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GluR(谷氨酸受体)

GluR (glutamate receptor) is a group of synaptic receptors located primarily on the membranes of neuronal cells.

Products for  GluR

  1. Cat.No. 产品名称 Information
  2. GC17079 ACDPP hydrochloride mGlu5 receptor antagonist
  3. GC11223 3-MATIDA mGlu1 receptor antagonist
  4. GC13126 DMeOB Negative allosteric modulator of mGlu5
  5. GC15385 DCB DCB (3,3'-dichlorobenzaldazine) 是代谢型谷氨酸受体代谢型谷氨酸受体亚型 5 (mGluR5) 的中性变构调节剂。
  6. GC10739 (S)-HexylHIBO Group I mGlu receptor antagonist
  7. GC17446 HexylHIBO

    HexylHIBO 是一种有效的 I 组 mGluR 拮抗剂,对 mGlu1a 和 mGlu5a 受体的 Kb 值分别为 140 和 110 μM。

  8. GC11246 DFB A positive allosteric modulator of mGluR5
  9. GC14227 MNI-caged-L-glutamate A caged neurotransmitter used with photolysis
  10. GC17722 (R)-3,4-DCPG AMPA receptor antagonist with weak activity at NMDA receptors and little activity at kainate receptors
  11. GC16542 (RS)-3,4-DCPG antagonist of AMPA receptors and agonist of mGluR8
  12. GC13046 UBP1112 group III mGlu receptor antagonist
  13. GC14639 (S)-3,4-DCPG A selective agonist of mGluR8
  14. GC12831 LY 367385 An antagonist of mGluR1α
  15. GC11433 (RS)-PPG (RS)-PPG 是 III 组 mGluR 的有效选择性激动剂。
  16. GC11233 SIB 1757 An antagonist of mGluR5a
  17. GC10452 SIB 1893 SIB 1893 是 (E)-SIB-1893 和 (Z)-SIB-1893 异构体的外消旋化合物。
  18. GC11379 (2R,4R)-APDC (2R,4R)-APDC 是一种选择性 II 族代谢型谷氨酸受体 (mGluRs) 激动剂。
  19. GC11771 (RS)-APICA (RS)-APICA 是一种选择性 II 组代谢型谷氨酸受体 (mGluR II) 拮抗剂。
  20. GC12532 CHPG A potent and selective mGluR5 agonist
  21. GC18134 CPCCOEt An mGluR1b antagonist
  22. GC17383 PHCCC PHCCC 是 I 组 mGluR 拮抗剂,IC50 为 3 μM。 PHCCC 是 mGlu4 受体的选择性正调节剂。抗帕金森效应。
  23. GC13192 E4CPG An antagonist of mGluR1 and mGluR2
  24. GC12100 CPPG An antagonist of group II and group III mGluRs
  25. GC17326 EGLU EGLU ((2S)-α-Ethylglutamic acid; (2S)-α-EGLU) 是一种有效的竞争性 mGluR-2 受体拮抗剂。
  26. GC14146 AIDA AIDA (AIDA) 是一种刚性(羧基苯基)甘氨酸衍生物,是一种相对有效和选择性的 I 组代谢型谷氨酸受体 (mGlu1a) 拮抗剂,IC50 为 214 μM.
  27. GC11428 MTPG MTPG 是一种有效的 mGluR2 和 mGluR3 拮抗剂。
  28. GC13548 MSPG mGlu receptor antagonist
  29. GC15769 MPPG MPPG 是一种有效的选择性 L-AP4 敏感受体拮抗剂,kD 值为 9.2 μM,正在新生大鼠脊髓上进行测试。
  30. GC16858 (S)-3,5-DHPG A selective agonist of group I mGluRs
  31. GC17185 MSOP MSOP 是一种选择性 III 族代谢型谷氨酸受体拮抗剂,对 L-AP4 敏感的突触前 mGluR 的表观 KD 为 51 μM。
  32. GC11571 MAP4 MAP4 在某些电生理系统中是一种选择性 III 组 mGluR 拮抗剂。
  33. GC11269 Salsolinol-1-carboxylic acid Salsolinol-1-carboxy acid 是中枢神经系统 (CNS) 中的一种内源性生物碱。
  34. GC13222 N-Acetylglycyl-D-glutamic acid Excitatory peptide that induces seizures
  35. GC15136 L-AP6 selective agonist for 'quis'-sensitized site
  36. GC16349 (S)-MCPG An mGluR antagonist
  37. GC12279 (RS)-MCPG (RS)-MCPG (alpha-MCPG) 是一种竞争性和选择性的 I 组/II 组代谢型谷氨酸受体 (mGluR) 拮抗剂。
  38. GC11536 (S)-3-Carboxy-4-hydroxyphenylglycine group I metabotropic glutamate receptor antagonist and group II mGlu agonist
  39. GC14124 (R)-3-Carboxy-4-hydroxyphenylglycine NMDA and AMPA/kainate receptor antagonist
  40. GC16234 (S)-3-Hydroxyphenylglycine group I metabotropic glutamate receptors agonist
  41. GC12985 (RS)-3-Hydroxyphenylglycine PI-linked metabotropic glutamate receptors agonist
  42. GC14176 (S)-4-Carboxyphenylglycine group I metabotropic glutamate receptor antagonist
  43. GC13773 (RS)-4-Carboxyphenylglycine broad spectrum EAA ligand
  44. GC12012 (S)-4-Carboxy-3-hydroxyphenylglycine group I mGlu1a/1a receptor antagonist and mGluR2 agonist
  45. GC13288 (RS)-4-Carboxy-3-hydroxyphenylglycine broad spectrum EAA agonist/antagonist
  46. GC16207 (1S,3R)-ACPD group I and II mGlu receptor agonist
  47. GC14752 2,4-Dihydroxyphenylacetyl-L-asparagine glutamate receptors blocker
  48. GC12394 (±)-trans-ACPD An mGluR agonist
  49. GC10026 S-Sulfo-L-cysteine sodium salt EAA receptor agonist
  50. GC12063 D-AP4 D-AP4 (D-APB; D-2-Amino-4-phosphonobutyric acid) 是一种谷氨酸的膦酰基类似物,是一种 NMDA 广谱兴奋性氨基酸受体拮抗剂。
  51. GC15435 RuBi-Glutamate Ruthenium-bipyridine-trimethylphosphine caged glutamate

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