Neuroscience(神经科学)

Neuroscience
Neurons communicate with each other, effector organs and sensory organs through the neurotransmitter – receptor pathway at synapses. Neurotransmitters can be divided into 4 major groups: 1. Amino acids (glumate, aspartate, serine, glycine and GABA); 2. Monoamines (norepinephrine, epinephrine, dopamine, histamine, and serotonin); 3. Peptides (opioid peptides, substance P, somatostatin); and 4. Others (acetylcholine, NO, nucleosides). read more
Products for Neuroscience
- 5-HT Receptor(420)
- AChR(53)
- AChE(100)
- Alzheimer(107)
- Amyloid β(118)
- BACE(4)
- CGRP (33)
- COX(294)
- DAPK(7)
- Dopamine Receptor(290)
- GABA Receptor(155)
- Gap Junction(16)
- GluR(116)
- Histamine(2)
- Histamine Receptor(236)
- mPEGS-1(4)
- Muscarinic Receptor(41)
- Neuroscience Peptides(38)
- Nicotinic Receptor(62)
- P2 Receptor(2)
- P2X7 receptor(3)
- SSRIs(5)
- Substance P/NK1 Receptor(20)
- NMDA(2)
- Beta-secretase(25)
- CaMK(32)
- Dopamine Transporter(20)
- Monoamine Oxidase(91)
- Serotonin Transporter(57)
- nAChR(100)
- iGluR(155)
- Neurokinin Receptor(75)
- MCHR1 (GPR24)(16)
- mAChR(183)
- GPR139(4)
- Cholecystokinin Receptor(25)
- Behavioral Neuroscience(353)
- DREADD(1)
- Huntington(14)
- Neuroendocrinology(64)
- Neuroprotection(117)
- Ophthalmology(158)
- Pain Research(229)
- Parkinson(73)
- Prion(7)
- Seizure Disorders(94)
- Cholinesterases(13)
- Tau Protein(4)
- Neurodegenerative Disorders(5)
- Cholinesterase (ChE)(3)
- Amyloid-β(9)
- γ-secretase(1)
- Ischemia(3)
- Cat.No. 产品名称 Information
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GC30904
Molindone hydrochloride (EN-1733A)
EN-1733A
A dopamine receptor antagonist -
GC30902
Dimenhydrinate
乘晕宁
Dimenhydrinate is an over-the-counter drug used to prevent nausea, vomiting, and dizziness caused by motion sickness. -
GC30901
Scopolamine N-oxide hydrobromide (Hyoscine N-oxide hydrobromide)
东莨菪碱N-氧化物氢溴酸盐一水合物
Scopolamine N-Oxide (Hyoscine N-oxide, Genoscopolamine) is a muscarinic antagonist used to study binding characteristics of muscarinic cholinergic receptors.
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GC30898
6-Methylflavone
6-甲基黄酮
6-methylflavone是α1β2γ2L和α1β2GABAA受体的激活剂。 -
GC30892
Glutaminyl Cyclase Inhibitor 1
GlutaminylCyclaseInhibitor1是谷氨酰胺酰基环化酶(glutaminylcyclase)抑制剂,IC50值为0.5μM。
-
GC30889
(-)-Securinine
一叶秋碱
An alkaloid -
GC30888
8-OH-DPAT (8-Hydroxy-DPAT)
8-Hydroxy-DPAT
8-OH-DPAT 是5-HT1A 激动剂, pIC50 值为 8.19 ,此外8-OH-DPAT对5-HT1B(pIC50 , 5.42)和5-HT (pIC50 <5)受体亲和力都很弱 。
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GC30884
LX2343
An inhibitor of BACE1 and PI3K
-
GC30880
LP-211
An agonist of 5-HT7 receptors
-
GC30876
PF-06751979
PF-06751979是一种有效的,脑渗透性的β-淀粉样前体蛋白裂解酶1(BACE1)抑制剂,IC50为7.3nM。
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GC30871
Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride)
6-羟基多巴胺盐酸盐; 6-Hydroxydopamine hydrochloride; 6-OHDA hydrochloride
Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride)(6-OHDA)是神经递质多巴胺的拮抗剂。 -
GC30870
Nialamide
烟肼酰胺
Nialamide是一种非选择性的,不可逆的单胺氧化酶抑制剂(MAOI),用作抗抑郁药。
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GC30866
Anabasine ((S)-Anabasine)
(+)-假木贼碱; (S)-Anabasine; (+)-Anabasine
Anabasine ((S)-Anabasine) ((S)-Anabasine ((S)-Anabasine)) 是一种生物碱,在烟草 (Nicotiana) 中是一种微量成分。 -
GC30865
TPA 023
TPA023是GABAAα2/α3的选择性的激动剂,Ki值为0.19-0.41nM。
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GC30862
L-Cycloserine ((S)-4-Amino-3-isoxazolidone)
环丝氨酸,(S)-Cycloserine; (S)-4-Amino-3-isoxazolidone
An inhibitor of sphingolipid synthesis and aminotransferases -
GC30861
Pavinetant (MLE-4901)
MLE-4901; AZD2624; AZD4901
An NK3 receptor antagonist -
GC30860
Neu2000
Salfaprodil free base; Neu2000
Neu2000 (Salfaprodil free base) 是 N-甲基-D-天冬氨酸 (NMDA) 的 NR2B 选择性和非竞争性拮抗剂。 -
GC30859
AC260584
AC260584是M1毒蕈碱受体变构激动剂,pEC50值为7.6。
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GC30856
Protriptyline hydrochloride
盐酸普罗替林
A tricyclic antidepressant
-
GC30854
Pridopidine (ACR16)
4-[3-(甲磺酰基)苯基]-1-丙基哌啶,ACR16; ASP2314; FR310826
Pridopidine (ACR16, ASP2314, FR310826) , a dopamine (DA) stabilizer, acts as an antagonist against sigma 1 receptor (S1R) and dopamine D2 receptor (D2R). -
GC30852
Org-26576
Org26576是AMPA受体的正变构调节剂。
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GC30849
DREADD agonist 21
A muscarinic hM3Dq DREADD agonist
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GC30848
(+)-PD 128907 hydrochloride
(+)-PD128907,盐酸盐
A potent D3 receptor agonist
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GC30847
IC87201
An inhibitor of the nNOS-PSD-95 protein-protein interaction
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GC30844
Afloqualone
氟喹酮; HQ-495
An Analytical Reference Standard -
GC30840
Quinagolide hydrochloride (CV205-502 hydrochloride)
盐酸喹高利特; CV205-502 hydrochloride
Quinagolide hydrochloride (CV205-502 hydrochloride) 是一种选择性多巴胺 D2 受体激动剂,也是一种催乳素抑制剂。
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GC30839
Traxoprodil
曲索罗地
An antagonist of NR2B subunit-containing NMDA receptors
-
GC30836
MK-7622 (M1 receptor modulator)
3-[(1S,2S)-2-羟基环己基]-6-[(6-甲基-3-吡啶基)甲基]苯并[H]喹唑啉-4(3H)-酮,M1 receptor modulator
A positive allosteric modulator of M1 mAChRs -
GC30835
Rislenemdaz (MK-0657)
MK-0657; CERC-301
Rislenemdaz (MK-0657) (CERC-301) 是一种口服生物可利用的选择性 N-甲基-D-天冬氨酸 (NMDA) 受体亚基 2B (GluN2B) 拮抗剂,其 Ki 和 IC 50 分别为 8.1 nM 和 3.6 nM。
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GC30827
Pipequaline (PK-8165)
哌夸林,PK-8165
A partial agonist of central benzodiazepine receptors -
GC30826
Temanogrel (APD791)
APD791
Temanogrel (APD791) 是一种高度选择性的 5-HT2A 受体拮抗剂,Ki 为 4.9 nM。 -
GC30824
Veralipride ((±)-Veralipride)
维拉必利,(±)-Veralipride; LIR166
Veralipride ((±)-Veralipride) 是一种 D2 受体拮抗剂。
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GC30823
Edonerpic maleate (T-817 maleate)
1-(3-(2-(苯并[B]噻吩-5-基)乙氧基)丙基)氮杂环丁烷-3-醇马来酸,T-817 maleate; T-817MA
T-817MA propyl}-3-azetidinol maleate] 是一种新合成的阿尔茨海默病 (AD) 治疗剂,具有神经保护作用β-淀粉样肽 (Aβ) 的毒性和促进神经突生长的作用.T-817MA 预处理 24 小时后,T-817MA 在 0.1 和 1 uM 时显着防止 H2O2 处理引起的神经元损伤。 -
GC30822
Solifenacin (YM905)
索利那新; YM905 free base
Solifenacin (YM905) is a competitive muscarinic receptor antagonist. The binding of acetylcholine to these receptors, particularly the M3 receptor subtype, plays a critical role in the contraction of smooth muscle.
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GC30821
JNJ-39758979
JNJ-39758979是一个有选择性且具有高亲和性的组胺H4受体拮抗剂,其Ki值为12.5nM。
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GC30818
ZL006
An nNOS/PSD-95 interaction inhibitor
-
GC30812
Imidafenacin (KRP-197)
咪达那新; KRP-197; ONO-8025
Imidafenacin (KRP-197, ONO-8025) is a urinary antispasmodic of the anticholinergic class. It is a novel antimuscarinic agent with safety and efficacy, has been clinically used for the treatment of overactive bladder. Imidafenacin(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM). IC50 value: 0.3 nM(M3). -
GC30810
Donepezil (E2020)
多奈哌齐; E2020 free base
Donepezil (E2020)是一种乙酰胆碱酯酶(AChE)抑制剂,IC50为6.7nM。 -
GC30809
VU0467154
5-氨基-3,4-二甲基-噻吩并[2,3-C]哒嗪-6-羧酸4-三氟甲磺酰基-苄基酰胺
A positive allosteric modulator of the M4 muscarinic acetylcholine receptor -
GC30807
ZSET1446 (ST-101)
ST-101
ZSET1446 (ST-101) 是一种新型认知增强剂,可显着改善各种类型的阿尔茨海默病 (AD) 模型中的学习缺陷。 -
GC30797
lumateperone Tosylate (ITI-007)
1-(4-氟苯基)-4-[(6BR,10AS)-2,3,6B,9,10,10A-六氢-3-甲基-1H-吡啶并[3',4':4,5]吡咯并[1,2,3-DE]喹喔啉-8(7H)-基]-1-丁酮对甲苯磺酸盐,ITI-007 tosylate
An atypical antipsychotic
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GC30796
Nelotanserin (APD125)
1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲,APD125
Nelotanserin (APD125) 是一种有效的 5-HT2A 反向激动剂、中度有效的 5-HT2C 部分反向激动剂和弱 5-HT2B 反向激动剂,在 IP 积累试验中 IC50 分别为 1.7、79、791 nM。 -
GC30790
Triflupromazine hydrochloride
盐酸三氟丙嗪
A phenothiazine with diverse biological activities -
GC30788
L-Glutamic acid monosodium salt (Monosodium glutamate)
谷氨酸单钠盐
L-Glutamic acid monosodium salt is the sodium salt of glutamic acid, found naturally in tomatoes, cheese and other foods. L-Glutamic acid monosodium salt acts as an excitatory transmitter and an agonist at all subtypes of glutamate receptors (metabotropic, kainate, NMDA, and AMPA). (S)-Glutamic acid shows a direct activating effect on the release of DA from dopaminergic terminals. -
GC30787
Sertindole (Lu 23-174)
舍吲哚; Lu 23-174
An atypical antipsychotic -
GC30780
Fipexide
非哌西特
Fipexide (hydrochloride) is a psychoactive drug of the piperazine class. -
GC30775
Histamine (Ergamine)
组胺; Ergamine
A biogenic amine
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GC30774
Tat-NR2B9c
Tat-NR2Bct; NA-1
Tat-NR2B9c 旨在通过阻止突触后密度蛋白 95 (PSD-95) 与 N-甲基-D-天冬氨酸 (NMDA) 受体和神经元一氧化氮结合来阻止一氧化氮 (NO) 的产生氧化物合成酶。 -
GC30773
Phenelzine sulfate
硫酸苯乙肼
An inhibitor of MAO -
GC30772
Dopamine serotonin antagonist-1
氯氮平杂质,Deschloroclozapine
Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs (muscarinic Designer Receptors Exclusively Activated by Designer Drugs) agonist, and binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively.