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Home >> Signaling Pathways >> Neuroscience >> Histamine Receptor

Histamine Receptor(组胺受体)

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

Products for Histamine Receptor

Cat.No. 产品名称 Information
GC31787 Mebhydrolin
美海屈林；美海洛林；甲苄咔啉；
Mebhydrolin是一种特异性组胺H1受体拮抗剂。
GC31767 Peptide 401 Peptide401是一种有效的来源于蜂毒中的肥大细胞脱颗粒肽，抑制血管通透性。
GC31750 Fenspiride Hydrochloride
Decaspiride
Fenspiride盐酸盐是肾上腺素能受体和H1受体拮抗剂。
GC31743 Mequitazine (LM-209)
美喹他嗪; LM-209
Mequitazine (LM-209) is a histamine H1 antagonist which competes with histamine for the normal H1-receptor sites on effector cells of the gastrointestinal tract, blood vessels and respiratory tract.
GC31708 Epinastine (WAL801)
依匹斯汀; WAL801
Epinastine (WAL801) (WAL801) 是一种抗组胺药和肥大细胞稳定剂。
GC31695 Acrivastine (BW825C)
阿伐斯汀; BW825C
A histamine H₁ receptor antagonist
GC31455 Niperotidine
尼匹鲁替定；尼培替丁
Niperotidine是一种组胺H2受体(histamineH2-receptor)拮抗剂。
GC31310 H3 receptor antagonist 1 H3receptorantagonist1是组胺H3(histamineH3)受体拮抗剂，可用于神经疾病的研究。
GC31269 Cipralisant (GT-2331)
GT-2331
Cipralisant (GT-2331) (GT-2331) 是一种具有口服活性、低毒、强效、选择性、高亲和力组胺 H3 受体的体内完全拮抗剂，在体外是一种激动剂，对组胺 H3 受体的 pKi 为 9.9，大鼠组胺 H3 受体的 Ki 为 0.47 nM。
GC31232 H4 Receptor antagonist 1 H4Receptorantagonist1是一种有效的、有选择性的组胺H4受体(H4R)的反向激动剂，其IC50值为19nM。
GC31220 Toreforant (JNJ-38518168)
JNJ-38518168
Toreforant (JNJ-38518168) 是一种有效的选择性组胺 H4 受体 (H4R) 拮抗剂，对人受体的 Ki 值为 8.4 nM。
GC31141 Antihistamine-1 Antihistamine-1是能够渗透血脑屏障的H1-抗组胺药(Ki=6.9nM),它也是CYP2D6和hERG通道的抑制剂，其IC50值分别为5.4和0.8μM。
GC31105 S 38093 S 38093 is a histamine H3 antagonist/inverse agonist with a moderate affinity for rat, mouse and human H3 receptors (Ki = 8.8, 1.44 and 1.2 μM, respectively) and no affinity for other histaminergic receptors.
GC31027 MK-0249 MK-0249是一种有效的histamineH3受体拮抗剂，对人体H3受体的Ki值为1.7nM。
GC31026 (±)-Tazifylline
(±)-他齐茶碱
(±)-Tazifylline是一种有效的，选择性的长效组胺H1受体拮抗剂。
GC30999 Pimethixene (Pimetixene)
匹美噻吨,Pimetixene
Pimethixene (Pimetixene) 是抗组胺药和抗血清素能化合物，用作抗偏头痛剂。
GC30948 Chlorphenoxamine
氯苯沙明；氯苯氧胺
Chlorphenoxamine是一种抗组胺剂和抗胆碱能药,用作抗帕金森氏病。
GC30902 Dimenhydrinate
乘晕宁
Dimenhydrinate is an over-the-counter drug used to prevent nausea, vomiting, and dizziness caused by motion sickness.
GC30821 JNJ-39758979 JNJ-39758979是一个有选择性且具有高亲和性的组胺H4受体拮抗剂,其Ki值为12.5nM。
GC30775 Histamine (Ergamine)
组胺; Ergamine

A biogenic amine
GC30759 H3 receptor-MO-1 H3receptor-MO-1是一种组胺H3受体(histamineH3receptor)调节剂。
GC30496 Doxylamine D5 succinate
琥珀酸多西拉敏 D5
DoxylamineD5琥珀酸盐是Doxylamine氘代化合物标准品。
GC30455 Rocastine (AHR-11325)
罗卡斯汀,AHR-11325
Rocastine (AHR-11325) 是一种选择性、非镇静 H1 拮抗剂，用作抗组胺药。
GC30423 CP-66948 CP-66948是histamineH2受体拮抗剂，能够抑制胃酸分泌，保护粘膜的作用。
GC19441 Levocabastine (hydrochloride)
R 50547 hydrochloride
A histamine H₁ receptor antagonist
GC19178 GSK189254A
GSK189254
A histamine H₃ receptor antagonist
GC18463 N-acetyl Histamine
N-Ω-乙酰基组胺,N-Omega-acetylhistamine
A histamine metabolite
GC18282 Lodoxamide
洛度沙胺,U-42585E free acid
A potent agonist of GPR35 and a mast cell stabilizer
GC18198 Carebastine
卡依巴司丁
An active metabolite of ebastine and a histamine H₁ receptor antagonist
GC12238 Oxomemazine
双氧异丁嗪
Oxomemazine 是一种基于吩噻嗪的组胺 H1 受体阻滞剂，具有明显的抗毒蕈碱特性。
GC17488 Trimipramine (maleate)
三甲丙咪嗪马来酸盐
A tricyclic antidepressant
GC15723 Dimebolin
2,3,4,5-四氢-2,8-二甲基-5-[2-(6-甲基吡啶-3-基)乙基]-1H-吡啶并[4,3-B]吲哚,Dimebon?
A neuroprotective agent
GC12892 Doxepin (hydrochloride)
盐酸多塞平
A tricyclic antidepressant
GC13465 Chlorcyclizine (hydrochloride)
盐酸氯环利嗪；盐酸氯环力嗪
A histamine H₁ antagonist
GC12293 Perphenazine
奋乃静
A typical antipsychotic
GC11695 Cinnarizine
桂利嗪
A calcium channel inhibitor and histamine H₄ receptor antagonist
GC13757 CarbinoxaMine Maleate
马来酸罗托沙敏
A histamine H₁ receptor antagonist
GC10321 Decloxizine
去氯羟嗪; UCB-1402; NSC289116
Decloxizine(UCB-1402; NSC289116) 是一种组胺 1 受体拮抗剂。
GC10814 Promethazine HCl
盐酸异丙嗪
A histamine H₁ receptor antagonist
GC17585 VUF 10460 A histamine H₄ receptor agonist
GC11046 JNJ 5207852 dihydrochloride Selective, non-imidazole histamine H₃R antagonist
GC11330 Tiotidine
硫替丁,ICI 125211
Tiotidine (ICI 125211) 是一种有效的选择性组胺 H2 受体拮抗剂（豚鼠右心房的 pA2=7.3-7.8）。
GC14742 DPPE fumarate
DPPE fumarate
An AEBS ligand
GC11809 (R)-(-)-α-Methylhistamine dihydrobromide
(R)-(-)-α-甲基组胺二氢溴酸盐
(R)-(-)-α-Methylhistamine dihydrobromide 是一种有效的、选择性的、可穿透脑的 H3 组胺受体激动剂，Kd 为 50.3 nM。
GC13537 A 331440 dihydrochloride H3 receptor antagonist,non-imidazole,high affinity
GC12371 JNJ 10181457 dihydrochloride Histamine H3 receptor antagonist
GC11121 A 943931 dihydrochloride Antagonist of histamine H4 receptor,potent and selective
GC17743 A 987306 A 987306 是一种有效的、可口服的组胺 H4 拮抗剂，对大鼠 H4 和人 H4 的 Kis 分别为 3.4 nM 和 5.8 nM。
GC17010 Methimepip dihydrobromide histamine H3 receptor agonist
GC17564 VUF 8430 dihydrobromide A histamine H₄ receptor agonist