin reuptake inhibitor
  43. GC11709 Fluoxetine HCl

    盐酸氟西汀; LY 110140

     An Analytical Reference Material
  44. GC10257 Losartan Potassium (DuP 753)

    氯沙坦钾; DuP-753 potassium

     A potent, synthetic AT1 receptor antagonist
  45. GC13443 Doxazosin Mesylate

    甲磺酸多沙唑嗪; UK 33274 mesylate

     An α1-AR antagonist
  46. GC11824 Asenapine

    阿塞那平; Org 5222

     An atypical antipsychotic
  47. GC15618 Melatonin

    褪黑素; N-Acetyl-5-methoxytryptamine

    An indoleamine neurohormone that entrains circadian rhythms
  48. GC17779 Levetiracetam

    左乙拉西坦; UCB L059

     An antiepileptic compound
  49. GC17536 Mosapride Citrate

    莫沙必利柠檬酸盐; TAK-370 citrate; AS-4370 citrate

     A 5-HT4 receptor agonist
  50. GC16029 Granisetron HCl

    盐酸格拉司琼; BRL 43694A

     A 5-HT3 receptor antagonist with antiemetic activity
  51. GC14860 Oncrasin 1

    1-(4-氯苄基)-1H-吲哚-3-甲醛

     An anticancer agent

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