Membrane Transporter/Ion Channel(跨膜转运)
- AMPAR(55)
 - ATPase(78)
 - Calcium Channel(322)
 - Cannabinoid Transporters(6)
 - CFTR(45)
 - Chloride Channels(12)
 - GABA Receptor(220)
 - Glucose Transporters(13)
 - Glutamate (EAAT) Transporters(18)
 - Glycine Receptors(2)
 - GlyT(18)
 - GTPase(28)
 - ICB(1)
 - MCT2(2)
 - Monoamine transporter(15)
 - Monocarboxylate Transporters(12)
 - Multidrug Transporters(4)
 - Na+/Ca2+ Exchanger(15)
 - NKCC(7)
 - NMDA Receptor(76)
 - Nucleoside Transporters(4)
 - Pannexin-1(2)
 - P2X purinergic receptor(65)
 - P-gp(10)
 - Proton Pump(55)
 - Potassium Channel(302)
 - Sodium Channel(204)
 - TRP Channel(162)
 - TRPV1(10)
 - URAT1(12)
 - Other Channel Modulators(10)
 - MCT(3)
 - Kainate Receptors(11)
 - Ionophore(3)
 - sodium-hydrogen exchanger(3)
 - Chloride Channel(27)
 - CRAC Channel(13)
 - EAAT2(5)
 - HCN Channel(6)
 - Na+/HCO3- Cotransporter(1)
 - Na+/K+ ATPase(27)
 - P-glycoprotein(49)
 - iGluR(156)
 - nAChR(100)
 - VDAC(2)
 - Aquaporins(1)
 - Piezo Channels(1)
 - GlyR(1)
 - Ferroportin(1)
 - Urea Transporter(1)
 - Na+/H+ Exchanger (NHE)(1)
 - NTPDase(1)
 - EAAT(1)
 - Piezo Channel(1)
 - ASCT(2)
 
- Cat.No. 产品名称 Information
 - 
                    
                     GC13997 
					
						
							Lomerizine HCl							
                                                           
盐酸洛美利嗪; KB-2796
A voltage-dependent calcium channel blocker
 
				 - 
                    
                     GC15978 
					
						
							Levobupivacaine HCl							
                                                           
盐酸左布比卡因,(S)-(-)-Bupivacaine monohydrochloride
A sodium channel blocker and local anesthetic
 
				 - 
                    
                     GC14764 
					
						
							Lamotrigine							
                                                           
拉莫三嗪; LTG; BW430C
An anticonvulsant
 
				 - 
                    
                     GC15178 
					
						
							Hexamethonium Bromide							
                                                           
六甲溴铵
A nondepolarizing neuromuscular blocking agent
 
				 - 
                    
                     GC16585 
					
						
							Golgicide A							
                                                           
GCA
A reversible inhibitor of GBF1
 
				 - 
                    
                     GC16561 
					
						
							Gliquidone							
                                                           
格列喹酮; AR-DF 26
A second generation sulfonylurea
 
				 - 
                    
                     GC17173 
					
						
							Felodipine							
                                                           
非洛地平
An L-type calcium channel inhibitor
 
				 - 
                    
                     GC10861 
					
						
							Domiphen Bromide							
                                                           
溴化度米芬
A quaternary ammonium compound and cationic surfactant with antimicrobial activity
 
				 - 
                    
                     GC16622 
					
						
							Dexlansoprazole							
                                                           
右旋兰索拉唑; Dexlansoprazole
A proton pump inhibitor
 
				 - 
                    
                     GC16354 
					
						
							Dequalinium Chloride							
                                                           
地喹氯铵
An ammonium cation with diverse biological activities
 
				 - 
                    
                     GC16255 
					
						
							Decamethonium Bromide							
                                                           
十烃溴铵
A depolarizing neuromuscular blocking agent
 
				 - 
                    
                     GC11120 
					
						
							Ciclopirox ethanolamine							
                                                           
环吡酮乙醇胺盐; Ciclopirox ethanolamine; HOE 296
An iron chelator, antifungal, and anticancer agent
 
				 - 
                    
                     GC17086 
					
						
							Chlorpropamide							
                                                           
氯磺丙脲
A first generation sulfonylurea
 
				 - 
                    
                     GC14421 
					
						
							CFTRinh-172							
                                                           
CFTR(inh)172, Cystic Fibrosis Transmembrane Conductance Regulator Inhibitor 172
CFTRinh-172被鉴定为囊性纤维化跨膜传导调节因子(CFTR)Cl-通道强效的选择性阻断剂。CFTRinh-172对野生型、G551D和G1349D CFTR的Cl-电流具有抑制作用,Ki值为0.5μM。
 
				 - 
                    
                     GC17683 
					
						
							Brefeldin A							
                                                           
布雷非德菌素 A; BFA; Cyanein; Decumbin
Brefeldin A(BFA)是一种真菌大环内酯,能够有效、可逆地抑制内质网和高尔基体之间的蛋白质运输和囊泡形成。
 
				 - 
                    
                     GC13125 
					
						
							Benzocaine							
                                                           
苯佐卡因
An Analytical Reference Standard
 
				 - 
                    
                     GC14339 
					
						
							Benzethonium Chloride							
                                                           
苄索氯铵
Benzethonium chloride 抑制非洲爪蟾卵母细胞中的人重组 α7 和 α4β2 神经元烟碱乙酰胆碱受体。
 
				 - 
                    
                     GC12414 
					
						
							Bemegride							
                                                           
贝美格; 3-Ethyl-3-methylglutarimide; Bemegrid
Bemegride (3-Ethyl-3-methylglutarimide) 是一种中枢神经系统兴奋剂和巴比妥类中毒的解毒剂。
 
				 - 
                    
                     GC13723 
					
						
							Amitriptyline HCl							
                                                           
盐酸阿米替林
A tricyclic antidepressant
 
				 - 
                    
                     GC15458 
					
						
							Ambroxol HCl							
                                                           
盐酸氨溴索,NA-872 hydrochloride
An expectorant
 
				 - 
                    
                     GC13430 
					
						
							(-)-Blebbistatin							
                                                           
(S)-(-)-Blebbistatin
(-)-Blebbistatin是外消旋体混合物(±)-Blebbistatin(货号:GC12341)的一种其中一个构型,是活性形式。(-)-Blebbistatin是一种非肌肉肌球蛋白II ATP酶的细胞渗透性抑制剂,有效抑制多种横纹肌肌球蛋白以及脊椎动物非肌肉肌球蛋白,IC50值范围为0.5-5μM,平滑肌肌球蛋白仅受到微弱抑制(IC50=80μM)。
 
				 - 
                    
                     GC14792 
					
						
							Reserpine hydrochloride							
                                                           
利血平盐酸盐
Irreversible inhibitor of VMAT1 and VMAT2
 
				 - 
                    
                     GC14703 
					
						
							Oxybutynin chloride							
                                                           
盐酸奥昔布宁
An antagonist of muscarinic acetylcholine receptors
 
				 - 
                    
                     GC13824 
					
						
							Indapamide							
                                                           
吲达帕胺
An Analytical Reference Standard
 
				 - 
                    
                     GC17340 
					
						
							Carbamazepine							
                                                           
卡马西平; CBZ; NSC 169864
卡马西平是一种钠通道阻滞剂,是一种抗惊厥药。
 
				 - 
                    
                     GC11213 
					
						
							Trichlormethiazide							
                                                           
三氯噻嗪
A thiazide diuretic
 
				 - 
                    
                     GC15363 
					
						
							Felbamate hydrate							
                                                           
W-554 hydrate; ADD-03055 hydrate
An inhibitor of NMDA receptors and a modulator of GABAA receptors
 
				 - 
                    
                     GC10522 
					
						
							Felbamate							
                                                           
非尔氨酯; W-554; ADD-03055
An inhibitor of NMDA receptors and a modulator of GABAA receptors
 
				 - 
                    
                     GC13162 
					
						
							Prilocaine hydrochloride							
                                                           
盐酸丙胺卡因
An Analytical Reference Standard
 
				 - 
                    
                     GC15071 
					
						
							Prilocaine							
                                                           
丙胺卡因
An Analytical Reference Standard
 
				 - 
                    
                     GC17952 
					
						
							Zonisamide sodium							
                                                           
唑尼沙胺钠; AD 810 sodium; CI 912 sodium
A broad-spectrum sulfonamide antiepileptic agent
 
				 - 
                    
                     GC10500 
					
						
							Oxcarbazepine							
                                                           
奥卡西平; GP 47680
A prodrug form of 10,11-dihydro-10-hydroxy carbamazepine
 
				 - 
                    
                     GC14977 
					
						
							Minoxidil							
                                                           
米诺地尔; U10858
An anti-hypertensive vasodilator
 
				 - 
                    
                     GC15101 
					
						
							Azelnidipine							
                                                           
阿折地平; CS 905
A calcium channel blocker
 
				 - 
                    
                     GC17106 
					
						
							Verapamil HCl							
                                                           
盐酸维拉帕米; (±)-Verapamil hydrochloride; CP-16533-1 hydrochloride
Verapamil HCl是 L 型钙通道阻滞剂和肾上腺素能受体拮抗剂,常用于高血压、心律失常和心绞痛的研究。
 
				 - 
                    
                     GC17316 
					
						
							Gabapentin HCl							
                                                           
加巴喷丁盐酸盐
An approved antiepileptic drug
 
				 - 
                    
                     GC13792 
					
						
							Rufinamide							
                                                           
卢非酰胺; CGP 33101; E 2080; RUF 331
An anticonvulsant
 
				 - 
                    
                     GC12234 
					
						
							Dronedarone HCl							
                                                           
盐酸决奈达隆
An antiarrhythmic agent
 
				 - 
                    
                     GC17804 
					
						
							GlyH-101							
                                                           
GlyH101, Cystic Fibrosis Transmembrane Conductance Regulator Inhibitor II
A reversible CFTR channel blocker
 
				 - 
                    
                     GC10443 
					
						
							Meclofenoxate hydrochloride							
                                                           
盐酸甲氯酚酯
A nootropic agent
 
				 - 
                    
                     GC16899 
					
						
							Coluracetam							
                                                           
考拉西坦; MKC-231
An Analytical Reference Standard
 
				 - 
                    
                     GC16359 
					
						
							Rosuvastatin							
                                                           
瑞舒伐他汀; ZD 4522
Rosuvastatin是一种竞争性HMG-CoA还原酶抑制剂,IC50值为11nM。
 
				 - 
                    
                     GC16128 
					
						
							Clevidipine Butyrate							
                                                           
氯维地平
An inhibitor of L-type calcium channels
 
				 - 
                    
                     GC15293 
					
						
							Manidipine 2HCl							
                                                           
盐酸马尼地平,CV-4093
An L- and T-type calcium channel blocker
 
				 - 
                    
                     GC16889 
					
						
							Nisoldipine							
                                                           
尼索地平; BAY-k 5552
A calcium channel inhibitor
 
				 - 
                    
                     GC11299 
					
						
							Mitiglinide Calcium							
                                                           
米格列奈钙; KAD-1229 anhydrous; S21403 anhydrous
A SUR1/Kir6.2 inhibitor
 
				 - 
                    
                     GC14111 
					
						
							(R)-baclofen							
                                                           
(R)-巴氯芬; Arbaclofen; STX209
(R)-巴氯芬 (Arbaclofen) 是一种选择性 GABAB 受体激动剂。
 
				 - 
                    
                     GC10599 
					
						
							Esomeprazole Sodium							
                                                           
埃索美拉唑钠,(S)-Omeprazole sodium; (-)-Omeprazole sodium
Esomeprazole Sodium是一种强效、具有口服活性的质子泵抑制剂。
 
				 - 
                    
                     GC13375 
					
						
							Dofequidar fumarate							
                                                           
MS-209
A quinoline derivative and inhibitor of multidrug resistance
 
				 - 
                    
                     GC11470 
					
						
							Flupirtine maleate							
                                                           
氟吡啶马来酸
An activator of Kv7 channels