CYP3A/CYP450

CYP3A4 is an enzyme of cytochrome P450 superfamily found in human liver. It catalyzes the metabolism of endogenous and exogenous agents ( e.g. xenobiotics).

Cat.No. 产品名称 Information
GC10762 4β-hydroxy Cholesterol An oxysterol
GC14618 PPOH Selective inhibitor of epoxygenation reactions catalyzed by CYP4A2 and CYP4A3
GC10778 DDMS A potent inhibitor of 20-HETE synthesis
GC11731 4-phenyl-1,2,3-Thiadiazole Selective inhibitor of CYP2B4 and CYP2E1
GC11864 6,7-dihydroxy Bergamottin A potent CYP3A4 inhibitor
GC16550 Diosmetin A flavonoid with diverse biological activities
GC13784 7-Ethoxyresorufin A fluorogenic substrate for, and inhibitor of, CYP1A1
GC16777 YM 511 YM 511 是一种高度特异性的非甾体芳香酶抑制剂。
GC10554 3-Cyano-7-ethoxycoumarin A fluorogenic CYP450 substrate
GC15445 TMS A potent inhibitor of CYP1B1
GC17552 Pentoxyresorufin A fluorogenic substrate for CYP enzymes
GC10886 Methoxyresorufin A fluorogenic CYP1A1/2 substrate
GC14781 ABT (1-Aminobenzotriazole) A non-specific CYP inhibitor
GC14382 VT-464 R enantiomer CYP17 lyase inhibitor
GC16073 Dronedarone An antiarrhythmic agent
GC16754 Clarithromycin A macrolide antibiotic
GC13079 Voriconazole A triazole antifungal agent
GC14269 Cobicistat (GS-9350) An inhibitor of CYP3A