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Hydrolase(水解酶)

  1. Cat.No. 产品名称 Information
  2. GP26151 FOLH1 Human FOLH1 produced in Sf9 Baculovirus cells is a single, glycosylated polypeptide chain containing 717 amino acids (44-750 a
  3. GP26130 BLMH Mouse BLMH Mouse Recombinant produced in E
  4. GC66450 sEH inhibitor-7 sEH inhibitor-7 (compound c-2) 是一种可溶性环氧化物水解酶 (sEH) 抑制剂,IC50 分别为 0.15 μM (mouse sEH)和6.2 μM (human sEH)。可溶性环氧化物水解酶 (sEH) 在调节血压和炎症的内源性化学介质的代谢中起着重要作用。
  5. GC62743 (Rac)-EC5026 (Rac)-EC5026 ((Rac)-BPN-19186) 是一种有效的可溶性环氧水解酶 (sEH) 抑制剂,Ki 值为 0.06 nM。详细信息请参考专利文献 WO2019156991A1 中的第 39 页。(Rac)-EC5026 可用于帕金森氏病和路易体痴呆 (DLB) 的研究。
  6. GC60073 BI-1935 BI-1935 是一种有效的可溶性环氧化物水解酶 (sEH) 抑制剂,用于与心血管疾病相关的疾病。
  7. GC39221 1-Cyclohexyl-3-dodecyl urea 1-Cyclohexyl-3-dodecyl urea (CDU, N-Cyclohexyl-N-dodecyl urea, NCND) is a highly selective inhibitor of soluble epoxide hydrolase (sEH) that increases epoxyeicosatrienoic acids (EETs) levels.
  8. GC10828 N,N'-Dicyclohexylurea A selective sEH inhibitor
  9. GC12755 trans-AUCB A potent, orally bioavailable sEH inhibitor
  10. GC15387 TPPU

    TPPU是一种可溶性环氧化物水解酶(sEH)抑制剂,对猴和人sEH的IC50值分别为37和3.7 nM。TPPU具有抗炎、镇痛、抗动脉粥样硬化和降压作用。

  11. GC10868 6,7-Dimethyltetrahydropterin (hydrochloride) GTP cyclohydrolase I inhibitor
  12. GC15209 WWL123 A selective inhibitor of ABHD6
  13. GC12150 ML-211 A dual inhibitor of lysophospholipase 1 and 2
  14. GC12043 CUDA A potent inhibitor of soluble epoxide hydrolase
  15. GC13763 KT203 A potent inhibitor of ABHD6
  16. GC16756 KT182 A potent inhibitor of ABHD6
  17. GC14713 3-Deazaadenosine

    Inhibitor of S-adenosylhomocysteine hydrolase

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