Hydrolase(水解酶)
- Cat.No. 产品名称 Information
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GP26151
FOLH1 Human
FOLH1 produced in Sf9 Baculovirus cells is a single, glycosylated polypeptide chain containing 717 amino acids (44-750 a
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GP26130
BLMH Mouse
BLMH Mouse Recombinant produced in E
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GC66450
sEH inhibitor-7
sEH inhibitor-7 (compound c-2) 是一种可溶性环氧化物水解酶 (sEH) 抑制剂,IC50 分别为 0.15 μM (mouse sEH)和6.2 μM (human sEH)。可溶性环氧化物水解酶 (sEH) 在调节血压和炎症的内源性化学介质的代谢中起着重要作用。
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GC62743
(Rac)-EC5026
(Rac)-EC5026 ((Rac)-BPN-19186) 是一种有效的可溶性环氧水解酶 (sEH) 抑制剂,Ki 值为 0.06 nM。详细信息请参考专利文献 WO2019156991A1 中的第 39 页。(Rac)-EC5026 可用于帕金森氏病和路易体痴呆 (DLB) 的研究。
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GC60073
BI-1935
BI-1935 是一种有效的可溶性环氧化物水解酶 (sEH) 抑制剂,用于与心血管疾病相关的疾病。
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GC39221
1-Cyclohexyl-3-dodecyl urea
1-Cyclohexyl-3-dodecyl urea (CDU, N-Cyclohexyl-N-dodecyl urea, NCND) is a highly selective inhibitor of soluble epoxide hydrolase (sEH) that increases epoxyeicosatrienoic acids (EETs) levels.
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GC10828
N,N'-Dicyclohexylurea
A selective sEH inhibitor
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GC12755
trans-AUCB
A potent, orally bioavailable sEH inhibitor
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GC15387
TPPU
Potent inhibitor of soluble epoxide hydrolase with good bioavailability
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GC10868
6,7-Dimethyltetrahydropterin (hydrochloride)
GTP cyclohydrolase I inhibitor
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GC15209
WWL123
A selective inhibitor of ABHD6
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GC12150
ML-211
A dual inhibitor of lysophospholipase 1 and 2
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GC12043
CUDA
A potent inhibitor of soluble epoxide hydrolase
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GC13763
KT203
A potent inhibitor of ABHD6
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GC16756
KT182
A potent inhibitor of ABHD6
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GC14713
3-Deazaadenosine
Inhibitor of S-adenosylhomocysteine hydrolase