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Home >> Signaling Pathways >> Metabolism

Metabolism(代谢)

  1. Cat.No. 产品名称 Information
  2. GC13683 Rivaroxaban

    利伐沙班; BAY 59-7939

     A selective inhibitor of Factor Xa
  3. GC15890 Cilostazol

    西洛他唑; OPC 13013

     A PDE3A inhibitor
  4. GC13614 Mycophenolate Mofetil

    吗替麦考酚酯; RS 61443; TM-MMF

     A prodrug form of mycophenolic acid
  5. GC15558 Mildronate

    米屈肼,Meldonium; MET-88; Quaterin

     An inhibitor of carnitine biosynthesis
  6. GC16856 Avanafil

    阿伐那非; TA1790

     A potent and selective PDE5 inhibitor
  7. GC14921 CPI-613

    6,8-双(苄硫基)辛酸,CPI-613

     An inhibitor of α-ketoglutarate dehydrogenase
  8. GC12596 Nepicastat (SYN-117) HCl

    盐酸内匹司他,SYN-117 hydrochloride; RS-25560-197 hydrochloride

     An inhibitor of dopamine β-hydroxylase
  9. GC14180 GSK256066

    6-[[3-[(二甲基氨基)羰基]苯基]磺酰]-4-[(3-甲氧基苯基)氨基]-8-甲基-3-喹啉甲酰胺

     A potent PDE4 inhibitor
  10. GC15382 Isotretinoin

    异维A酸; 13-cis-Retinoic acid

     A retinoid
  11. GC17598 Cilomilast

    西洛司特; SB-207499

     A PDE4 inhibitor
  12. GC16629 Rolipram

    诺普利兰,(R,S)-Rolipram; SB 95952; ZK 62711

     A phosphodiesterase-4 inhibitor
  13. GC17074 Tadalafil

    他达那非; IC-351

     A PDE5 inhibitor
  14. GC15194 PF-2545920

    2-[[4-[1-(甲基-11C)-4-(4-吡啶基)-1H-吡唑-3-基]苯氧基]甲基]喹啉

     A potent inhibitor of PDE10A
  15. GC11152 Pioglitazone HCl

    盐酸吡格列酮,U 72107A; AD 4833

     A PPARγ agonist
  16. GC10588 Vardenafil HCl Trihydrate

    盐酸瓦地那非三水合物

     An inhibitor of PDE5 and PDE6
  17. GC16754 Clarithromycin

    克拉霉素

     A macrolide antibiotic
  18. GC17685 Sildenafil Citrate

    西地那非柠檬酸盐; UK-92480 citrate

     A PDE5 inhibitor
  19. GC13079 Voriconazole

    伏立康唑,(±)-UK-109496

     A triazole antifungal agent
  20. GC16347 Roflumilast

    罗氟司特

     A PDE4 inhibitor
  21. GC10999 Avasimibe

    阿伐麦布,CI-1011; PD-148515

     Avasimibe是一种选择性口服酰基辅酶A：胆固醇酰基转移酶（ACAT）抑制剂（IC50=12μmol/L）。
  22. GC10420 Apremilast (CC-10004)

    阿普司特; CC-10004

     An orally available PDE4 inhibitor
  23. GC17337 Ketoconazole

    酮康唑

     A triazole antifungal agent
  24. GC14269 Cobicistat (GS-9350)

    可比司他,GS-9350

     An inhibitor of CYP3A
  25. GC12280 PF-4981517

    CYP3cide,PF-04981517,PF4981517

     A potent, selective inhibitor of CYP3A4
  26. GC15516 Rosiglitazone HCl

    盐酸罗格列酮; BRL 49653 hydrochloride

     A PPARγ agonist
  27. GC15318 GW501516

    2-(4-((2-(4-(三氟甲基)苯基)-5-甲基噻唑-4-基)甲基硫基)-2-甲基苯氧基)乙酸,GW 1516; GSK-516

     A selective PPARδ-agonist with anti-obesity activity
  28. GC16575 Alizarin

    1,2-二羟基蒽醌

     A CYP450 inhibitor
  29. GC14983 GW0742

    GW 0742

     A selective agonist of PPARδ
  30. GC13633 Ciprofibrate

    环丙贝特; Win35833

     A selective PPARα agonist
  31. GC14403 WY-14643 (Pirinixic Acid)

    匹立尼酸,WY 14643,WY14643

     WY-14643 (Pirinixic Acid)是一种高效、具备选择性高亲和力的过氧化物酶体增殖物激活受体α（PPARα）受体激动剂，对小鼠的 PPARα受体的EC50为0.63μM，对人的 PPARα受体的EC50为5μM。
  32. GC16444 Rosiglitazone

    罗格列酮; BRL 49653

     Rosiglitazone是一种具有口服活性的过氧化物酶体增殖物活化受体γ（PPARγ ）选择性激动剂，选择性地激活含有PPARγ配体结合域（LBD）的嵌合体，而不是PPARα和PPARδ，EC50为60 nM，Kd为40 nM。
  33. GC16009 GSK3787

    GSK-3787,GSK 3787

     A selective, irreversible PPARβ/δ antagonist
  34. GC11318 Rosiglitazone maleate

    马来酸罗格列酮; BRL 49653C

     A PPARγ agonist
  35. GC12820 T0070907 A potent and selective PPARγ antagonist
  36. GC13969 GW9662

    2-氯-5-硝基-N-苯基苯酰胺

     GW9662是一种特异性的过氧化物酶体增殖物激活受体-γ(PPAR-γ)抑制剂,其IC50为3.3 nM。
  37. GC17645 Abiraterone

    阿比特龙,CB 7598,16-dien-3-ol,CB7598

     A CYP17A1 inhibitor and an active metabolite of abiraterone acetate
  38. GC11108 Abiraterone acetate

    乙酸阿比特龙酯,CB7630

     A CYP17A1 inhibitor
  39. GC10538 Pifithrin-α (PFTα)

    2-(2-亚氨基-4,5,6,7-四氢苯并噻唑-3-基)-1-P-甲苯基乙酮氢溴酸盐,Pifithrin hydrobromide; PFTα hydrobromide

     Pifithrin-α是一种p53抑制剂。
  40. GC15442 Tipifarnib (Zarnestra)

    替吡法尼; IND 58359; R115777

     A farnesyltransferase inhibitor with antitumor activity
  41. GC11008 Necrostatin-1

    MTH-DL-Tryptophan,Nec-1

     Necrostatin-1主要作用于细胞中的RIP1，Necrostatin-1是一种RIP1激酶抑制剂，IC50值为0.32 mM。
  42. GC10240 Atazanavir sulfate (BMS-232632-05)

    硫酸阿扎那韦; BMS-232632 sulfate

     An inhibitor of HIV-1 protease
  43. GC12945 Atazanavir

    阿扎那韦; BMS-232632

    An inhibitor of HIV-1 protease
  44. GC15130 Alogliptin (SYR-322)

    阿格列汀; SYR-322 free base

     Alogliptin (SYR-322) (SYR-322 free base) 是一种有效的、选择性的、具有口服活性的 DPP-4 抑制剂，IC50 <10 nM，选择性比 DPP-8 和 DPP-9 高 10,000 倍以上.
  45. GC16733 Vildagliptin (LAF-237)

    维格列汀; LAF237; NVP-LAF 237

     A DPP-4 inhibitor
  46. GC14827 Linagliptin (BI-1356)

    利格列汀; BI 1356

     A potent DPP-4 inhibitor
  47. GC13139 FG-4592 (ASP1517)

    罗沙司他,Roxadustat

     FG-4592 作为一种口服生物可利用的缺氧诱导因子 (HIF) 脯氨酰羟化酶抑制剂，可通过 HIF 介导的转录促进协调性红细胞生成。
  48. GC13946 SNX-2112

    PF-04928473

     A potent Hsp90 inhibitor
  49. GC11403 Radicicol

    根赤壳菌素; Monorden

     An inhibitor of Hsp90
  50. GC11179 NVP-BEP800

    NVP-BEP800

     An Hsp90 inhibitor
  51. GC14322 MPC-3100 An inhibitor of Hsp90

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