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Home >> Signaling Pathways >> Neuroscience >> AChR

AChR(乙酰胆碱受体)

AChR, also known as acetylcholine receptor, is an integral membrane protein that responds to the binding of acetylcholine.

  1. Cat.No. 产品名称 Information
  2. GC26093 α-Conotoxin GI α-Conotoxin GI, a 13-residue peptide originally isolated from the venom of the fish-hunting cone snail Conus geographus, acts as a competitive antagonist for the muscle-type nicotinic acetylcholine receptor (nAChR) with excellent selectivity for α/δ receptor subunit binding over α/γ.
  3. GC26032 Varenicline (CP 526555) dihydrochloride Varenicline (CP 526555, Chantix, Champix,CP 526555 dihydrochloride) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation.
  4. GC25994 Thonzylamine Thonzylamine (Neohetramine) is an antihistamine and anticholinergic drug.
  5. GC25583 Lobelin sulphate Lobelin sulphate (Lobeline sulfate, Bantron) is an alkaloid that has actions similar to nicotine on nicotinic cholinergic receptors but is less potent. It has a variety of therapeutic uses including in respiratory disorders, peripheral vascular disorders, insomnia, and smoking cessation.
  6. GC25387 Ethyl (triphenylphosphoranylidene) acetate Ethyl (triphenylphosphoranylidene) acetate (Triphenylcarbethoxymethylenephosphorane, (Carbethoxymethylene)triphenylphosphorane) may act as an inhibitor of cholinesterase that inhibits AChE and BChE.
  7. GC17885 VU0364572 (trifluoroacetate salt) A selective muscarinic M1 receptor agonist
  8. GC13314 L-Acetylcarnitine (hydrochloride) A mitochondrial metabolite
  9. GC12507 ML352 An inhibitor of the presynaptic choline transporter
  10. GC13445 LY2119620 A positive allosteric modulator of M2 and M4 mAChRs
  11. GC17627 Nitenpyram An insecticide
  12. GC11128 (±)-Vesamicol hydrochloride (±)-Vesamicol hydrochloride ((±)-AH5183 hydrochloride) 是一种有效的囊泡乙酰胆碱转运抑制剂，Ki 为 2 nM。
  13. GC13361 Flavoxate hydrochloride An internal standard for the quantification of flavoxate
  14. GC10508 Solifenacin hydrochloride Solifenacin hydrochloride (YM905 hydrochloride) 是一种毒蕈碱受体拮抗剂，对 M1、M2 和 M3 受体的 pKis 分别为 7.6、6.9 和 8.0。
  15. GC14419 Bethanechol chloride A muscarinic acetylcholine receptor agonist
  16. GC14142 Acetylcholine Chloride A neurotransmitter
  17. GC11773 Pancuronium dibromide Pancuronium dibromide 是一种双季铵盐类固醇，是一种神经肌肉松弛剂。
  18. GC10972 Gallamine Triethiodide An allosteric modulator of muscarinic acetylcholine receptors
  19. GC17483 Trospium chloride An antagonist of muscarinic receptors
  20. GC13134 Tiotropium Bromide hydrate A muscarinic receptor antagonist
  21. GC17229 Paroxetine HCl A selective serotonin reuptake inhibitor
  22. GC17825 Methscopolamine A muscarinic acetylcholine receptor antagonist
  23. GC13779 Orphenadrine Citrate Orphenadrine citrate 是一种具有口服活性且非竞争性的 NMDA 受体拮抗剂（穿过血脑屏障），Ki 为 6.0 μM。
  24. GC15150 Tropicamide A selective muscarinic M4 antagonist
  25. GC12453 Succinylcholine Chloride Dihydrate An agonist of muscle-type nAChRs
  26. GC16056 Neostigmine Bromide 溴化新斯的明是一种胆碱酯酶抑制剂，用于治疗重症肌无力。
  27. GC10863 Otilonium Bromide An L- and T-type calcium channel inhibitor and mAChR antagonist
  28. GC11035 Hyoscyamine A muscarinic receptor antagonist
  29. GC17908 Homatropine Methylbromide An anticholinergic agent
  30. GC13897 Homatropine Bromide An anticholinergic agent
  31. GC15178 Hexamethonium Bromide A nondepolarizing neuromuscular blocking agent
  32. GC16255 Decamethonium Bromide A depolarizing neuromuscular blocking agent
  33. GC14703 Oxybutynin chloride An antagonist of muscarinic acetylcholine receptors
  34. GC12920 Pregnenolone A natural steroid hormone
  35. GC11219 (R)-(+)-Tolterodine (R)-(+)-Tolterodine(PNU-200583) 是一种有效的毒蕈碱受体拮抗剂，在体内对膀胱的选择性优于唾液腺。
  36. GC15029 Glycopyrrolate A muscarinic acetylcholine receptor antagonist
  37. GC16059 Tarafenacin D-tartrate Tarafenacin D-tartrate (SVT-40776 D-tartrate) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM)，选择性是 M2 受体的约 200 倍。
  38. GC13618 Tarafenacin Tarafenacin(SVT-40776) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM)，选择性比 M2 受体高约 200 倍。
  39. GC16819 VU0152100 A muscarinic M4 receptor positive allosteric modulator
  40. GC11643 PNU-120596 An α7 neuronal nAChR modulator
  41. GC12717 Ipratropium Bromide A muscarinic receptor antagonist
  42. GC16635 Diphemanil Methylsulfate An anticholinergic agent
  43. GC12994 Rivastigmine Tartrate A cholinesterase inhibitor
  44. GC14113 Oxybutynin An antagonist of muscarinic acetylcholine receptors
  45. GC16526 Atropine A non-selective muscarinic acetylcholine receptor antagonist
  46. GC11786 Acetylcysteine An antioxidant and glutathione precursor
  47. GC10948 Varenicline Tartrate An agonist of α7 and α4β2 nAChRs
  48. GC11210 Vecuronium Bromide A non-depolarizing muscle relaxant
  49. GC14624 Galanthamine HBr An alkaloid with AChE inhibitory and nAChR potentiating activities
  50. GC13449 Rocuronium Bromide A non-depolarizing muscle relaxant
  51. GC12554 Tiotropium Bromide A muscarinic receptor antagonist

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