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Home >> Signaling Pathways >> Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel(跨膜转运)

Cat.No. 产品名称 Information
GC15898 BzATP triethylammonium salt
2-3-(4-苯甲酰苯甲酰)腺苷5-三磷酸三乙铵盐
An activator of P2X purinergic receptors
GC10953 Tetraethylammonium chloride
四乙基氯化铵
Tetraethylammonium chloride 是一种非选择性钾通道阻滞剂。
GC10152 RO-3 A dual P2X₃ and P2X_2/3 receptor antagonist
GC11600 Valerenic acid
缬草素,(-)-Valerenic Acid
Valerenic acid ((-)-Valerenic Acid) 是一种倍半萜类化合物，是一种具有口服活性的 GABAA 受体正变构调节剂。
GC11195 Sarcosine
肌氨酸; N-Methylglycine; Sarcosin
An intermediate in the biosynthesis of glycine
GC10835 NBMPR
S-(4-硝基苄基)-6-硫代肌苷,NBMPR
A nucleoside transport inhibitor
GC10874 Fumitremorgin C
烟曲酶毒素C; 12α-Fumitremorgin C
Inhibitor of BCRP multidrug transporter
GC16937 Carbamoylcholine chloride
Carbachol

Cholinergic receptor agonist
GC12608 ω-Agatoxin TK ω-Agatoxin TK 是 Agelenopsis aperta 毒液的肽基毒素，是一种有效的选择性 P/Q 型 Ca2+ 通道阻滞剂。
GC15513 ω-Agatoxin IVA
OMEGA-漏斗网蛛毒素IVA
A P-type calcium channel blocker
GC13349 Naspm trihydrochloride
N-[3-[[4-[(3-氨基丙基)氨基]丁基]氨基]丙基]-1-萘乙酰胺三盐酸盐,1-Naphthylacetyl spermine trihydrochloride
A synthetic analog of Joro spider toxin
GC16795 DCA
二氯乙酸钠
DCA 是癌细胞中的代谢调节剂'；具有抗癌活性的线粒体。 DCA 抑制 PDHK，导致肿瘤微环境中的乳酸减少。 DCA 增加活性氧 (ROS) 生成并促进癌细胞凋亡。 DCA 也可作为 NKCC 抑制剂。
GC14712 ACET
UBP316
ACET (ACET) 是一种高效的选择性红藻氨酸受体 GluK1 (GluR5) 拮抗剂，Kb 值为 1.4 nM。
GC17027 POM 1
聚钨酸钠,Sodium polyoxotungstate; POM-1
POM 1是一种核苷三磷酸二磷酸水解酶（NTPDase）抑制剂，对NTPDase1（CD39）、NTPDase3和NTPDase2的K_i值分别为2.58μM、3.26μM和28.8μM。
GC12357 Pentylenetetrazole
戊四唑
A seizure-inducing compound
GC14326 Calmidazolium chloride
钙调蛋白抑制剂,R 24571
An inhibitor of calmodulin
GC12090 Nonactin
无活菌素; Ammonium ionophore I
A mixture of macrotetralide antibiotics that act as ionophores
GC17355 TNP-ATP triethylammonium salt An antagonist of P2X₁, P2X₃, and P2X_2/3 receptors and a fluorescent probe
GC17495 QX 314 chloride
N-Ethyllidocaine
A selective sodium channel blocker
GC16911 CGS 9343B
CGS-9343B; KW 5617
A calmodulin inhibitor
GC13735 (±)-HIP-B
excitatory amino acid transporter (EAAT) blocker
GC11138 (±)-HIP-A excitatory amino acid transporter (EAAT) blocker
GC15417 STEARDA
N-[2-(3,4-二羟基苯基)乙基]十八烷酰胺
potentiates TRPV1-mediated effects of NADA
GC16700 PALDA
PALDA
A naturally-occurring N-acyl dopamine
GC12359 Hispidulin
高车前素; Dinatin
A flavonoid with diverse biological activities
GC10844 SCS
亚水杨基水杨基肼
GABAA receptor antagonist
GC15446 Ionomycin free acid
离子霉素,SQ23377

Ionomycin free acid 是一种选择性的强效钙离子载体，可作为活性 Ca2+ 载体。
GC11082 Paxilline
蕈青霉素
Paxilline是一种致震颤真菌生物碱,可有效抑制高电导Ca2+ 激活K+ (BK)通道,IC50约为10nM,Ki=1.9nM。
GC10351 SR 33805 oxalate Ca2+ channel antagonist
GC15467 ALX 5407 hydrochloride
N-[(3R)-3-([1,1'-联苯]-4-基氧)-3-(4-氟苯基)丙基]-N-甲基甘氨酸盐酸盐
An inhibitor of GlyT1
GC15099 Autocamtide-2-related inhibitory peptide A CaMKII inhibitor
GC14893 Apamin
蜂毒明肽,Apamine
An inhibitor of K_Ca2.2/SK2 channels
GC11483 8-CPT-2Me-cAMP, sodium salt
8-CPT-2MecAMP, 8-pCPTcAMP, 8-pCPT-2′-OMe-cAMP
A selective super-activator of Epacs
GC10188 6'-Iodoresiniferatoxin TRPV1 (VR1) vanilloid receptor partial agonist
GC16832 Suramin hexasodium salt
苏拉明钠; Suramin hexasodium salt
苏拉明六钠盐是一种具有多种生物活性的多磺化萘脲。
GC11293 PPAHV
vanilloid TRPV1 (VR1) receptor agonist
GC16766 Ruthenium Red
钌红; Ammoniated ruthenium oxychloride
A polycationic dye that blocks Ca²⁺ release
GC16801 5'-Iodoresiniferatoxin TRPV1 (VR1) receptor antagonist
GC15900 UCL 1684 UCL 1684（二溴化物）是第一个纳摩尔、非肽类小电导钙激活钾 (SK) 通道阻滞剂。
GC11587 Ochratoxin A
赭曲霉素,Phe-OTA

A mycotoxin
GC17225 ARL 67156 trisodium salt
FPL 67156 trisodium
ARL67156 (FPL 67156) trisodium 是一种选择性 ecto-ATPase 抑制剂。
GC14484 (-)-Xestospongin C
XeC, Araguspongine E
A membrane-permeable antagonist of the inositol-1,4,5-triphosphate receptor
GC10043 D-CPP-ene NMDA antagonist
GC14664 BHQ
2,5-二特丁基对苯二酚
间接食品添加剂 BHQ (DTBHQ) 调节 5-脂氧合酶的活性以及 COX-2 的活性（IC50=1.8 和 14.1 ⋼；M 分别代表 5-LO 和 COX-2）。
GC11200 A23187
离子载体(钙镁盐混合物),Calcimycin

A23187自由酸是一种Ca2+离子载体。
GC11482 Thapsigargin
毒胡萝卜素
他普西加林是一种肌浆网/内质网Ca2+ ATP酶泵的抑制剂。
GC12783 Resiniferatoxin Resiniferatoxin (RTX)是一种超强辣椒素类似物,是一种结合瞬时受体电位通道,香草蛋白亚家族成员1 (TRPV1)的香草蛋白激动剂。
GC17272 Charybdotoxin
卡律(布德)蝎毒素
A blocker of K+ channels
GC16254 Iberiotoxin
IBERIOTOXIN毒素肽
Selective blocker of K_Ca1.1/BK channels
GC14157 (-)-Lobeline hydrochloride
盐酸洛贝林; α-Lobeline hydrochloride; L-Lobeline hydrochloride
An alkaloid with diverse biological activities