GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(482)
- Acetylcholine(28)
- Adenosine Deaminase(9)
- Adenosine Receptor(130)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(407)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(111)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(118)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(80)
- Chemokine Receptors(23)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(77)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(96)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(12)
- LPL Receptor(59)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(54)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(23)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(47)
- Oxytocin Receptors(22)
- P2Y Receptor(60)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(170)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(58)
- Vasopressin Receptor(33)
- 17,20-lyase(4)
- Ras(138)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(183)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(26)
- GRK(1)
- GCGR(2)
- GLP Receptor(2)
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
- Cat.No. 产品名称 Information
-
GC13000
Acebutolol HCl
盐酸醋丁洛尔;盐酸醋丁酰心安
A β1-AR antagonist -
GC11551
Hydrocortisone
氢化可的松; Cortisol
氢化可的松是一种由肾上腺和肾上腺外组织分泌的天然糖皮质激素,通过与其同源糖皮质激素受体 (GR) 结合,局部控制参与炎症、免疫反应、新陈代谢和能量稳态的基因的转录 。 -
GC14703
Oxybutynin chloride
盐酸奥昔布宁
An antagonist of muscarinic acetylcholine receptors -
GC15690
Desonide
地索奈德
A nonfluorinated synthetic corticosteroid -
GC15668
Meprednisone
泼尼松
A corticosteroid -
GC17808
Zolmitriptan
佐米曲普坦,BW-311C90; 311C90
An agonist of 5-HT1B and 5-HT1D receptors -
GC16401
L-(-)-α-Methyldopa hydrochloride
L-3-(3,4-二羟基苯基)-2-甲基丙氨酸盐酸盐,L-(-)-α-Methyldopa hydrochloride; MK-351 hydrochloride
A DOPA decarboxylase inhibitor -
GC16490
Methyldopa
甲基多巴; L-(-)-α-Methyldopa; MK-351
A DOPA decarboxylase inhibitor -
GC16450
Prednisone
强的松; Dehydrocortisone
A synthetic glucocorticoid
-
GC13906
Nebivolol hydrochloride
盐酸奈必洛尔; R 065824 hydrochloride
A β1-AR antagonist -
GC11959
Naratriptan
盐酸那拉曲坦,GR-85548A
A potent 5-HT1B and 5-HT1D receptor agonist -
GC12443
Tranilast Sodium
曲尼司特钠; MK-341 sodium; SB 252218 sodium
An antiallergic agent -
GC17891
Tizanidine HCl
盐酸替扎尼定
An α2-adrenergic receptor agonist -
GC15629
Tizanidine
替扎尼定
An α2-adrenergic receptor agonist -
GC16785
Prazosin
哌唑嗪
哌唑嗪是一种 α-肾上腺素能阻滞剂,是一种用于治疗高血压和焦虑症、创伤后应激障碍和恐慌症的交感神经药物。 -
GC16740
Alfuzosin
阿夫唑嗪; SL 77499
Alfuzosin (SL 77499-10) 是一种具有口服活性、选择性和竞争性的 α1-肾上腺素受体拮抗剂。 -
GC12687
Bimatoprost
比马前列素; AGN 192024
The ocular hypotensive ingredient in Lumigan -
GC13428
Mosapride
莫沙必利; TAK-370; AS-4370
A 5-HT4 receptor agonist -
GC17081
Detomidine HCl
盐酸地托咪定
An α2-adrenoceptor agonist -
GC17197
Detomidine
地托咪定
Detomidine 是一种咪唑衍生物,是一种有效的 α2-肾上腺素能激动剂。 -
GC10194
Ivabradine HCl
盐酸伊伐布雷定
An HCN channel blocker -
GC13371
Fluticasone propionate
丙酸氟替卡松
A synthetic corticosteroid and glucocorticoid receptor agonist -
GC16496
Ticlopidine
盐酸噻氯匹定,PCR 5332
A P2Y12 receptor antagonist with antiplatelet activity -
GC12920
Pregnenolone
孕烯醇酮; 3β-Hydroxy-5-pregnen-20-one
A natural steroid hormone -
GC17347
Alprostadil
前列地尔; Alprostadil; PGE1;Prostaglandin E1
前列地尔Alprostadil作为前列腺素受体配体,对小鼠EP3、EP4、EP2、IP和EP1的结合亲和Kis分别为1.1 nM、2.1 nM、10 nM、33 nM和36 nM。 -
GC16871
Perindopril
培哚普利; S-9490
An orally active ACE inhibitor -
GC13478
Pizotifen Malate
苯噻啶苹果酸盐,Pizotyline malate; BC-105 malate
A triptan -
GC13053
Pizotifen
苯噻啶; Pizotyline; BC-105
A triptan -
GC13092
Fluvoxamine
氟伏沙明; DU-23000
A selective serotonin reuptake inhibitor -
GC13447
Doxazosin
多沙唑嗪; UK 33274
An α1-AR antagonist -
GC17593
Lurasidone HCl
盐酸鲁拉西酮; SM-13496 Hydrochloride
An atypical antipsychotic -
GC16891
Quetiapine Fumarate
富马酸喹硫平
An antagonist of diverse neurological receptors -
GC15223
Tropisetron Hydrochloride
盐酸托烷司琼
A 5-HT3 receptor antagonist -
GC15918
Formoterol Hemifumarate
富马酸福莫特罗,(±)Formoterol fumarate
强效、选择性和长效 β2-肾上腺素能受体激动剂 -
GC14769
Carvedilol
卡维地洛; BM 14190
A β-adrenergic receptor antagonist -
GC11651
Ondansetron hydrochloride dihydrate
盐酸昂丹司琼二水物; GR 38032 hydrochloride dihydrate; SN 307 hydrochloride dihydrate
An Analytical Reference Material -
GC16087
Fesoterodine Fumarate
富马酸非索罗定
A muscarinic acetylcholine receptor antagonist -
GC14512
Fenspiride HCl
盐酸芬司必利
A histamine H1 receptor antagonist -
GC11219
(R)-(+)-Tolterodine
托特罗定; (R)-(+)-Tolterodine; (+)-Tolterodine; (R)-Tolterodine; PNU-200583
(R)-(+)-Tolterodine(PNU-200583) 是一种有效的毒蕈碱受体拮抗剂,在体内对膀胱的选择性优于唾液腺。 -
GC17917
Palonosetron HCl
盐酸帕洛诺司琼
A 5-HT3 receptor antagonist -
GC11465
Bosentan Hydrate
波生坦水合物
An antagonist of endothelin receptors -
GC16269
Bosentan
波生坦
An antagonist of endothelin receptors -
GC15772
Darifenacin HBr
氢溴酸达非那新; UK-88525 hydrobromide
A muscarinic M3 receptor antagonist -
GC17053
Eletriptan HBr
依来曲普坦氢溴酸盐; Eletriptan HBr; UK-116044 hydrobromide
An agonist of 5-HT1B and 5-HT1D receptors -
GC17182
Solifenacin succinate
索非那新琥珀酸盐; YM905
A muscarinic M1, M2, and M3 receptor antagonist -
GC17954
Tolterodine tartrate
酒石酸托特罗定,Kabi-2234; PNU-200583E
A muscarinic acetylcholine receptor antagonist -
GC15317
SB408124
A potent orexin 1 receptor antagonist
-
GC16708
Cinacalcet HCl
盐酸西那卡塞; AMG-073 hydrochloride
An allosteric agonist of the CaSR -
GC17949
Plerixafor 8HCl (AMD3100 8HCl)
盐酸普乐沙福; AMD3100 octahydrochloride; JM3100 octahydrochloride; SID791 octahydrochloride
An antagonist of CXCR4 -
GC11182
LY404039
(1R,4S,5S,6S)-4-氨基-2-硫杂双环[3.1.0]己烷-4,6-二甲酸2,2-二氧化物
An agonist of mGluR2 and mGluR3