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Home >> Signaling Pathways >> Neuroscience >> Histamine Receptor

Histamine Receptor(组胺受体)

Histamine receptor has 4 subtypes (H1,H2,H3 and H4) which mediates various biological fuctions, including allergic reaction, gastric acid secretion and inflammation etc.

Products for  Histamine Receptor

  1. Cat.No. 产品名称 Information
  2. GC31269 Cipralisant (GT-2331) Cipralisant (GT-2331) (GT-2331) 是一种具有口服活性、低毒、强效、选择性、高亲和力组胺 H3 受体的体内完全拮抗剂，在体外是一种激动剂，对组胺 H3 受体的 pKi 为 9.9，大鼠组胺 H3 受体的 Ki 为 0.47 nM。
  3. GC31232 H4 Receptor antagonist 1 H4Receptorantagonist1是一种有效的、有选择性的组胺H4受体(H4R)的反向激动剂，其IC50值为19nM。
  4. GC31220 Toreforant (JNJ-38518168) Toreforant (JNJ-38518168) 是一种有效的选择性组胺 H4 受体 (H4R) 拮抗剂，对人受体的 Ki 值为 8.4 nM。
  5. GC31141 Antihistamine-1 Antihistamine-1是能够渗透血脑屏障的H1-抗组胺药(Ki=6.9nM),它也是CYP2D6和hERG通道的抑制剂，其IC50值分别为5.4和0.8μM。
  6. GC31105 S 38093 S 38093 is a histamine H3 antagonist/inverse agonist with a moderate affinity for rat, mouse and human H3 receptors (Ki = 8.8, 1.44 and 1.2 μM, respectively) and no affinity for other histaminergic receptors.
  7. GC31027 MK-0249 MK-0249是一种有效的histamineH3受体拮抗剂，对人体H3受体的Ki值为1.7nM。
  8. GC31026 (±)-Tazifylline (±)-Tazifylline是一种有效的，选择性的长效组胺H1受体拮抗剂。
  9. GC30999 Pimethixene (Pimetixene) Pimethixene (Pimetixene) 是抗组胺药和抗血清素能化合物，用作抗偏头痛剂。
  10. GC30948 Chlorphenoxamine Chlorphenoxamine是一种抗组胺剂和抗胆碱能药,用作抗帕金森氏病。
  11. GC30902 Dimenhydrinate Dimenhydrinate is an over-the-counter drug used to prevent nausea, vomiting, and dizziness caused by motion sickness.
  12. GC30821 JNJ-39758979 JNJ-39758979是一个有选择性且具有高亲和性的组胺H4受体拮抗剂,其Ki值为12.5nM。
  13. GC30775 Histamine (Ergamine)

    A biogenic amine
  14. GC30759 H3 receptor-MO-1 H3receptor-MO-1是一种组胺H3受体(histamineH3receptor)调节剂。
  15. GC30496 Doxylamine D5 succinate DoxylamineD5琥珀酸盐是Doxylamine氘代化合物标准品。
  16. GC30455 Rocastine (AHR-11325) Rocastine (AHR-11325) 是一种选择性、非镇静 H1 拮抗剂，用作抗组胺药。
  17. GC30423 CP-66948 CP-66948是histamineH2受体拮抗剂，能够抑制胃酸分泌，保护粘膜的作用。
  18. GC19441 Levocabastine (hydrochloride) A histamine H1 receptor antagonist
  19. GC19178 GSK189254A A histamine H3 receptor antagonist
  20. GC18463 N-acetyl Histamine A histamine metabolite
  21. GC18282 Lodoxamide A potent agonist of GPR35 and a mast cell stabilizer
  22. GC18198 Carebastine An active metabolite of ebastine and a histamine H1 receptor antagonist
  23. GC12238 Oxomemazine Oxomemazine 是一种基于吩噻嗪的组胺 H1 受体阻滞剂，具有明显的抗毒蕈碱特性。
  24. GC17488 Trimipramine (maleate) A tricyclic antidepressant
  25. GC15723 Dimebolin A neuroprotective agent
  26. GC12892 Doxepin (hydrochloride) A tricyclic antidepressant
  27. GC13465 Chlorcyclizine (hydrochloride) A histamine H1 antagonist
  28. GC12293 Perphenazine A typical antipsychotic
  29. GC11695 Cinnarizine A calcium channel inhibitor and histamine H4 receptor antagonist
  30. GC13757 CarbinoxaMine Maleate A histamine H1 receptor antagonist
  31. GC10321 Decloxizine Decloxizine(UCB-1402; NSC289116) 是一种组胺 1 受体拮抗剂。
  32. GC10814 Promethazine HCl A histamine H1 receptor antagonist
  33. GC17585 VUF 10460 A histamine H4 receptor agonist
  34. GC11046 JNJ 5207852 dihydrochloride Selective, non-imidazole histamine H3R antagonist
  35. GC11330 Tiotidine Tiotidine (ICI 125211) 是一种有效的选择性组胺 H2 受体拮抗剂（豚鼠右心房的 pA2=7.3-7.8）。
  36. GC14742 DPPE fumarate An AEBS ligand
  37. GC11809 (R)-(-)-α-Methylhistamine dihydrobromide (R)-(-)-α-Methylhistamine dihydrobromide 是一种有效的、选择性的、可穿透脑的 H3 组胺受体激动剂，Kd 为 50.3 nM。
  38. GC13537 A 331440 dihydrochloride H3 receptor antagonist,non-imidazole,high affinity
  39. GC12371 JNJ 10181457 dihydrochloride Histamine H3 receptor antagonist
  40. GC11121 A 943931 dihydrochloride Antagonist of histamine H4 receptor,potent and selective
  41. GC17743 A 987306 A 987306 是一种有效的、可口服的组胺 H4 拮抗剂，对大鼠 H4 和人 H4 的 Kis 分别为 3.4 nM 和 5.8 nM。
  42. GC17010 Methimepip dihydrobromide histamine H3 receptor agonist
  43. GC17564 VUF 8430 dihydrobromide A histamine H4 receptor agonist
  44. GC16018 VUF 5681 dihydrobromide histamine H3 receptor silent antagonist
  45. GC15957 Proxyfan oxalate 组胺H3受体配体
  46. GC14429 JNJ 10191584 maleate histamine H4 receptor silent antagonist
  47. GC16180 GT 2016 A histamine H3 receptor antagonist
  48. GC12737 4-Methylhistamine dihydrochloride A histamine H4 receptor agonist
  49. GC14260 Immethridine dihydrobromide A potent histamine H3 receptor agonist
  50. GC12085 ROS 234 dioxalate ROS 234 dioxalate 是一种有效的 H3 拮抗剂，对豚鼠回肠 H3 受体的 pKB 为 9.46，对大鼠大脑皮层 H3 受体的 pKi 为 8.90，在体外的 ED50 为 19.12 mg/kg (ip)大鼠大脑皮层。
  51. GC10241 Impentamine dihydrobromide histamine H3 receptor antagonist

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