GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(482)
- Acetylcholine(28)
- Adenosine Deaminase(9)
- Adenosine Receptor(130)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(407)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(111)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(118)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(80)
- Chemokine Receptors(23)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(77)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(96)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(12)
- LPL Receptor(59)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(54)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(23)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(47)
- Oxytocin Receptors(22)
- P2Y Receptor(60)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(170)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(58)
- Vasopressin Receptor(33)
- 17,20-lyase(4)
- Ras(138)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(183)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(26)
- GRK(1)
- GCGR(2)
- GLP Receptor(2)
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
- Cat.No. 产品名称 Information
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GC15926
BAN ORL 24
(2R)-1-苄基-N-(3-螺[异苯并呋喃-1(3H),4'-哌啶]-1'-丙基)-2-吡咯烷甲酰胺,BAN-ORL-24;BAN ORL-24
A nociceptin receptor antagonist
-
GC11405
Avosentan
N-[6-甲氧基-5-(2-甲氧基苯氧基)-2-(4-吡啶基)-4-嘧啶基]-5-甲基吡啶-2-磺酰胺,Ro 67-0565; SPP-301
Avosentan (Ro 67-0565; SPP-301) 是一种有效的选择性内皮素受体 (ETA 受体) 拮抗剂。
-
GC11783
Atrasentan hydrochloride
盐酸阿曲生坦; ABT-627 hydrochloride; (+)-A 127722 hydrochloride; A-147627 hydrochloride
Atrasentan hydrochloride (ABT-627 hydrochloride) 是一种选择性内皮素 A 受体拮抗剂，对 ETA 的 IC50 为 0.0551 nM。
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GC14518
Asenapine hydrochloride
阿塞那平盐酸盐
Asenapine hydrochloride 是一种抗精神病药，是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂，Ki 值为 0.03-4.0 nM，作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。
-
GC13253
Anamorelin
阿拉莫林,RC-1291;ONO-7643;RC1291;ONO7643;RC 1291;ONO 7643
A small molecule agonist of GHS-R1a
-
GC17018
AMD-070 hydrochloride
N-(1H-苯并咪唑-2-基甲基)-N-[(8S)-5,6,7,8-四氢-8-喹啉基]-1,4-丁二胺单盐酸盐,AMD070 hydrochloride;AMD 070 hydrochloride
CXCR4 antagonist,potent and selective
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GC12196
AMD-070
N'-(1H-苯并咪唑-2-甲基)-N'-((S)-5,6,7,8-四氢喹啉-8-基)丁烷-1,4-二胺,AMD 070; AMD070
A CXCR4 antagonist
-
GC13476
AM966
4'-[4-[[[(1R)-1-(2-氯苯基)乙氧基]羰基]氨基]-3-甲基-5-异恶唑基]-联苯-4-乙酸,AM 966;AM-966
A potent and selective LPA1 receptor antagonist
-
GC10147
AM630
[6-碘-2-甲基-1-[2-(4-吗啉基)乙基]-1H-吲哚-3-基](4-甲氧基苯基)甲酮,AM 630;AM-630
An inverse agonist at CB2 and partial agonist at CB1 receptors
-
GC15908
AM-095 free base
[4'-[3-甲基-4-[[[((R)-1-苯基乙基)氧基]羰基]氨基]异恶唑-5-基]联苯-4-基]乙酸,AM 095;AM095
A selective LPA1 receptor antagonist
-
GC15220
AM095
4'-[3-甲基-4-[[[(1R)-1-苯基乙氧基]羰基]氨基]-5-异恶唑基]联苯-4-乙酸钠盐,AM 095;AM-095
A selective LPA1 receptor antagonist
-
GC11166
Alosetron Hydrochloride
盐酸阿洛司琼,GR 68755C;GR 68755;GR 68755X;Lotronex;GR-68755;GR68755
A 5-HT3 receptor antagonist
-
GC13654
Alosetron
阿洛司琼; GR 68755; GR 68755X
A 5-HT3 receptor antagonist
-
GC14879
AH 6809
6-异丙氧基-9-氧代氧杂蒽-2-羧酸,AH6809;AH-6809
An EP and DP receptor antagonist
-
GC14801
5-Iodotubercidin
5-碘代杀结核菌素,NSC 113939; 5-ITu
An adenosine kinase inhibitor
-
GC14145
(R,R)-Formoterol
(-)-Formoterol;Arformoterol;Formoterol
β2-selective adrenergic agonist
-
GC13652
Dyphylline
二羟丙茶碱; Diprophylline
An adenosine receptor antagonist and phosphodiesterase inhibitor
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GC15505
Methylprednisolone
甲泼尼龙; U 7532
甲泼尼龙是皮质类固醇,可作用于糖皮质激素受体并抑制皮质醇分泌,其IC50为1.7ng/ml。
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GC16752
Olmesartan medoxomil
奥美沙坦酯; CS 866
A prodrug form of olmesartan
-
GN10542
Scopolamine butylbromide
丁溴东莨菪碱,Hyoscine butylbromide; (-)-Scopolamine butylbromide; Butylscopolamine bromide
An antispasmodic agent
-
GN10074
Xanthotoxol
花椒毒醇,8-Hydroxypsoralen
A coumarin with diverse biological activities
-
GN10507
Baohuoside I
宝藿苷 I; Icariin-II; Icariside-II
宝活苷 I 是一种从淫羊藿中分离出来的黄酮类化合物，可作为 CXCR4 抑制剂，下调 CXCR4 表达，诱导细胞凋亡并具有抗肿瘤活性。
-
GN10652
Norisoboldine
去甲异波尔定,(+)-Laurelliptine
Norisoboldine 是一种具有口服活性的天然芳烃受体 (AhR) 激动剂。
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GN10419
Ligustroflavone
女贞苷; Nuezhenoside
An apigenin triglycoside with diverse biological activities
-
GN10104
Gramine
芦竹碱,Donaxine
An Analytical Reference Standard
-
GN10186
Isocorynoxeine
异去氢钩藤碱; 7-Isocorynoxeine
An alkaloid with diverse biological activities
-
GN10606
Yohimbine Hydrochloride
盐酸育亨宾；育酚；育亨宾盐酸盐；柯楠质盐酸盐；萝芙根 (皮) 碱盐酸盐；盐酸萝芙根 (皮) 碱
An α2-adrenoceptor antagonist
-
GN10489
Hyodeoxycholic acid
猪去氧胆酸; HDCA
A secondary bile acid
-
GN10112
Ginsenoside Rb2
人参皂苷 Rb2; Ginsenoside C
A natural steroid glycoside with diverse effects
-
GN10607
Nuciferine
荷叶碱
An alkaloid with diverse biological activities
-
GN10285
Theobromine
可可碱; 3,7-Dimethylxanthine
A methylxanthine alkaloid with diverse biological activities
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GN10659
Theophylline
茶碱,Theolix
A phosphodiesterase inhibitor and adenosine receptor antagonist
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GN10069
Ginsenoside Ro
人参皂苷 Ro; Polysciasaponin P3; Chikusetsusaponin 5; Chikusetsusaponin V
A non-steroid glycoside with diverse biological activities
-
GN10169
3-Hydroxy-4-methoxycinnamic acid
3-羟基-4-甲氧基肉桂酸,3-Hydroxy-4-methoxycinnamic acid
A cinnamic acid derivative
-
GN10680
Puerarin
葛根素
A natural isoflavonoid
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GP10110
Angiotensin III (human, mouse)
血管紧张素III,Arg-Val-Tyr-Ile-His-Pro-Phe
An agonist at AT1 and AT2 receptors
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GP10077
Angiotensin (1-7)
Asp-Arg-Val-Tyr-Ile-His-Pro
血管紧张素 1-7 (Ang-(1-7)) 是来自肾素-血管紧张素系统 (RAS) 的内源性七肽，由于其在心脏细胞中的抗炎和抗纤维化活性而具有心脏保护作用。
