Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

qq在线咨询
Home >> Signaling Pathways >> Endocrinology and Hormones

Endocrinology and Hormones(内分泌和激素)

Endocrinology and Hormones

The endocrine system is an information signaling system that coordinates most bodily functions. It senses environmental changes and secretes corresponding hormones to coordinate metabolism, maintain homeostasis, and regulate growth and development.read more

Products for  Endocrinology and Hormones

  1. Cat.No. 产品名称 Information
  2. GC63431 DPDPE TFA DPDPE TFA 是一种阿片肽，是一种具有抗惊厥作用的选择性阿片受体 (DOR) 激动剂。
  3. GC63402 Rezvilutamide Rezvilutamide (SHR3680) 雄激素受体 (androgen receptor) 的拮抗剂。Rezvilutamide (SHR3680) 可用于前列腺癌的研究。
  4. GC63292 (rac)-PF-998425 (rac)-PF-998425 是一种有效、选择性的非甾体雄激素受体 (AR) 拮抗剂。(rac)-PF-998425 在 AR 结合和细胞分析中的 IC50 值分别为 26 和 90 nM。(rac)-PF-998425 具有用于研究雄激素性脱发的潜力。
  5. GC63217 Testosterone undecanoate Testosterone undecanoate是睾酮酯，用做男性节育。
  6. GC63200 Spiradoline Spiradoline (U-62066) 是一种芳基乙酰胺，是一种选择性 kappa 阿片受体 (κ-opioid receptor, KOR) 激动剂，在豚鼠中的 Ki 为 8.6 nM。Spiradoline 对 μ 和 δ 受体的 Ki 值分别为 252 nM 和 9400 nM。Spiradoline 具有强效的利尿，止痛，抗心律失常，镇咳，神经保护作用，并易于穿过血脑屏障。
  7. GC63115 Nociceptin (1-13), amide TFA Nociceptin (1-13), amide TFA 是一种有效的阿片受体 ORL1 (OP4) 受体激动剂，对小鼠输精管 pEC50 值为 7.9，与大鼠前脑膜结合的 Ki 值为 0.75 nM。
  8. GC63096 Nandrolone phenylpropionate Nandrolone phenylpropionate，19-nortestosterone 的衍生物，是一种合成代谢类固醇，可促进蛋白质合成。Nandrolone phenylpropionate 用于缓解组织分解代谢，可以用于骨质疏松症和特纳综合征的研究。
  9. GC63072 Methyl-6-alpha-Naltrexol Methyl-6-alpha-Naltrexol 是甲基纳曲酮 (MNTX) 的代谢物 (metabolite)。Methyl-6-alpha-Naltrexol 是一种选择性的 mu-阿片受体 (mu-opioid receptor) 拮抗剂，在胃肠道组织中起外周作用的受体拮抗剂作用。
  10. GC63066 Methenolone acetate

    Metenolone醋酸盐是一种长效的蛋白同化激素，具有较低的雄激素特性。IC50 value:Target:Metenolone醋酸盐是一种天然存在的化合物，在驯养的怀孕猫科肾上腺腺体内发现。Metenolone醋酸盐用于口服给药。Methenolone醋酸盐可抑制下丘脑 - 垂体 - 性腺通路。[1] Methenolone醋酸盐作为口服制剂时，Methenolone不是17-α-烷基化，而是1-甲基化，便于提高口服生物利用度，且降低肝脏应力。[2]
  11. GC62992 Glutaurine A dipeptide
  12. GC62761 1α-Hydroxy-3-epi-vitamin D3 1α-Hydroxy-3-epi-vitamin D3 是 1alpha,25-dihydroxyvitamin D3 的天然代谢物，是甲状旁腺激素 (?PTH?) 分泌的有效抑制剂
  13. GC49427 3,5-Diiodo-L-thyronine A thyroid hormone metabolite
  14. GC49423 Metanephrine-d3 (hydrochloride) An internal standard for the quantification of metanephrine
  15. GC49408 Ramipril Diketopiperazine Acid A potential impurity found in commercial preparations of ramipril
  16. GC49399 N-Desbutyl Dronedarone (hydrochloride) An active metabolite of dronedarone
  17. GC49393 all-trans-13,14-Dihydroretinol A metabolite of all-trans retinoic acid
  18. GC49391 7α-Thiospironolactone An active metabolite of spironolactone
  19. GC49389 Tritylolmesartan Medoxomil An intermediate in the synthesis of olmesartan medoxomil
  20. GC49385 Halometasone A synthetic corticosteroid
  21. GC49342 Glucagon-d9 (trifluoroacetate salt) An internal standard for the quantification of glucagon
  22. GC49329 Turkesterone (hydrate) A phytoecdysteroid with diverse biological activities
  23. GC49326 5β-Dihydroprogesterone A progesterone receptor agonist and metabolite of progesterone
  24. GC49321 AZ-GHS-22 An inverse agonist of GHS-R1a
  25. GC49306 Isopimaric Acid A diterpenoid resin acid
  26. GC49303 Ganoderic Acid DM A triterpenoid with diverse biological activities
  27. GC49254 Estrone-3-Glucuronide (sodium salt hydrate) A metabolite of 17β-estradiol
  28. GC49207 Lumisterol 3 A photoisomer of previtamin D3
  29. GC49206 7α-hydroxy Dehydroepiandrosterone An active metabolite of dehydroepiandrosterone
  30. GC49189 (E/Z)-4-hydroxy Tamoxifen-d5 An internal standard for the quantification of (E/Z)-4-hydroxy tamoxifen
  31. GC49180 3-epi-25-hydroxy Vitamin D3 The C-3 epimer of 25-hydroxy vitamin D3
  32. GC49176 5β-Tetrahydrocortisol An endogenous metabolite of cortisol
  33. GC49172 2-hydroxy Estrone An active metabolite of estrone
  34. GC49161 16α-hydroxy Dehydroepiandrosterone A metabolite of dehydroepiandrosterone
  35. GC49143 Deslorelin (acetate) A peptide agonist of GnRH
  36. GC49123 Somatorelin (1-44) amide (human) (trifluoroacetate salt) A synthetic GHRH peptide
  37. GC49108 Racecadotril-d5 An internal standard for the quantification of racecadotril
  38. GC49068 16-Epiestriol A metabolite of estrone
  39. GC49055 Tebuconazole-d9 An internal standard for the quantification of tebuconazole
  40. GC49048 Guanylin (human) (trifluoroacetate salt) A peptide hormone activator of GC-C
  41. GC49025 Desogestrel-13C2-d2 An internal standard for the quantification of desogestrel
  42. GC49012 Tauro-β-muricholic Acid-d4 (sodium salt) tauro-β-muricholic acid 定量的内标
  43. GC49011 Tauro-α-muricholic Acid-d4 (sodium salt) An internal standard for the quantification of tauro-α-muricholic acid
  44. GC48981 Senktide (trifluoroacetate salt) A potent NK3 receptor agonist
  45. GC48979 Estradiol 17-(β-D-Glucuronide) (sodium salt hydrate) A substrate of multidrug resistance protein 2
  46. GC62683 Ralaniten Ralaniten (EPI-002) 是一种有效和具有口服活性的雄激素受体 N 端结构域 (AR-NTD) 拮抗剂。Ralaniten 抑制 AR 转录活性，IC50 值为 7.4 μM。Ralanites 可用于去势抵抗性前列腺癌 (CRPC) 的研究。
  47. GC62644 GnRH antagonist 2 GnRH antagonist 2 (formula I) 是一种 GnRH 受体拮抗剂，可用于子宫内膜异位的研究。
  48. GC62603 Ralaniten triacetate Ralaniten triacetate (EPI-506) 是 Ralaniten 的前药，是一种首创的，具有口服活性的雄激素受体 (AR) N 端结构域 (NTD) 抑制剂。Ralaniten triacetate 对全长和与抗性相关的 AR 物种，包括 AR-v7 都有活性。
  49. GC62329 VPC-14449 VPC-14449 是一种有效和选择性的雄激素受体 DNA 结合结构域 (AR-DBD) 抑制剂，对全长人 AR 的 IC50 值为 0.34 μM。VPC-14449 可降低全长 AR 以及 AR 变体与染色质相互作用的能力。VPC-14449 可用于前列腺癌的研究。
  50. GC62249 Honokiol DCA Honokiol DCA (Honokiol dichloroacetate) 是 Honokiol 的二氯乙酸酯类似物。Honokiol DCA 在体外可以抑制人前列腺癌细胞的生长并抑制雄激素受体 (AR) 蛋白水平。
  51. GC62209 CLP-3094 CLP-3094, a potent inhibitor targeting the binding function 3 (BF3) site of androgen receptor (AR), inhibits AR transcriptional activity with IC50 of 4 μM, also is a selective, potent GPR142 antagonist.

Items 101 to 150 of 818 total

per page
  2. 1
  3. 2
  4. 3
  5. 4
  6. 5

Set Descending Direction