GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
 - Formyl Peptide Receptors(10)
 - 5-HT Receptor(482)
 - Acetylcholine(28)
 - Adenosine Deaminase(9)
 - Adenosine Receptor(130)
 - Adenosine Kinase(4)
 - Adiponectin Receptor(3)
 - Adrenergic Receptor(407)
 - Adrenergic Transporters(5)
 - Apelin Receptor(9)
 - Angiotensin Receptor(111)
 - Bombesin Receptors(23)
 - Bradykinin Receptors(29)
 - Calcitonin and Related Receptors(10)
 - Cannabinoid Receptor(118)
 - Calcimimetic Agent(2)
 - CaSR(20)
 - CCK1 Receptors(7)
 - CCK2 Receptors(7)
 - CCR(80)
 - Chemokine Receptors(23)
 - CRF1 Receptors(9)
 - CRF2 Receptors(3)
 - CXCR(77)
 - CysLT1 receptor(1)
 - Endothelin Receptor(50)
 - EP1 Receptor(2)
 - EP4 Receptor(2)
 - ERRγ(1)
 - ETA Receptors(5)
 - ETB Receptors(5)
 - Free Fatty Acid Receptors(16)
 - Galanin Receptors(11)
 - Ghrelin Receptors(11)
 - GHSR(19)
 - GIP Receptor(5)
 - Glucagon Receptor(58)
 - Glucocorticoid Receptor(96)
 - GLUT1(1)
 - Gonadotropin-Releasing Hormone Receptors(3)
 - GPCR19(12)
 - GPR109A(4)
 - GPR119(10)
 - GPR120(9)
 - GPR35(10)
 - GPR55(10)
 - Hydroxycarboxylic Acid Receptors(5)
 - Leukotriene Receptor(55)
 - LPA Receptor(12)
 - LPL Receptor(59)
 - LTD4 Receptor(1)
 - mGluR (119)
 - Melanin-concentrating Hormone Receptors(7)
 - Melanocortin (MC) Receptors(54)
 - Melatonin Receptors(23)
 - Motilin Receptor(7)
 - MT Receptor(1)
 - Non-selective CRF(7)
 - Neurotensin Receptors(23)
 - NK2 Receptors(7)
 - NK3 Receptor(5)
 - NOP Receptor(19)
 - NPY Receptors(26)
 - Orexin(3)
 - Orphan 7-TM Receptors(6)
 - OX Receptor(47)
 - Oxytocin Receptors(22)
 - P2Y Receptor(60)
 - PACAP Receptors(3)
 - PAF Receptors(7)
 - Peptide Receptors(14)
 - PGD2 Receptor(1)
 - Prostaglandin Receptor(170)
 - Protease-Activated Receptors(9)
 - RGS(2)
 - S1P receptor(8)
 - Secretin Receptors(1)
 - Sensory Neuron-Specific Receptors(1)
 - Somatostatin Receptor(39)
 - Sigma Receptor(58)
 - Vasopressin Receptor(33)
 - 17,20-lyase(4)
 - Ras(138)
 - Urotensin-II Receptor(10)
 - VIP Receptors(6)
 - EBI2/GPR183(7)
 - TSH Receptor(10)
 - NK Receptor(1)
 - GPR81(1)
 - C3aR(1)
 - CysLT2 receptor(1)
 - S1P receptor inhibitor(22)
 - CCKB(1)
 - FFAR1 (GPR40)(20)
 - GPR84(8)
 - Neuromedin U Receptors(2)
 - Kisspeptin Receptor(5)
 - CRFR(25)
 - RGS Protein(5)
 - Urotensin Receptor(6)
 - Cholecystokinin Receptor(25)
 - GPR139(4)
 - mAChR(183)
 - MCHR1 (GPR24)(16)
 - Neurokinin Receptor(75)
 - Neuropeptide S Receptor(1)
 - GPBA Receptor(1)
 - Trace Amine 1 Receptor(2)
 - GPCR protein(1)
 - FFAR3(1)
 - cGMP(26)
 - GRK(1)
 - GCGR(2)
 - GLP Receptor(2)
 - PTHR(1)
 - Protease Activated Receptor (PAR)(2)
 - Free Fatty Acid Receptor(1)
 - Formyl Peptide Receptor (FPR)(1)
 
- Cat.No. 产品名称 Information
 - 
                    
                     GC10028 
					
						
							(R)-SLV 319							
                            									            
                    The inactive enantiomer of SLV 319           
					
					 
 
				 - 
                    
                     GC15347 
					
						
							Bufuralol (hydrochloride)							
                                                           
丁呋洛尔盐酸盐,Ro 3-4787
An antagonist of β-adrenergic receptors
 
				 - 
                    
                     GC17757 
					
						
							1H-1-ethyl Candesartan Cilexetil							
                                                           
坎地沙坦EP杂质E
A potential impurity found in bulk preparations of candesartan cilexetil
 
				 - 
                    
                     GC14115 
					
						
							AVE-1625							
                                                           
屈那班,Drinabant
A potent CB1 receptor antagonist
 
				 - 
                    
                     GC18097 
					
						
							Arachidonoyl Serinol							
                            									            
                    A CB1 receptor agonist           
					
					 
 
				 - 
                    
                     GC10360 
					
						
							Lorglumide (sodium salt)							
                                                           
CR-1409 sodium salt
A selective antagonist of CCK1
 
				 - 
                    
                     GC15765 
					
						
							CYM 5520							
                            									            
                    A selective S1P2 receptor agonist           
					
					 
 
				 - 
                    
                     GC13315 
					
						
							ML-098							
                                                           
CID-7345532
A selective Rab7 activator
 
				 - 
                    
                     GC16414 
					
						
							ML-233							
                                                           
CID-46905036
A selective apelin receptor agonist
 
				 - 
                    
                     GC11453 
					
						
							ML-191							
                                                           
CCG-152883,CID-23612552
An antagonist of GPR55
 
				 - 
                    
                     GC10189 
					
						
							LY223982							
                                                           
CGS 23131,SKF 107324
A LTB4 receptor antagonist
 
				 - 
                    
                     GC13497 
					
						
							BML-111							
                                                           
BML-111
A potent bioactive analog of lipoxin A4
 
				 - 
                    
                     GC11002 
					
						
							5'-(N-Cyclopropyl)carboxamidoadenosine							
                                                           
CPCA
A specific adenosine A2 receptor agonist
 
				 - 
                    
                     GC14661 
					
						
							AM6545							
                            									            
                    A peripherally restricted CB1 receptor antagonist           
					
					 
 
				 - 
                    
                     GC12948 
					
						
							CID-1067700							
                                                           
2-[[(苯甲酰基氨基)硫代甲酰]氨基]-4,7-二氢-5,5-二甲基-5H-噻吩并[2,3-C]吡喃-3-羧酸,ML-282
A competitive GTPase inhibitor
 
				 - 
                    
                     GC14026 
					
						
							ML-193							
                                                           
CID-1261822
A selective GPR55 antagonist
 
				 - 
                    
                     GC12023 
					
						
							Celiprolol (hydrochloride)							
                                                           
盐酸塞利洛尔
A β1 adrenergic receptor antagonist
 
				 - 
                    
                     GC16216 
					
						
							Asterric Acid							
                                                           
曲地酸,Dimethylosoic Acid,RES-1214-1,TAN 1415A
An antiangiogenic agent
 
				 - 
                    
                     GC11952 
					
						
							(R)-(+)-Atenolol							
                                                           
(R)-(+)-阿替洛尔
An enantiomer of (±)-atenolol
 
				 - 
                    
                     GC15087 
					
						
							(±)-Talinolol							
                                                           
他林洛尔,Cordanum
A β1-adrenergic receptor blocker
 
				 - 
                    
                     GC13720 
					
						
							TY 52156							
                            									            
                    A S1P3 receptor antagonist           
					
					 
 
				 - 
                    
                     GC11239 
					
						
							Midodrine (hydrochloride)							
                                                           
盐酸米多君; (±)-Midodrine hydrochloride
A prodrug form of desglymidodrine
 
				 - 
                    
                     GC10673 
					
						
							E7046							
                                                           
E7046
An EP4 receptor antagonist
 
				 - 
                    
                     GC11201 
					
						
							ARM1							
                                                           
4BSA
An inhibitor of LTA4 hydrolase
 
				 - 
                    
                     GC14859 
					
						
							BW 246C							
                                                           
8-epi BW 245C
The less active C-8 diastereomer of BW 245C
 
				 - 
                    
                     GC17719 
					
						
							5-trans U-46619							
                                                           
5,6-trans U-46619
An isomer of U-46619
 
				 - 
                    
                     GC10433 
					
						
							ML-178							
                                                           
CID 44620892,CYM 50179,SID 87544119
A selective S1P4 agonist
 
				 - 
                    
                     GC17720 
					
						
							W123							
                            									            
                    Antagonist of spingosine 1-phosphate type 1 receptor           
					
					 
 
				 - 
                    
                     GC14433 
					
						
							7α,25-dihydroxy Cholesterol							
                                                           
7Α,25-二羟基胆固醇,7α,25-DHC
A potent and selective agonist of GPR183
 
				 - 
                    
                     GC11603 
					
						
							AG-041R							
                            									            
                    A potent gastrin/CCKB receptor antagonist           
					
					 
 
				 - 
                    
                     GC13712 
					
						
							FTY720 Phosphate							
                                                           
2-氨基-2-(羟基甲基)-4-(4-辛基苯基)丁基磷酸二氢酯,FTY720P
The active metabolite of FTY720
 
				 - 
                    
                     GC16826 
					
						
							Arachidonoyl amide							
                                                           
Arachidonamide,Arachidonic Acid amide
An AEA analog with similar biological activity
 
				 - 
                    
                     GC16663 
					
						
							(±)-4-hydroxy Propranolol (hydrochloride)							
                                                           
4-羟基普萘洛尔盐酸盐,(±)-4-hydroxy Propranolol hydrochloride
An active metabolite of propranolol
 
				 - 
                    
                     GC13284 
					
						
							CJ-42794							
                                                           
4-[(1S)-1-[[5-氯-2-(4-氟苯氧基)苄基]氨基]乙基]苯甲酸,RQ-00015986
A selective EP4 receptor antagonist
 
				 - 
                    
                     GC12290 
					
						
							Norgestimate							
                                                           
诺孕酯
A progestin
 
				 - 
                    
                     GC15640 
					
						
							BAY u3405							
                                                           
雷马曲班; BAY u3405
A dual TP and DP2/CRTH2 receptor antagonist
 
				 - 
                    
                     GC18111 
					
						
							Seratrodast							
                                                           
塞曲司特; AA 2414
A thromboxane A2 receptor antagonist
 
				 - 
                    
                     GC14758 
					
						
							BM 567							
                            									            
                    A dual thromboxane synthase inhibitor/TP receptor antagonist           
					
					 
 
				 - 
                    
                     GC12538 
					
						
							LH 21							
                            									            
                    Weak CB1 antagonist           
					
					 
 
				 - 
                    
                     GC10771 
					
						
							CJ-023423							
                                                           
RQ-00000007
An EP4 receptor antagonist
 
				 - 
                    
                     GC10284 
					
						
							Apelin-13							
                                                           
人牛APELIN-13
Apelin-13 是一种肽,被称为 G 蛋白偶联受体 APJ 的配体。
 
				 - 
                    
                     GC17699 
					
						
							O-1821							
                                                           
Cannabidiorcin, Cannabidiorcol, Cannabidiorocol, CBD-C1, CBDO
An analog of O-1918, a selective antagonist of a non-CB1/CB2 receptor
 
				 - 
                    
                     GC13333 
					
						
							Zilpaterol							
                                                           
齐帕特罗,RU-42173,Zilmax?
β-adrenergic receptor agonist
 
				 - 
                    
                     GC16800 
					
						
							MF498							
                            									            
                    A selective EP4 antagonist           
					
					 
 
				 - 
                    
                     GC13020 
					
						
							BayCysLT2							
                                                           
CAY10633
A potent CysLT2 receptor antagonist
 
				 - 
                    
                     GC10116 
					
						
							2-chloro-3-Deazaadenosine							
                                                           
6-Amino-2-chloropurine riboside,2-CADO,NSC 158900
Agonist of adenosine receptors
 
				 - 
                    
                     GC15758 
					
						
							BQCA							
                                                           
1-(4-甲氧基苄基)-4-氧代-1,4-二氢喹啉-3-羧酸
A positive allosteric modulator of the M1 mAChR
 
				 - 
                    
                     GC13302 
					
						
							Guanabenz (hydrochloride)							
                                                           
Wytensin
An α2-adrenergic receptor agonist
 
				 - 
                    
                     GC16027 
					
						
							ONO-8711							
                                                           
(5Z)-6-[(2R,3S)-3-[[[(4-氯-2-甲基苯基)磺酰基]氨基]甲基]双环[2.2.2]辛-2-基]-5-己烯酸
A potent EP1 receptor antagonist
 
				 - 
                    
                     GC17064 
					
						
							Lofexidine (hydrochloride)							
                                                           
盐酸洛非西定; Baq-168; MDL-14042
An α2-adrenergic receptor agonist