Dopamine β-hydroxylase(多巴胺β-羟化酶)
DBH (Dopamine-β-hydroxylase) is a copper-containing monooxygenase that catalyzes the biosynthesis of catecholamine neurotransmitter, norepinephrine from dopamine. Deficiency in DBH causes orthostatic hypotension, autonomic disorders etc.
- Cat.No. 产品名称 Information
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GC60519
4-Hydroxyderricin
4-Hydroxyderricin(4-HD), the major active ingredients of Angelica keiskei Koidzumi, is a potent selective monoamine oxidase (MAO) inhibitor with mild inhibitory effect on dopamine β-hydroxylase.
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GC36722
Nepicastat
An inhibitor of dopamine β-hydroxylase
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GC32593
Zamicastat (BIA 5-1058)
Zamicastat (BIA 5-1058) (BIA 5-1058) 是一种多巴胺 β-羟化酶 (DBH) 抑制剂,可穿过血脑屏障 (BBB) 引起中枢和外周效应。
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GC32575
Etamicastat (BIA 5-453)
Etamicastat (BIA 5-453) (BIA 5-453) 是一种有效且可逆的多巴胺-β-羟化酶 (DBH) 抑制剂,IC50 值为 107 nM。
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GC18061
Fusaric Acid
A mycotoxin
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GC10718
PF 915275
PF 915275 是一种有效的、选择性的、具有口服活性的人 11β-羟基类固醇脱氢酶 1 型 (11βHSD1) 抑制剂,Ki 为 2.3 nM,EC50 为 15 nM(在 HEK293 细胞中)。
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GC15558
Mildronate
An inhibitor of carnitine biosynthesis
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GC12596
Nepicastat (SYN-117) HCl
An inhibitor of dopamine β-hydroxylase
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GC15382
Isotretinoin
A retinoid
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GC10801
Disulfiram
An irreversible inhibitor of aldehyde dehydrogenase