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Neuroscience(神经科学)

Neuroscience

Neurons communicate with each other, effector organs and sensory organs through the neurotransmitter – receptor pathway at synapses. Neurotransmitters can be divided into 4 major groups: 1. Amino acids (glumate, aspartate, serine, glycine and GABA); 2. Monoamines (norepinephrine, epinephrine, dopamine, histamine, and serotonin); 3. Peptides (opioid peptides, substance P, somatostatin); and 4. Others (acetylcholine, NO, nucleosides). read more

Products for  Neuroscience

  1. Cat.No. 产品名称 Information
  2. GC30904 Molindone hydrochloride (EN-1733A)

    EN-1733A

    A dopamine receptor antagonist
  3. GC30902 Dimenhydrinate

    乘晕宁

    Dimenhydrinate is an over-the-counter drug used to prevent nausea, vomiting, and dizziness caused by motion sickness.
  4. GC30901 Scopolamine N-oxide hydrobromide (Hyoscine N-oxide hydrobromide)

    东莨菪碱N-氧化物氢溴酸盐一水合物

    Scopolamine N-Oxide (Hyoscine N-oxide, Genoscopolamine) is a muscarinic antagonist used to study binding characteristics of muscarinic cholinergic receptors.

  5. GC30898 6-Methylflavone

    6-甲基黄酮

    6-methylflavone是α1β2γ2L和α1β2GABAA受体的激活剂。
  6. GC30892 Glutaminyl Cyclase Inhibitor 1 GlutaminylCyclaseInhibitor1是谷氨酰胺酰基环化酶(glutaminylcyclase)抑制剂,IC50值为0.5μM。
  7. GC30889 (-)-Securinine

    一叶秋碱

    An alkaloid
  8. GC30888 8-OH-DPAT (8-Hydroxy-DPAT)

    8-Hydroxy-DPAT

    8-OH-DPAT 是5-HT1A 激动剂, pIC50 值为 8.19 ,此外8-OH-DPAT对5-HT1B(pIC50 , 5.42)和5-HT (pIC50 <5)受体亲和力都很弱 。

  9. GC30884 LX2343 An inhibitor of BACE1 and PI3K
  10. GC30880 LP-211 An agonist of 5-HT7 receptors
  11. GC30876 PF-06751979 PF-06751979是一种有效的,脑渗透性的β-淀粉样前体蛋白裂解酶1(BACE1)抑制剂,IC50为7.3nM。
  12. GC30871 Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride)

    6-羟基多巴胺盐酸盐; 6-Hydroxydopamine hydrochloride; 6-OHDA hydrochloride

    Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride)(6-OHDA)是神经递质多巴胺的拮抗剂。
  13. GC30870 Nialamide

    烟肼酰胺

    Nialamide是一种非选择性的,不可逆的单胺氧化酶抑制剂(MAOI),用作抗抑郁药。

  14. GC30866 Anabasine ((S)-Anabasine)

    (+)-假木贼碱; (S)-Anabasine; (+)-Anabasine

    Anabasine ((S)-Anabasine) ((S)-Anabasine ((S)-Anabasine)) 是一种生物碱,在烟草 (Nicotiana) 中是一种微量成分。
  15. GC30865 TPA 023 TPA023是GABAAα2/α3的选择性的激动剂,Ki值为0.19-0.41nM。
  16. GC30862 L-Cycloserine ((S)-4-Amino-3-isoxazolidone)

    环丝氨酸,(S)-Cycloserine; (S)-4-Amino-3-isoxazolidone

    An inhibitor of sphingolipid synthesis and aminotransferases
  17. GC30861 Pavinetant (MLE-4901)

    MLE-4901; AZD2624; AZD4901

    An NK3 receptor antagonist
  18. GC30860 Neu2000

    Salfaprodil free base; Neu2000

    Neu2000 (Salfaprodil free base) 是 N-甲基-D-天冬氨酸 (NMDA) 的 NR2B 选择性和非竞争性拮抗剂。
  19. GC30859 AC260584 AC260584是M1毒蕈碱受体变构激动剂,pEC50值为7.6。
  20. GC30856 Protriptyline hydrochloride

    盐酸普罗替林

    A tricyclic antidepressant

  21. GC30854 Pridopidine (ACR16)

    4-[3-(甲磺酰基)苯基]-1-丙基哌啶,ACR16; ASP2314; FR310826

    Pridopidine (ACR16, ASP2314, FR310826) , a dopamine (DA) stabilizer, acts as an antagonist against sigma 1 receptor (S1R) and dopamine D2 receptor (D2R).
  22. GC30852 Org-26576 Org26576是AMPA受体的正变构调节剂。
  23. GC30849 DREADD agonist 21 A muscarinic hM3Dq DREADD agonist
  24. GC30848 (+)-PD 128907 hydrochloride

    (+)-PD128907,盐酸盐

    A potent D3 receptor agonist

  25. GC30847 IC87201 An inhibitor of the nNOS-PSD-95 protein-protein interaction
  26. GC30844 Afloqualone

    氟喹酮; HQ-495

    An Analytical Reference Standard
  27. GC30840 Quinagolide hydrochloride (CV205-502 hydrochloride)

    盐酸喹高利特; CV205-502 hydrochloride

    Quinagolide hydrochloride (CV205-502 hydrochloride) 是一种选择性多巴胺 D2 受体激动剂,也是一种催乳素抑制剂。

  28. GC30839 Traxoprodil

    曲索罗地

    An antagonist of NR2B subunit-containing NMDA receptors

  29. GC30836 MK-7622 (M1 receptor modulator)

    3-[(1S,2S)-2-羟基环己基]-6-[(6-甲基-3-吡啶基)甲基]苯并[H]喹唑啉-4(3H)-酮,M1 receptor modulator

    A positive allosteric modulator of M1 mAChRs
  30. GC30835 Rislenemdaz (MK-0657)

    MK-0657; CERC-301

    Rislenemdaz (MK-0657) (CERC-301) 是一种口服生物可利用的选择性 N-甲基-D-天冬氨酸 (NMDA) 受体亚基 2B (GluN2B) 拮抗剂,其 Ki 和 IC 50 分别为 8.1 nM 和 3.6 nM。

  31. GC30827 Pipequaline (PK-8165)

    哌夸林,PK-8165

    A partial agonist of central benzodiazepine receptors
  32. GC30826 Temanogrel (APD791)

    APD791

    Temanogrel (APD791) 是一种高度选择性的 5-HT2A 受体拮抗剂,Ki 为 4.9 nM。
  33. GC30824 Veralipride ((±)-Veralipride)

    维拉必利,(±)-Veralipride; LIR166

    Veralipride ((±)-Veralipride) 是一种 D2 受体拮抗剂。

  34. GC30823 Edonerpic maleate (T-817 maleate)

    1-(3-(2-(苯并[B]噻吩-5-基)乙氧基)丙基)氮杂环丁烷-3-醇马来酸,T-817 maleate; T-817MA

    T-817MA propyl}-3-azetidinol maleate] 是一种新合成的阿尔茨海默病 (AD) 治疗剂,具有神经保护作用β-淀粉样肽 (Aβ) 的毒性和促进神经突生长的作用.T-817MA 预处理 24 小时后,T-817MA 在 0.1 和 1 uM 时显着防止 H2O2 处理引起的神经元损伤。
  35. GC30822 Solifenacin (YM905)

    索利那新; YM905 free base

    Solifenacin (YM905) is a competitive muscarinic receptor antagonist. The binding of acetylcholine to these receptors, particularly the M3 receptor subtype, plays a critical role in the contraction of smooth muscle.

  36. GC30821 JNJ-39758979 JNJ-39758979是一个有选择性且具有高亲和性的组胺H4受体拮抗剂,其Ki值为12.5nM。
  37. GC30818 ZL006 An nNOS/PSD-95 interaction inhibitor
  38. GC30812 Imidafenacin (KRP-197)

    咪达那新; KRP-197; ONO-8025

    Imidafenacin (KRP-197, ONO-8025) is a urinary antispasmodic of the anticholinergic class. It is a novel antimuscarinic agent with safety and efficacy, has been clinically used for the treatment of overactive bladder. Imidafenacin(KRP-197; ONO-8025) is a potent and selective inhibitor of M3 receptors with Kb of 0.317 nM; less potent for M2 receptors(IC50=4.13 nM). IC50 value: 0.3 nM(M3).
  39. GC30810 Donepezil (E2020)

    多奈哌齐; E2020 free base

    Donepezil (E2020)是一种乙酰胆碱酯酶(AChE)抑制剂,IC50为6.7nM。
  40. GC30809 VU0467154

    5-氨基-3,4-二甲基-噻吩并[2,3-C]哒嗪-6-羧酸4-三氟甲磺酰基-苄基酰胺

    A positive allosteric modulator of the M4 muscarinic acetylcholine receptor
  41. GC30807 ZSET1446 (ST-101)

    ST-101

    ZSET1446 (ST-101) 是一种新型认知增强剂,可显着改善各种类型的阿尔茨海默病 (AD) 模型中的学习缺陷。
  42. GC30797 lumateperone Tosylate (ITI-007)

    1-(4-氟苯基)-4-[(6BR,10AS)-2,3,6B,9,10,10A-六氢-3-甲基-1H-吡啶并[3',4':4,5]吡咯并[1,2,3-DE]喹喔啉-8(7H)-基]-1-丁酮对甲苯磺酸盐,ITI-007 tosylate

    An atypical antipsychotic

  43. GC30796 Nelotanserin (APD125)

    1-[3-(4-溴-1-甲基-1H-吡唑-5-基)-4-甲氧基苯基]-3-(2,4-二氟苯基)脲,APD125

    Nelotanserin (APD125) 是一种有效的 5-HT2A 反向激动剂、中度有效的 5-HT2C 部分反向激动剂和弱 5-HT2B 反向激动剂,在 IP 积累试验中 IC50 分别为 1.7、79、791 nM。
  44. GC30790 Triflupromazine hydrochloride

    盐酸三氟丙嗪

    A phenothiazine with diverse biological activities
  45. GC30788 L-Glutamic acid monosodium salt (Monosodium glutamate)

    谷氨酸单钠盐

    L-Glutamic acid monosodium salt is the sodium salt of glutamic acid, found naturally in tomatoes, cheese and other foods. L-Glutamic acid monosodium salt acts as an excitatory transmitter and an agonist at all subtypes of glutamate receptors (metabotropic, kainate, NMDA, and AMPA). (S)-Glutamic acid shows a direct activating effect on the release of DA from dopaminergic terminals.
  46. GC30787 Sertindole (Lu 23-174)

    舍吲哚; Lu 23-174

    An atypical antipsychotic
  47. GC30780 Fipexide

    非哌西特

    Fipexide (hydrochloride) is a psychoactive drug of the piperazine class.
  48. GC30775 Histamine (Ergamine)

    组胺; Ergamine

    A biogenic amine

  49. GC30774 Tat-NR2B9c

    Tat-NR2Bct; NA-1

    Tat-NR2B9c 旨在通过阻止突触后密度蛋白 95 (PSD-95) 与 N-甲基-D-天冬氨酸 (NMDA) 受体和神经元一氧化氮结合来阻止一氧化氮 (NO) 的产生氧化物合成酶。
  50. GC30773 Phenelzine sulfate

    硫酸苯乙肼

    An inhibitor of MAO
  51. GC30772 Dopamine serotonin antagonist-1

    氯氮平杂质,Deschloroclozapine

    Deschloroclozapine, a metabolite of Clozapine, is a highly potent muscarinic DREADDs (muscarinic Designer Receptors Exclusively Activated by Designer Drugs) agonist, and binds to DREADD receptor subtypes hM3Dq and hM4Di with Ki of 6.3 and 4.2 nM, respectively.

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