Muscarinic Receptor(毒蕈碱受体)
Muscarinic receptor is a group of G-protein coupled receptors that binds to acetylcholine and mediates cellular responses, including inhibition of acetylate cyclase, phosphoinositide degradation and regulation of potassium channels. It is involved in the neurological diseases such as Alzheimer's and Parkinson's.
- Cat.No. 产品名称 Information
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GC12787
Aceclidine (hydrochloride)
A muscarinic receptor agonist
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GC10378
N-Isopropylnoratropine
An intermediate in the synthesis of ipratropium
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GC15758
BQCA
A positive allosteric modulator of the M1 mAChR
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GC15845
Guvacoline (hydrobromide)
A muscarinic receptor agonist
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GC12311
Trihexyphenidyl hydrochloride
A muscarinic M1 receptor antagonist
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GC14508
PTAC oxalate
muscarinic receptor ligand
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GC17821
VU 0365114
A positive allosteric modulator of muscarinic M5 receptors
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GC16655
VU 0357017 hydrochloride
An M1 muscarinic acetylcholine receptor agonist
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GC10464
VU 0255035
A selective muscarinic M1 receptor antagonist
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GC15990
VU 0238429
A muscarinic M5 receptor positive allosteric modulator
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GC10725
VU 10010
VU 10010 是一种有效的、高选择性的变构 M4 mAChR 增强剂,EC50 为 400 nM。
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GC14619
Milameline hydrochloride
Muscarinic receptor agonist
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GC18082
Zamifenacin fumarate
A muscarinic M3 receptor antagonist
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GC13340
AQ-RA 741
M2 antagonist,selective and high affinity
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GC10633
DAU 5884 hydrochloride
muscarinic M3 receptor antagonist
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GC17876
PD 102807
PD 102807 是一种 M4 毒蕈碱受体拮抗剂,IC50 为 90.7 nM。
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GC14479
(S)-(+)-Dimethindene maleate
(S)-(+)-Dimethindene maleate 是一种对映异构体,是一种有效的 M2 选择性毒蕈碱受体拮抗剂 (pA2 =7.86/7.74; pKi =7.78)。
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GC16458
McN-A 343
A partial agonist of muscarinic acetylcholine receptors
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GC15510
AF-DX 384
An M2 and M4 muscarinic acetylcholine receptor antagonist
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GC13174
Telenzepine dihydrochloride
Telenzepine dihydrochloride 是一种选择性和口服活性的毒蕈碱 M1 受体拮抗剂,Ki 为 0.94 nM。
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GC10219
AF-DX 116
A muscarinic M2 receptor antagonist
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GC13129
W-84 dibromide
W-84 (dibromide) 是一种有效的 M2-胆碱受体变构调节剂,可延缓 [3H]N-甲基东莨菪碱的解离。
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GC10525
Nitrocaramiphen hydrochloride
M1 muscarinic antagonist
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GC16504
Arecaidine propargyl ester tosylate
muscarinic receptor agonist
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GC11415
Arecaidine but-2-ynyl ester tosylate
mAChR M2 激动剂
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GC10736
(+)-Muscarine iodide
毒蕈碱 ((+)-Muscarine) 碘化物是一种可以刺激副交感神经系统的毒素。
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GC12056
J 104129 fumarate
M3 muscarinic receptor antagonist
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GC13403
Pirenzepine dihydrochloride
A muscarinic M1 receptor antagonist
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GC16463
Oxotremorine M
A muscarinic receptor agonist and KCNQ2/3 potassium channel blocker
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GC16156
Oxotremorine sesquifumarate
A muscarinic acetylcholine receptor agonist
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GC14604
5-Methylfurmethiodide
muscarinic agonist
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GC13348
4-DAMP
An antagonist of the muscarinic M3 receptor
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GC16087
Fesoterodine Fumarate
A muscarinic acetylcholine receptor antagonist
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GC15772
Darifenacin HBr
A muscarinic M3 receptor antagonist
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GC17182
Solifenacin succinate
A muscarinic M1, M2, and M3 receptor antagonist
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GC17954
Tolterodine tartrate
A muscarinic acetylcholine receptor antagonist
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GC14096
Aclidinium Bromide
A muscarinic acetylcholine receptor antagonist
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GC10621
Biperiden HCl
A muscarinic acetylcholine receptor antagonist
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GC11831
Umeclidinium bromide
A muscarinic acetylcholine receptor antagonist
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GC17157
Cevimeline hydrochloride hemihydrate
Cevimeline hydrochloride hemihydrate (SNI-2011) 是乙酰胆碱的奎宁环衍生物,是一种选择性和口服活性的毒蕈碱 M1 和 M3 受体激动剂。
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GC14215
Cevimeline
A muscarinic receptor agonist