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Histamine Receptor(组胺受体)

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

  1. Cat.No. 产品名称 Information
  2. GC25785 Promethazine Promethazine is a potent histamine H1 receptor antagonist. Promethazine is a medication used in the management and treatment of allergic conditions, nausea and vomiting, motion sickness, and sedation. Promethazine exhibits antiparasitic properties.
  3. GC25571 Levocetirizine Levocetirizine (LCZ, (R)-Cetirizine), the R-enantiomer of cetirizine, is an antagonist of histamine H(1) receptor.
  4. GC25136 Betazole Dihydrochloride Betazole Dihydrochloride (Ametazole, 2-(3-Pyrazolyl)ethanamine) is a histamine H2 agonist used clinically to test gastric secretory function.
  5. GC25060 Amitriptyline Amitriptyline (MK-230, N-750, Ro41575) is a tricyclic antidepressant (TCA) with analgesic properties, widely used to treat depression and neuropathic pain. Amitriptyline is an inhibitor of both serotonin transporter (SERT) and norepinephrine transporter (NET) with Ki of 3.45 nM and 13.3 nM, respectively. Amitriptyline also inhibits histamine receptor H1, histamine receptor H4, 5-HT2 and sigma 1 receptor with Ki of 0.5 nM, 7.31 nM, 235 nM and 287 nM, respectively. This product is a waxy solid.
  6. GC67995 Ketotifen-d3 fumarate
  7. GC67944 Cetirizine D4
  8. GC66445 Dimethindene maleate
  9. GC65937 INCB38579
  10. GC65296 Pimethixene maleate Pimethixene (Pimetixene) maleate, an antihistamine, anntimigraine agent and antiserotonergic compound, is a highly potent antagonist of a broad range of monoamine receptors, including a variety of serotonin receptors. Pimethixene maleate inhibits 5-HT2A, 5-HT2B, 5-HT2C, 5-HT1A, 5-HT1B, 5-HT6, 5-HT7, Adrenergic α-1A, Dopamine D1 Receptor, Dopamine D2 Receptor, Dopamine D4.4 Receptor, Histamine H1 Receptor, Muscarinic M1 and Muscarinic M2 with pKi of 10.22, 10.44, 8.42, 7.63, < 5, 7.30, 7.28, 7.61, 6.37, 8.19, 7.54, 10.14, 8.61 and 9.38, respectively.
  11. GC64935 Thiethylperazine dimaleate
  12. GC64934 Thiethylperazine
  13. GC64661 H3R antagonist 1 hydrochloride
  14. GC64646 Psoralenoside
  15. GC64577 Cetirizine Impurity C dihydrochloride
  16. GC64545 Tecastemizole
  17. GC64088 Cyclizine A histamine H1 receptor antagonist
  18. GC64084 Samelisant
  19. GC63923 Betahistine-d3 dihydrochloride An internal standard for the quantification of betahistine
  20. GC63666 Chlorcyclizine A histamine H1 antagonist
  21. GC63318 Bilastine-d6
  22. GC63312 Promethazine-d6 hydrochloride
  23. GC62267 Cimetidine sulfoxide
  24. GC61539 Betazole Betazole Dihydrochloride (Ametazole, 2-(3-Pyrazolyl)ethanamine) is a histamine H2 agonist used clinically to test gastric secretory function.
  25. GC61467 Niaprazine
  26. GC61401 Oxatomide
  27. GC48892 NSC 19005 A potential impurity found in commercial preparations of betahistine
  28. GC48855 Mirtazapine (CRM) An Analytical Reference Material
  29. GC48835 Diphenylpyraline A histamine H1 receptor antagonist
  30. GC61256 Rupatadine D4 fumarate
  31. GC60924 Hydroxyzine D8 An internal standard for the quantification of hydroxyzine
  32. GC60791 Doxepin D3 Hydrochloride
  33. GC60709 Cinnarizine D8 An internal standard for the quantification of cinnarizine
  34. GC60691 Cetirizine Impurity C
  35. GC60641 Betahistine mesylate Betahistine mesylate is the mesylate salt form of Betahistine, a histamine analog and H3 receptor agonist that serves as a vasodilator.
  36. GC60563 Acrivastine D7
  37. GC60072 Betahistine A histamine H3 receptor antagonist and histamine H1 receptor agonist
  38. GC39735 Triprolidine hydrochloride monohydrate Triprolidine Hydrochloride is the hydrochloride salt form of Triprolidine, which is the first generation histamine H1 antagonist used in allergic rhinitis.
  39. GC39479 Bepotastine A histamine H1 receptor antagonist
  40. GC39378 Emedastine A histamine H1 receptor antagonist
  41. GC50405 JNJ 39758979 dihydrochloride 高亲和力和选择性组胺H4拮抗剂;口服生物利用度
  42. GC46185 Nimbin A limonoid with diverse biological activities
  43. GC38558 PF-03654746 Tosylate
  44. GC38450 LML134
  45. GC37959 Zaltidine
  46. GC36932 Pitolisant oxalate A histamine H3 receptor antagonist and inverse agonist
  47. GC36931 Pitolisant A histamine H3 receptor antagonist and inverse agonist
  48. GC36878 PF-03654746
  49. GC36875 Perphenazine D8 Dihydrochloride
  50. GC36476 Lodoxamide tromethamine A potent agonist of GPR35 and a mast cell stabilizer
  51. GC36279 Hydroxyzine pamoate Hydroxyzine Pamoate is the pamoate salt form of hydroxyzine, a synthetic piperazine histamine H1-receptor antagonist with anti-allergic, antispasmodic, sedative, anti-emetic and anti-anxiety properties.

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