GPCR/G protein(G 蛋白偶联受体/G 蛋白)
- Neuropeptide FF/AF Receptors(49)
- Formyl Peptide Receptors(10)
- 5-HT Receptor(482)
- Acetylcholine(28)
- Adenosine Deaminase(9)
- Adenosine Receptor(130)
- Adenosine Kinase(4)
- Adiponectin Receptor(3)
- Adrenergic Receptor(407)
- Adrenergic Transporters(5)
- Apelin Receptor(9)
- Angiotensin Receptor(111)
- Bombesin Receptors(23)
- Bradykinin Receptors(29)
- Calcitonin and Related Receptors(10)
- Cannabinoid Receptor(118)
- Calcimimetic Agent(2)
- CaSR(20)
- CCK1 Receptors(7)
- CCK2 Receptors(7)
- CCR(80)
- Chemokine Receptors(23)
- CRF1 Receptors(9)
- CRF2 Receptors(3)
- CXCR(77)
- CysLT1 receptor(1)
- Endothelin Receptor(50)
- EP1 Receptor(2)
- EP4 Receptor(2)
- ERRγ(1)
- ETA Receptors(5)
- ETB Receptors(5)
- Free Fatty Acid Receptors(16)
- Galanin Receptors(11)
- Ghrelin Receptors(11)
- GHSR(19)
- GIP Receptor(5)
- Glucagon Receptor(58)
- Glucocorticoid Receptor(96)
- GLUT1(1)
- Gonadotropin-Releasing Hormone Receptors(3)
- GPCR19(12)
- GPR109A(4)
- GPR119(10)
- GPR120(9)
- GPR35(10)
- GPR55(10)
- Hydroxycarboxylic Acid Receptors(5)
- Leukotriene Receptor(55)
- LPA Receptor(12)
- LPL Receptor(59)
- LTD4 Receptor(1)
- mGluR (119)
- Melanin-concentrating Hormone Receptors(7)
- Melanocortin (MC) Receptors(54)
- Melatonin Receptors(23)
- Motilin Receptor(7)
- MT Receptor(1)
- Non-selective CRF(7)
- Neurotensin Receptors(23)
- NK2 Receptors(7)
- NK3 Receptor(5)
- NOP Receptor(19)
- NPY Receptors(26)
- Orexin(3)
- Orphan 7-TM Receptors(6)
- OX Receptor(47)
- Oxytocin Receptors(22)
- P2Y Receptor(60)
- PACAP Receptors(3)
- PAF Receptors(7)
- Peptide Receptors(14)
- PGD2 Receptor(1)
- Prostaglandin Receptor(170)
- Protease-Activated Receptors(9)
- RGS(2)
- S1P receptor(8)
- Secretin Receptors(1)
- Sensory Neuron-Specific Receptors(1)
- Somatostatin Receptor(39)
- Sigma Receptor(58)
- Vasopressin Receptor(33)
- 17,20-lyase(4)
- Ras(138)
- Urotensin-II Receptor(10)
- VIP Receptors(6)
- EBI2/GPR183(7)
- TSH Receptor(10)
- NK Receptor(1)
- GPR81(1)
- C3aR(1)
- CysLT2 receptor(1)
- S1P receptor inhibitor(22)
- CCKB(1)
- FFAR1 (GPR40)(20)
- GPR84(8)
- Neuromedin U Receptors(2)
- Kisspeptin Receptor(5)
- CRFR(25)
- RGS Protein(5)
- Urotensin Receptor(6)
- Cholecystokinin Receptor(25)
- GPR139(4)
- mAChR(183)
- MCHR1 (GPR24)(16)
- Neurokinin Receptor(75)
- Neuropeptide S Receptor(1)
- GPBA Receptor(1)
- Trace Amine 1 Receptor(2)
- GPCR protein(1)
- FFAR3(1)
- cGMP(26)
- GRK(1)
- GCGR(2)
- GLP Receptor(2)
- PTHR(1)
- Protease Activated Receptor (PAR)(2)
- Free Fatty Acid Receptor(1)
- Formyl Peptide Receptor (FPR)(1)
- Cat.No. 产品名称 Information
-
GC10028
(R)-SLV 319
The inactive enantiomer of SLV 319
-
GC15347
Bufuralol (hydrochloride)
丁呋洛尔盐酸盐,Ro 3-4787
An antagonist of β-adrenergic receptors -
GC17757
1H-1-ethyl Candesartan Cilexetil
坎地沙坦EP杂质E
A potential impurity found in bulk preparations of candesartan cilexetil -
GC14115
AVE-1625
屈那班,Drinabant
A potent CB1 receptor antagonist -
GC18097
Arachidonoyl Serinol
A CB1 receptor agonist
-
GC10360
Lorglumide (sodium salt)
CR-1409 sodium salt
A selective antagonist of CCK1 -
GC15765
CYM 5520
A selective S1P2 receptor agonist
-
GC13315
ML-098
CID-7345532
A selective Rab7 activator -
GC16414
ML-233
CID-46905036
A selective apelin receptor agonist -
GC11453
ML-191
CCG-152883,CID-23612552
An antagonist of GPR55 -
GC10189
LY223982
CGS 23131,SKF 107324
A LTB4 receptor antagonist -
GC13497
BML-111
BML-111
A potent bioactive analog of lipoxin A4 -
GC11002
5'-(N-Cyclopropyl)carboxamidoadenosine
CPCA
A specific adenosine A2 receptor agonist -
GC14661
AM6545
A peripherally restricted CB1 receptor antagonist
-
GC12948
CID-1067700
2-[[(苯甲酰基氨基)硫代甲酰]氨基]-4,7-二氢-5,5-二甲基-5H-噻吩并[2,3-C]吡喃-3-羧酸,ML-282
A competitive GTPase inhibitor -
GC14026
ML-193
CID-1261822
A selective GPR55 antagonist -
GC12023
Celiprolol (hydrochloride)
盐酸塞利洛尔
A β1 adrenergic receptor antagonist -
GC16216
Asterric Acid
曲地酸,Dimethylosoic Acid,RES-1214-1,TAN 1415A
An antiangiogenic agent -
GC11952
(R)-(+)-Atenolol
(R)-(+)-阿替洛尔
An enantiomer of (±)-atenolol -
GC15087
(±)-Talinolol
他林洛尔,Cordanum
A β1-adrenergic receptor blocker -
GC13720
TY 52156
A S1P3 receptor antagonist
-
GC11239
Midodrine (hydrochloride)
盐酸米多君; (±)-Midodrine hydrochloride
A prodrug form of desglymidodrine -
GC10673
E7046
E7046
An EP4 receptor antagonist -
GC11201
ARM1
4BSA
An inhibitor of LTA4 hydrolase -
GC14859
BW 246C
8-epi BW 245C
The less active C-8 diastereomer of BW 245C -
GC17719
5-trans U-46619
5,6-trans U-46619
An isomer of U-46619 -
GC10433
ML-178
CID 44620892,CYM 50179,SID 87544119
A selective S1P4 agonist -
GC17720
W123
Antagonist of spingosine 1-phosphate type 1 receptor
-
GC14433
7α,25-dihydroxy Cholesterol
7Α,25-二羟基胆固醇,7α,25-DHC
A potent and selective agonist of GPR183 -
GC11603
AG-041R
A potent gastrin/CCKB receptor antagonist
-
GC13712
FTY720 Phosphate
2-氨基-2-(羟基甲基)-4-(4-辛基苯基)丁基磷酸二氢酯,FTY720P
The active metabolite of FTY720 -
GC16826
Arachidonoyl amide
Arachidonamide,Arachidonic Acid amide
An AEA analog with similar biological activity -
GC16663
(±)-4-hydroxy Propranolol (hydrochloride)
4-羟基普萘洛尔盐酸盐,(±)-4-hydroxy Propranolol hydrochloride
An active metabolite of propranolol -
GC13284
CJ-42794
4-[(1S)-1-[[5-氯-2-(4-氟苯氧基)苄基]氨基]乙基]苯甲酸,RQ-00015986
A selective EP4 receptor antagonist -
GC12290
Norgestimate
诺孕酯
A progestin -
GC15640
BAY u3405
雷马曲班; BAY u3405
A dual TP and DP2/CRTH2 receptor antagonist -
GC18111
Seratrodast
塞曲司特; AA 2414
A thromboxane A2 receptor antagonist -
GC14758
BM 567
A dual thromboxane synthase inhibitor/TP receptor antagonist
-
GC12538
LH 21
Weak CB1 antagonist
-
GC10771
CJ-023423
RQ-00000007
An EP4 receptor antagonist -
GC10284
Apelin-13
人牛APELIN-13
Apelin-13 是一种肽,被称为 G 蛋白偶联受体 APJ 的配体。 -
GC17699
O-1821
Cannabidiorcin, Cannabidiorcol, Cannabidiorocol, CBD-C1, CBDO
An analog of O-1918, a selective antagonist of a non-CB1/CB2 receptor -
GC13333
Zilpaterol
齐帕特罗,RU-42173,Zilmax?
β-adrenergic receptor agonist -
GC16800
MF498
A selective EP4 antagonist
-
GC13020
BayCysLT2
CAY10633
A potent CysLT2 receptor antagonist -
GC10116
2-chloro-3-Deazaadenosine
6-Amino-2-chloropurine riboside,2-CADO,NSC 158900
Agonist of adenosine receptors -
GC15758
BQCA
1-(4-甲氧基苄基)-4-氧代-1,4-二氢喹啉-3-羧酸
A positive allosteric modulator of the M1 mAChR -
GC13302
Guanabenz (hydrochloride)
Wytensin
An α2-adrenergic receptor agonist -
GC16027
ONO-8711
(5Z)-6-[(2R,3S)-3-[[[(4-氯-2-甲基苯基)磺酰基]氨基]甲基]双环[2.2.2]辛-2-基]-5-己烯酸
A potent EP1 receptor antagonist -
GC17064
Lofexidine (hydrochloride)
盐酸洛非西定; Baq-168; MDL-14042
An α2-adrenergic receptor agonist