GluR(谷氨酸受体)
GluR (glutamate receptor) is a group of synaptic receptors located primarily on the membranes of neuronal cells.
Products for GluR
- Cat.No. 产品名称 Information
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GC26056
WAY-303290
GluR6 antagonist-1
WAY-303290 (GluR6 antagonist-1) is a benzothiophene derivative acting as an ionotropic glutamate receptor 6 (GluR6) antagonist, which can be used for researching acute and chronic neurological disorders. -
GC18309
LSN2463359
N-异丙基-5-(吡啶-4-基乙炔基)吡啶酰胺
A brain penetrant positive allosteric modulator of the mGluR5 -
GC16247
DCG IV
DCG IV 是 II 组 mGluRs 的有效激动剂,对 mGlu2R 和 mGlu3R 的 EC50 分别为 0.35 和 0.09 μM。
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GC17950
MMPIP hydrochloride
A reversible allosteric antagonist of mGluR7
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GC17932
L-AP4
L(+)-2-氨基-4-膦酰基丁酸,L-APB
A selective Group III metabotropic glutamate receptor agonist -
GC17095
ML 337
ML 337 是一种选择性和脑渗透性的 mGlu3 负变构调节剂,IC50 为 593 nM。
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GC14869
ML 289
VU0463597
A negative allosteric modulator of mGlu3 -
GC10045
MFZ 10-7
MFZ 10-7 是一种有效的 mGluR5 拮抗剂。
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GC12460
ADX 10059 hydrochloride
Negative allosteric modulator at mGlu5
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GC11986
VU 0360223
CAY10651
A negative allosteric modulator of the mGlu5 receptor -
GC10238
MNI 137
MNI 137 是一种有效的、选择性的负变构调节剂,适用于 II 组 mGluR。
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GC16643
VU 0285683
negative allosteric modulator of mGlu5 receptors
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GC11750
TC-N 22A
TC-N 22A 是一种有效的、选择性的、具有口服活性和脑渗透性的 mGlu4 PAM,在表达人 mGlu4 的 BHK 细胞中的 EC50 为 9 nM。
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GC12485
Ro 67-7476
A positive allosteric modulator of mGluR1
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GC10323
VU 0360172 hydrochloride
A positive allosteric modulator of mGluR5
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GC11563
NPS 2390
Type I metabotropic glutamate receptor antagonist
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GC18063
YM 230888
Selective mGlu1 antagonist
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GC12435
ACPT-I
An mGluR4a and mGluR8 agonist
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GC16557
LY 379268 disodium salt
group II mGlu receptor agonist
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GC14722
LY 2389575 hydrochloride
negative allosteric modulator of mGlu3
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GC17289
VU 29
VU 29 是代谢型谷氨酸 5 (mGlu5) 受体的正变构调节剂(对于 rmGluR5,EC50\u003d9 nM 和 Ki\u003d244 nM)。
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GC14383
Ro 01-6128
A positive allosteric modulator of mGLUR1
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GC14172
Ro 67-4853
A positive allosteric modulator of mGlu1 receptors
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GC11501
TCN 238
A positive allosteric modulator of mGluR4
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GC12705
Cinnabarinic acid
朱砂精酸
An agonist of mGluR4 and active metabolite of 3-hydroxyanthranilic acid
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GC12510
BINA
3'-[[(2-环戊基-6,7-二甲基-1-氧代-2,3-二氢-1H-茚-5-基)氧基]甲基]联苯-4-羧酸,BINA
A positive allosteric modulator of mGluR2 -
GC12899
CBiPES hydrochloride
positive allosteric modulator of the mGlu2 receptor
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GC11997
(RS)-MCPG disodium salt
group I/group II metabotropic glutamate receptor antagonist
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GC17963
CHPG Sodium salt
CHPG 钠盐是一种选择性 mGluR5 激动剂,可通过 BV2 小胶质细胞中的 TSG-6/NF-κB 通路减弱 SO2 诱导的氧化应激和炎症。
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GC11970
YM 202074
metabotropic glutamate receptor type 1 (mGlu1) antagonist
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GC17604
NPEC-caged-(1S,3R)-ACPD
group I and II mGlu receptor agonist
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GC11554
NPEC-caged-(S)-3,4-DCPG
mGlu8a agonist
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GC17749
VU 1545
VU 1545 是一种代谢型谷氨酸受体 5 正变构调节剂 (mGluR5 PAM),Ki 为 156 nM,EC50 为 9.6 nM。
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GC14003
VU 0155041 sodium salt
A selective positive allosteric modulator of mGluR4
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GC14097
LY 487379 hydrochloride
LY 487379 hydrochloride 是一种选择性人 mGluR2 正变构调节剂 (PAM)。
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GC12699
(±)-LY 395756
ligand for mGlu2 and mGlu3 receptor
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GC17531
Z-Cyclopentyl-AP4
Group III mGlu receptor agonist
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GC15198
VU 0155041
A selective positive allosteric modulator of mGluR4
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GC10605
LY 354740
(1S,2S,5R,6S)-2-氨基二环[3.1.0]己烷-2,6-二羧酸,LY354740; Eglumetad
An agonist of mGluR2 and mGluR3 -
GC10422
CDPPB
3-氰基-N-(1,3-二苯基吡唑-5-基)苯甲酰胺
A positive allosteric modulator of mGluR5 -
GC16068
A 841720
An mGluR1 antagonist
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GC11704
Ro 64-5229
mGlu2 antagonist
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GC14861
LY 379268
A selective group II mGlu2/3 receptor agonist
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GC15566
YM 298198 hydrochloride
A non-competitive antagonist of mGluR1
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GC13120
Desmethyl-YM 298198
mGlu1-selective antagonist
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GC17492
LY 456236 hydrochloride
mGlu1 receptor antagonist
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GC11766
Fenobam
非诺班
A noncompetitive antagonist and inverse agonist of mGluR5 -
GC11287
AMN 082 dihydrochloride
An allosteric mGluR7 agonist
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GC17217
JNJ 16259685
An antagonist of mGluR1a
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GC17079
ACDPP hydrochloride
mGlu5 receptor antagonist