Home >> Signaling Pathways >> GPCR/G protein

GPCR/G protein(G 蛋白偶联受体/G 蛋白)

  1. Cat.No. 产品名称 Information
  2. GC13000 Acebutolol HCl

    盐酸醋丁洛尔;盐酸醋丁酰心安

    A β1-AR antagonist
  3. GC11551 Hydrocortisone

    氢化可的松; Cortisol

    氢化可的松是一种由肾上腺和肾上腺外组织分泌的天然糖皮质激素,通过与其同源糖皮质激素受体 (GR) 结合,局部控制参与炎症、免疫反应、新陈代谢和能量稳态的基因的转录 。
  4. GC14703 Oxybutynin chloride

    盐酸奥昔布宁

    An antagonist of muscarinic acetylcholine receptors
  5. GC15690 Desonide

    地索奈德

    A nonfluorinated synthetic corticosteroid
  6. GC15668 Meprednisone

    泼尼松

    A corticosteroid
  7. GC17808 Zolmitriptan

    佐米曲普坦,BW-311C90; 311C90

    An agonist of 5-HT1B and 5-HT1D receptors
  8. GC16401 L-(-)-α-Methyldopa hydrochloride

    L-3-(3,4-二羟基苯基)-2-甲基丙氨酸盐酸盐,L-(-)-α-Methyldopa hydrochloride; MK-351 hydrochloride

    A DOPA decarboxylase inhibitor
  9. GC16490 Methyldopa

    甲基多巴; L-(-)-α-Methyldopa; MK-351

    A DOPA decarboxylase inhibitor
  10. GC16450 Prednisone

    强的松; Dehydrocortisone

    A synthetic glucocorticoid

  11. GC13906 Nebivolol hydrochloride

    盐酸奈必洛尔; R 065824 hydrochloride

    A β1-AR antagonist
  12. GC11959 Naratriptan

    盐酸那拉曲坦,GR-85548A

    A potent 5-HT1B and 5-HT1D receptor agonist
  13. GC12443 Tranilast Sodium

    曲尼司特钠; MK-341 sodium; SB 252218 sodium

    An antiallergic agent
  14. GC17891 Tizanidine HCl

    盐酸替扎尼定

    An α2-adrenergic receptor agonist
  15. GC15629 Tizanidine

    替扎尼定

    An α2-adrenergic receptor agonist
  16. GC16785 Prazosin

    哌唑嗪

    哌唑嗪是一种 α-肾上腺素能阻滞剂,是一种用于治疗高血压和焦虑症、创伤后应激障碍和恐慌症的交感神经药物。
  17. GC16740 Alfuzosin

    阿夫唑嗪; SL 77499

    Alfuzosin (SL 77499-10) 是一种具有口服活性、选择性和竞争性的 α1-肾上腺素受体拮抗剂。
  18. GC12687 Bimatoprost

    比马前列素; AGN 192024

    The ocular hypotensive ingredient in Lumigan
  19. GC13428 Mosapride

    莫沙必利; TAK-370; AS-4370

    A 5-HT4 receptor agonist
  20. GC17081 Detomidine HCl

    盐酸地托咪定

    An α2-adrenoceptor agonist
  21. GC17197 Detomidine

    地托咪定

    Detomidine 是一种咪唑衍生物,是一种有效的 α2-肾上腺素能激动剂。
  22. GC10194 Ivabradine HCl

    盐酸伊伐布雷定

    An HCN channel blocker
  23. GC13371 Fluticasone propionate

    丙酸氟替卡松

    A synthetic corticosteroid and glucocorticoid receptor agonist
  24. GC16496 Ticlopidine

    盐酸噻氯匹定,PCR 5332

    A P2Y12 receptor antagonist with antiplatelet activity
  25. GC12920 Pregnenolone

    孕烯醇酮; 3β-Hydroxy-5-pregnen-20-one

    A natural steroid hormone
  26. GC17347 Alprostadil

    前列地尔; Alprostadil; PGE1;Prostaglandin E1

    前列地尔Alprostadil作为前列腺素受体配体,对小鼠EP3、EP4、EP2、IP和EP1的结合亲和Kis分别为1.1 nM、2.1 nM、10 nM、33 nM和36 nM。
  27. GC16871 Perindopril

    培哚普利; S-9490

    An orally active ACE inhibitor
  28. GC13478 Pizotifen Malate

    苯噻啶苹果酸盐,Pizotyline malate; BC-105 malate

    A triptan
  29. GC13053 Pizotifen

    苯噻啶; Pizotyline; BC-105

    A triptan
  30. GC13092 Fluvoxamine

    氟伏沙明; DU-23000

    A selective serotonin reuptake inhibitor
  31. GC13447 Doxazosin

    多沙唑嗪; UK 33274

    An α1-AR antagonist
  32. GC17593 Lurasidone HCl

    盐酸鲁拉西酮; SM-13496 Hydrochloride

    An atypical antipsychotic
  33. GC16891 Quetiapine Fumarate

    富马酸喹硫平

    An antagonist of diverse neurological receptors
  34. GC15223 Tropisetron Hydrochloride

    盐酸托烷司琼

    A 5-HT3 receptor antagonist
  35. GC15918 Formoterol Hemifumarate

    富马酸福莫特罗,(±)Formoterol fumarate

    强效、选择性和长效 β2-肾上腺素能受体激动剂
  36. GC14769 Carvedilol

    卡维地洛; BM 14190

    A β-adrenergic receptor antagonist
  37. GC11651 Ondansetron hydrochloride dihydrate

    盐酸昂丹司琼二水物; GR 38032 hydrochloride dihydrate; SN 307 hydrochloride dihydrate

    An Analytical Reference Material
  38. GC16087 Fesoterodine Fumarate

    富马酸非索罗定

    A muscarinic acetylcholine receptor antagonist
  39. GC14512 Fenspiride HCl

    盐酸芬司必利

    A histamine H1 receptor antagonist
  40. GC11219 (R)-(+)-Tolterodine

    托特罗定; (R)-(+)-Tolterodine; (+)-Tolterodine; (R)-Tolterodine; PNU-200583

    (R)-(+)-Tolterodine(PNU-200583) 是一种有效的毒蕈碱受体拮抗剂,在体内对膀胱的选择性优于唾液腺。
  41. GC17917 Palonosetron HCl

    盐酸帕洛诺司琼

    A 5-HT3 receptor antagonist
  42. GC11465 Bosentan Hydrate

    波生坦水合物

    An antagonist of endothelin receptors
  43. GC16269 Bosentan

    波生坦

    An antagonist of endothelin receptors
  44. GC15772 Darifenacin HBr

    氢溴酸达非那新; UK-88525 hydrobromide

    A muscarinic M3 receptor antagonist
  45. GC17053 Eletriptan HBr

    依来曲普坦氢溴酸盐; Eletriptan HBr; UK-116044 hydrobromide

    An agonist of 5-HT1B and 5-HT1D receptors
  46. GC17182 Solifenacin succinate

    索非那新琥珀酸盐; YM905

    A muscarinic M1, M2, and M3 receptor antagonist
  47. GC17954 Tolterodine tartrate

    酒石酸托特罗定,Kabi-2234; PNU-200583E

    A muscarinic acetylcholine receptor antagonist
  48. GC15317 SB408124 A potent orexin 1 receptor antagonist
  49. GC16708 Cinacalcet HCl

    盐酸西那卡塞; AMG-073 hydrochloride

    An allosteric agonist of the CaSR
  50. GC17949 Plerixafor 8HCl (AMD3100 8HCl)

    盐酸普乐沙福; AMD3100 octahydrochloride; JM3100 octahydrochloride; SID791 octahydrochloride

    An antagonist of CXCR4
  51. GC11182 LY404039

    (1R,4S,5S,6S)-4-氨基-2-硫杂双环[3.1.0]己烷-4,6-二甲酸2,2-二氧化物

    An agonist of mGluR2 and mGluR3

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