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GPCR/G protein(G 蛋白偶联受体/G 蛋白)

  1. Cat.No. 产品名称 Information
  2. GC10972 Gallamine Triethiodide

    三碘季胺酚

    An allosteric modulator of muscarinic acetylcholine receptors
  3. GC15746 Mometasone furoate

    糠酸莫米松; Sch32088

    A synthetic glucocorticoid prodrug
  4. GC14094 Pranlukast

    普鲁司特; ONO-1078

    A CysLT1 receptor antagonist
  5. GC10714 Fluocinonide

    氟轻松

    A synthetic corticosteroid
  6. GC11976 Clobetasol propionate

    丙酸氯倍他索

    A corticosteroid
  7. GC12931 Deflazacort

    地夫可特

    A prodrug for an active glucocorticoid
  8. GC17483 Trospium chloride

    曲司氯铵

    An antagonist of muscarinic receptors
  9. GC12974 Medroxyprogesterone acetate

    醋酸甲羟孕酮; Medroxyprogesterone 17-acetate; Farlutin

    Medroxyprogesterone acetate(MPA)是一种人工合成的孕激素。
  10. GC11257 Fluocinolone Acetonide

    醋酸肤轻松

    A synthetic corticosteroid
  11. GC16836 Naftopidil

    萘哌地尔; KT-611; BM-15275

    Naftopidil (KT-611) 是一种选择性 alpha1-adrenoceptor 拮抗剂,对克隆的人 α1a-、α1b- 和 α1d-adrenoceptor 亚型的 Kis 分别为 3.7 nM、20 nM 和 1.2 nM。
  12. GC14818 Bisoprolol fumarate

    比索洛尔富马酸盐

    A β1-AR antagonist
  13. GC14563 Ketanserin

    酮色林; R41468

    A potent 5-HT2 receptor antagonist
  14. GC11191 Buspirone HCl

    盐酸丁螺环酮

    An Analytical Reference Standard
  15. GC10434 Triamcinolone

    曲安西龙

    A synthetic glucocorticoid
  16. GC17974 Latrepirdine dihydrochloride

    2,3,4,5-四氢-2,8-二甲基-5-[2-(6-甲基-3-吡啶基)乙基]-1H-吡啶并[4,3-B]吲哚二盐酸盐,Dimebolin dihydrochloride

    A neuroprotective agent
  17. GC17061 Dapoxetine HCl

    盐酸达泊西汀; LY-210448 hydrochloride

    An Analytical Reference Standard
  18. GC15829 Urapidil HCl

    盐酸乌拉地尔

    An α1-AR antagonist and 5-HT1A receptor partial agonist
  19. GC12376 Maprotiline HCl

    盐酸马普替林

    A tricyclic antidepressant
  20. GC13993 Terazosin HCl

    盐酸特拉唑嗪(二水合物)

    A potent and selective α1-AR antagonist
  21. GC15107 Clomipramine HCl

    盐酸氯米帕明; Chlorimipramine hydrochloride; G-34586 hydrochloride; NSC-169865 hydrochloride

    A tricyclic antidepressant
  22. GC13134 Tiotropium Bromide hydrate

    噻托溴铵一水合物,BA-679 BR (hydrate)

    A muscarinic receptor antagonist
  23. GC14927 Trazodone HCl

    盐酸曲唑酮; AF-1161

    An Analytical Reference Material
  24. GC17367 Rebamipide

    瑞巴派特; OPC12759; Proamipide

    A gastroprotective agent and mucin secretagogue
  25. GC14021 Betaxolol

    倍他洛尔

    An Analytical Reference Standard
  26. GC17825 Methscopolamine

    甲溴东莨菪碱

    A muscarinic acetylcholine receptor antagonist
  27. GC12724 Phenoxybenzamine HCl

    盐酸酚苄明

    An α-AR antagonist
  28. GC16142 Ondansetron

    昂丹司琼; GR 38032; SN 307

    A Certified Reference Material
  29. GC15153 Almotriptan Malate

    马来酸阿莫曲坦; PNU180638

    An agonist of 5-HT1B and 5-HT1D receptors
  30. GC15063 Ritodrine HCl

    盐酸利托君; DU21220 hydrochloride

    A β2-AR agonist
  31. GC15150 Tropicamide

    托吡卡胺; Ro 1-7683

    A selective muscarinic M4 antagonist
  32. GC15687 Azasetron HCl

    盐酸阿扎司琼; Y-25130 hydrochloride

    A 5-HT3 receptor antagonist
  33. GC16291 Phentolamine Mesylate

    甲磺酸酚妥拉明; Phentolamine methanesulfonate

    A reversible α-adrenergic receptor antagonist
  34. GC11447 Mirtazapine

    米氮平

    An Analytical Reference Material
  35. GC14216 Chlorpromazine HCl

    盐酸氯丙嗪

    Chlorpromazine HCl是一种口服有效的、可透过血脑屏障的吩噻嗪类抗精神病药,能够有效抑制D2多巴胺受体和5-HT2A,具有很强的镇静作用。
  36. GC11343 Propranolol HCl

    盐酸普萘洛尔

    A β-adrenergic receptor antagonist
  37. GC10738 Brimonidine Tartrate

    酒石酸溴莫尼定; UK 14304 tartrate; AGN190342 tartrate

    An α2-adrenergic receptor agonist
  38. GC14988 Naphazoline HCl

    盐酸萘甲唑啉; Naphthazoline hydrochloride

    A vasoconstrictor
  39. GC13974 Salbutamol Sulfate

    沙丁胺醇半硫酸盐; Albuterol hemisulfate; AH-3365 hemisulfate

    A β2-AR agonist
  40. GC10750 Dexmedetomidine HCl

    盐酸右美托咪定; (+)-Medetomidine hydrochloride; (S)-Medetomidine hydrochloride

    An α2-adrenoceptor agonist
  41. GC12403 Ozagrel HCl

    盐酸奥扎格雷,OKY-046 hydrochloride

    A selective inhibitor of TXA synthase
  42. GC13173 Sotalol

    索他洛尔,(R)-Sotalol

    An Analytical Reference Standard
  43. GC17296 Xylazine HCl

    盐酸甲苯噻嗪,BAY 1470 hydrochloride

    An α2-adrenergic receptor agonist

  44. GC11029 Isoprenaline HCl

    盐酸异丙肾上腺素; Isoproterenol hydrochloride

    A β1- and β2-AR agonist

  45. GC12231 Sulfisoxazole

    磺胺异恶唑; Sulfafurazole

    An antibiotic and endothelin receptor antagonist
  46. GC15243 Carbazochrome sodium sulfonate (AC-17)

    卡络磺钠; AC-17

    Carbazochrome sodium sulfonate (AC-17) (AC-17) 是一种毛细血管稳定剂,用于研究出血。
  47. GC14536 Metoprolol Tartrate

    酒石酸美托洛尔

    An Analytical Reference Standard
  48. GC11479 Xylometazoline HCl

    盐酸赛洛唑啉

    An α-adrenergic receptor agonist
  49. GC15754 WAY-100635 Maleate A serotonin 5-HT1A antagonist
  50. GC13501 VUF 10166 A 5-HT3 receptor antagonist
  51. GC13281 VU 0364770 An mGluR4 and mGluR6 positive allosteric modulator and mGluR5 antagonist

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