GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(482)
- Acetylcholine(28)
- Adenosine Deaminase(9)
- Adenosine Receptor(130)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(407)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(111)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(118)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(80)
- Chemokine Receptors(23)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(77)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(96)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(12)
- LPL Receptor(59)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(54)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(23)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(47)
- Oxytocin Receptors(22)
- P2Y Receptor(60)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(170)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(58)
- Vasopressin Receptor(33)
- 17,20-lyase(4)
- Ras(138)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(183)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(26)
- GRK(1)
- GCGR(2)
- GLP Receptor(2)
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
- Cat.No. 产品名称 Information
-
GC15292
(S)-(+)-Niguldipine hydrochloride
L-type Ca2+ channel blocker and α1A-adrenoceptor antagonist
-
GC16480
AM 281
1-(2,4-二氯苯基)-5-(4-碘苯基)-4-甲基-N-吗啉-1H-吡唑-3-甲酰胺
AM 281是一种高亲和力和特异性的选择性CB2受体拮抗剂,其IC50为13μM。AM 281用于研究内源性大麻素系统在各种生理和病理过程中的作用,具有在炎症、疼痛和神经退行性疾病研究中的潜在应用价值。 -
GC14036
ACPT-II
An antagonist of metabotropic glutamate receptors
-
GC10219
AF-DX 116
11-((2-((二乙氨基)甲基)-1-哌啶基)乙酰基)-5,11-二氢-(6H)-吡啶并[2.3-B][1.4]苯并二氮杂-6-酮,AF-DX 116
A muscarinic M2 receptor antagonist -
GC17503
2-Cl-IB-MECA
CF-102; 2-Cl-IB-MECA
An adenosine A3 receptor agonist -
GC17085
Procaterol hydrochloride
盐酸丙卡特罗
A β2-adrenergic receptor agonist -
GC17301
(+)-SK&F 10047 hydrochloride
原型 σ1 受体激动剂
-
GC15039
(S)-(-)-Pindolol
S-吲哚洛尔
beta-adrenergic antagonist -
GC11231
BW 723C86 hydrochloride
BW723C86盐酸盐
A selective HT2B receptor agonist -
GC17933
WIN 64338 hydrochloride
WIN 64338 hydrochloride 是一种有效的、选择性的、非肽竞争性缓激肽 B2 受体拮抗剂。
-
GC17524
GR 55562 dihydrochloride
5-HT1B (5-HT1Dβ) silent antagonist
-
GC14527
A 61603 hydrobromide
A61603氢溴酸
An α1A-adrenoceptor agonist -
GC16111
Zinterol hydrochloride
净特罗,MJ 9184 hydrochloride
Zinterol hydrochloride (MJ 9184) 是一种有效的选择性 β2-adrenoceptor 激动剂。 -
GC12532
CHPG
Chlorohydroxyphenylglycine, CHPG
A potent and selective mGluR5 agonist -
GC11017
ZM 241385
An A2A adenosine receptor antagonist
-
GC16020
8-M-PDOT
AH-002
An MT2 receptor agonist -
GC16186
4-P-PDOT
AH 024
An antagonist of the MT2 receptor -
GC10068
CP 93129 dihydrochloride
A 5-HT1B receptor agonist
-
GC17383
PHCCC
N-苯基-7-(羟基亚胺基)环丙烯并[B]苯并吡喃-1A-甲酰胺
PHCCC 是 I 组 mGluR 拮抗剂,IC50 为 3 μM。 PHCCC 是 mGlu4 受体的选择性正调节剂。抗帕金森效应。 -
GC15482
Nisoxetine hydrochloride
盐酸尼索西汀
A NET inhibitor -
GC15354
CGP 20712 dihydrochloride
β1 antagonist,highly potent and selective
-
GC11305
LY 225910
2-[2-(5-溴-1H-吲哚-3-基)乙基]-3-[3-(1-甲基乙氧基)苯基]-4-(3H-)-喹唑啉酮
CCK2受体拮抗剂 -
GC15979
RS 16566 dihydrochloride
(R)-zacopride 结合位点的配体
-
GC13192
E4CPG
(RS)-ECPG
An antagonist of mGluR1 and mGluR2 -
GC16553
N-Desmethylclozapine
N-去甲基氯氮平; Norclozapine; Desmethylclozapine; Normethylclozapine
An active metabolite of clozapine -
GC10197
AH 11110 hydrochloride
α1B-AR ligand,subtype-selective
-
GC14696
RS 67506 hydrochloride
potent and selective 5-HT4 partial agonist
-
GC15137
RS 56812 hydrochloride
5-HT3 partial agonist
-
GC10723
RS 79948 hydrochloride
α2-adrenoreceptor antagonist
-
GC11077
Imiloxan hydrochloride
α2-adrenoceptor antagonist
-
GC17070
RS 17053 hydrochloride
RS-17053
An α1A-adrenergic receptor antagonist -
GC15374
BD 1047 dihydrobromide
BD-1047盐酸盐
A selective antagonist of σ1 receptors -
GC17666
Xamoterol hemifumarate
富马酸扎莫特罗,Corwin hemifumarate; ICI 118587 hemifumarate
A β1-adrenergic receptor partial agonist -
GC13785
BRL 37344, sodium salt
BRL37344钠盐,BRL 37344A
A selective β3-adrenergic receptor agonist -
GC17745
MK 212 hydrochloride
2-氯-6-哌嗪吡嗪盐酸盐,CPP monohydrochloride
A 5-HT2C receptor agonist -
GC17543
ZD 7114 hydrochloride
β3-adrenoceptor agonist
-
GC10965
ARC 239 dihydrochloride
ARC?239二盐酸盐
An α2B-adrenergic receptor antagonist -
GC11188
GR 135531
N-甲氧基羰基琥珀酰亚胺,5-METHOXYCARBONYLAMINO-N-ACETYLTRYPTAMINE
MT3 receptor agonist -
GC15838
BD 1063 dihydrochloride
BD1063(盐酸盐)
An antagonist of σ1 receptors -
GC17777
Palmitoylethanolamide
十六酰胺乙醇,Palmidrol; Loramine P 256
An endogenous cannabinoid -
GC14042
Oleamide
油酸酰胺
An amide of oleic acid and agonist of CB1 receptors -
GC17898
Luzindole
N-乙酰-2-苄基色胺,N-0774
A melatonin receptor antagonist -
GC11119
MDL 11,939
MDL11939
A potent 5-HT2A receptor antagonist -
GC18128
L-732,138
An NK1 receptor antagonist
-
GC12761
ICI 89406
N-[2-[[3-(2-氰基苯氧基)-2-羟基丙基]氨基]乙基]-N'-苯基脲
ICI 89406 是一种选择性 β1 肾上腺素能受体拮抗剂,适合用正电子发射器标记,用于 PET。 -
GC17185
MSOP
MSOP 是一种选择性 III 族代谢型谷氨酸受体拮抗剂,对 L-AP4 敏感的突触前 mGluR 的表观 KD 为 51 μM。
-
GC15813
Idazoxan hydrochloride
盐酸咪唑克生
盐酸咪唑克生(Idazoxan hydrochloride ,RX 781094 hydrochloride ,IDA)是一种分子量为241的α2-肾上腺和咪唑啉受体配体。 -
GC15672
Efaroxan hydrochloride
盐酸盐依法克生
An α2-AR and I1 receptor antagonist -
GC15465
N-[2-(Piperidinylamino)ethyl]-4-iodobenzamide
σ-1 selective ligand
-
GC11575
SM-21 maleate
Increases release of acetylcholine,σ2 antagonist