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GPCR/G protein(G 蛋白偶联受体/G 蛋白)

  1. Cat.No. 产品名称 Information
  2. GC15926 BAN ORL 24

    (2R)-1-苄基-N-(3-螺[异苯并呋喃-1(3H),4'-哌啶]-1'-丙基)-2-吡咯烷甲酰胺,BAN-ORL-24;BAN ORL-24

    A nociceptin receptor antagonist
  3. GC11405 Avosentan

    N-[6-甲氧基-5-(2-甲氧基苯氧基)-2-(4-吡啶基)-4-嘧啶基]-5-甲基吡啶-2-磺酰胺,Ro 67-0565; SPP-301

    Avosentan (Ro 67-0565; SPP-301) 是一种有效的选择性内皮素受体 (ETA 受体) 拮抗剂。
  4. GC11783 Atrasentan hydrochloride

    盐酸阿曲生坦; ABT-627 hydrochloride; (+)-A 127722 hydrochloride; A-147627 hydrochloride

    Atrasentan hydrochloride (ABT-627 hydrochloride) 是一种选择性内皮素 A 受体拮抗剂,对 ETA 的 IC50 为 0.0551 nM。
  5. GC14518 Asenapine hydrochloride

    阿塞那平盐酸盐

    Asenapine hydrochloride 是一种抗精神病药,是一种 5-HT (1A, 1B, 2A, 2B, 2C, 5A, 6, 7) 和多巴胺 (D2, D3, D4) 受体拮抗剂,Ki 值为 0.03-4.0 nM,作用 5- HT 和多巴胺受体分别为 1.3、0.42、1.1 nM。
  6. GC13253 Anamorelin

    阿拉莫林,RC-1291;ONO-7643;RC1291;ONO7643;RC 1291;ONO 7643

    A small molecule agonist of GHS-R1a
  7. GC17018 AMD-070 hydrochloride

    N-(1H-苯并咪唑-2-基甲基)-N-[(8S)-5,6,7,8-四氢-8-喹啉基]-1,4-丁二胺单盐酸盐,AMD070 hydrochloride;AMD 070 hydrochloride

    CXCR4 antagonist,potent and selective
  8. GC12196 AMD-070

    N'-(1H-苯并咪唑-2-甲基)-N'-((S)-5,6,7,8-四氢喹啉-8-基)丁烷-1,4-二胺,AMD 070; AMD070

    A CXCR4 antagonist
  9. GC13476 AM966

    4'-[4-[[[(1R)-1-(2-氯苯基)乙氧基]羰基]氨基]-3-甲基-5-异恶唑基]-联苯-4-乙酸,AM 966;AM-966

    A potent and selective LPA1 receptor antagonist
  10. GC10147 AM630

    [6-碘-2-甲基-1-[2-(4-吗啉基)乙基]-1H-吲哚-3-基](4-甲氧基苯基)甲酮,AM 630;AM-630

    An inverse agonist at CB2 and partial agonist at CB1 receptors
  11. GC15908 AM-095 free base

    [4'-[3-甲基-4-[[[((R)-1-苯基乙基)氧基]羰基]氨基]异恶唑-5-基]联苯-4-基]乙酸,AM 095;AM095

    A selective LPA1 receptor antagonist
  12. GC15220 AM095

    4'-[3-甲基-4-[[[(1R)-1-苯基乙氧基]羰基]氨基]-5-异恶唑基]联苯-4-乙酸钠盐,AM 095;AM-095

    A selective LPA1 receptor antagonist
  13. GC11166 Alosetron Hydrochloride

    盐酸阿洛司琼,GR 68755C;GR 68755;GR 68755X;Lotronex;GR-68755;GR68755

    A 5-HT3 receptor antagonist
  14. GC13654 Alosetron

    阿洛司琼; GR 68755; GR 68755X

    A 5-HT3 receptor antagonist
  15. GC14879 AH 6809

    6-异丙氧基-9-氧代氧杂蒽-2-羧酸,AH6809;AH-6809

    An EP and DP receptor antagonist
  16. GC14801 5-Iodotubercidin

    5-碘代杀结核菌素,NSC 113939; 5-ITu

    An adenosine kinase inhibitor
  17. GC14145 (R,R)-Formoterol

    (-)-Formoterol;Arformoterol;Formoterol

    β2-selective adrenergic agonist
  18. GC13652 Dyphylline

    二羟丙茶碱; Diprophylline

    An adenosine receptor antagonist and phosphodiesterase inhibitor
  19. GC15505 Methylprednisolone

    甲泼尼龙; U 7532

    甲泼尼龙是皮质类固醇,可作用于糖皮质激素受体并抑制皮质醇分泌,其IC50为1.7ng/ml。
  20. GC16752 Olmesartan medoxomil

    奥美沙坦酯; CS 866

    A prodrug form of olmesartan
  21. GN10542 Scopolamine butylbromide

    丁溴东莨菪碱,Hyoscine butylbromide; (-)-Scopolamine butylbromide; Butylscopolamine bromide

    An antispasmodic agent
  22. GN10074 Xanthotoxol

    花椒毒醇,8-Hydroxypsoralen

    A coumarin with diverse biological activities
  23. GN10507 Baohuoside I

    宝藿苷 I; Icariin-II; Icariside-II

    宝活苷 I 是一种从淫羊藿中分离出来的黄酮类化合物,可作为 CXCR4 抑制剂,下调 CXCR4 表达,诱导细胞凋亡并具有抗肿瘤活性。
  24. GN10652 Norisoboldine

    去甲异波尔定,(+)-Laurelliptine

    Norisoboldine 是一种具有口服活性的天然芳烃受体 (AhR) 激动剂。
  25. GN10419 Ligustroflavone

    女贞苷; Nuezhenoside

    An apigenin triglycoside with diverse biological activities
  26. GN10104 Gramine

    芦竹碱,Donaxine

    An Analytical Reference Standard
  27. GN10186 Isocorynoxeine

    异去氢钩藤碱; 7-Isocorynoxeine

    An alkaloid with diverse biological activities
  28. GN10606 Yohimbine Hydrochloride

    盐酸育亨宾;育酚;育亨宾盐酸盐;柯楠质盐酸盐;萝芙根 (皮) 碱盐酸盐;盐酸萝芙根 (皮) 碱

    An α2-adrenoceptor antagonist
  29. GN10489 Hyodeoxycholic acid

    猪去氧胆酸; HDCA

    A secondary bile acid
  30. GN10112 Ginsenoside Rb2

    人参皂苷 Rb2; Ginsenoside C

    A natural steroid glycoside with diverse effects
  31. GN10607 Nuciferine

    荷叶碱

    An alkaloid with diverse biological activities
  32. GN10285 Theobromine

    可可碱; 3,7-Dimethylxanthine

    A methylxanthine alkaloid with diverse biological activities
  33. GN10659 Theophylline

    茶碱,Theolix

    A phosphodiesterase inhibitor and adenosine receptor antagonist
  34. GN10069 Ginsenoside Ro

    人参皂苷 Ro; Polysciasaponin P3; Chikusetsusaponin 5; Chikusetsusaponin V

    A non-steroid glycoside with diverse biological activities
  35. GN10169 3-Hydroxy-4-methoxycinnamic acid

    3-羟基-4-甲氧基肉桂酸,3-Hydroxy-4-methoxycinnamic acid

    A cinnamic acid derivative
  36. GN10680 Puerarin

    葛根素

    A natural isoflavonoid
  37. GP10110 Angiotensin III (human, mouse)

    血管紧张素III,Arg-Val-Tyr-Ile-His-Pro-Phe

    An agonist at AT1 and AT2 receptors
  38. GP10077 Angiotensin (1-7)

    Asp-Arg-Val-Tyr-Ile-His-Pro

    血管紧张素 1-7 (Ang-(1-7)) 是来自肾素-血管紧张素系统 (RAS) 的内源性七肽,由于其在心脏细胞中的抗炎和抗纤维化活性而具有心脏保护作用。

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