ROR/RAR/RXR
RAR/RXR is a heterodimer of RAR (retinoic acid receptor) and RXR (retinoid X receptor) that cause dissociation of corepressor and recruitment of coactivator protein that, in turn, promotes transcription of the downstream target gene into mRNA and eventually protein.
- Cat.No. 产品名称 Information
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GC50708
(±)-ML 209
An RORγt antagonist
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GC34960
(+)-Talarozole
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GC18632
6-hydroxy Bexarotene
An oxidative metabolite of bexarotene
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GC46740
7β,27-dihydroxy Cholesterol
An oxysterol and agonist of RORγ and RORγt
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GC40464
9(R)-HETE
Enantiomer of (±)9-HETE; RXRγ activator
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GC40465
9(S)-HETE
A monohydroxy fatty acid and RXRγ agonist
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GC14596
9-cis-Retinoic Acid
An agonist of RAR and RXR isoforms
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GC11852
AC 261066
AC 261066 是一种有效的、可口服的、异构体选择性视黄酸β2 (RARbeta2) 受体激动剂,pEC50 为 8.0。
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GC10871
AC 55649
AC 55649 是一种有效的、高度异构体选择性的人 RARβ2 受体激动剂,pEC50 为 6.9。
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GC17094
Acitretin
A retinoid
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GC17113
Acitretin sodium
A retinoid
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GC10610
Adapalene
An RARβ and RARγ agonist
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GC14379
Adapalene sodium salt
An RARβ and RARγ agonist
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GC46798
Adapalene-d3
An internal standard for the quantification of adapalene
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GC13959
Adarotene
An atypical retinoid
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GC32817
AGN 193109
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GC33315
AGN 194078
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GC12598
AGN 194310
AGN 194310 (VTP-194310) 是一种高亲和力、有效和选择性的视黄酸受体 (RARs) 泛拮抗剂,对 RARα、RARβ、RARγ 的 Kd 值分别为 3 nM、2 nM、5 nM。
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GC35265
AGN 195183
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GC35266
AGN 196996
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GC35267
AGN 205327
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GC35268
AGN 205728
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GC39584
AGN194204
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GC14511
all-trans Retinal
A natural retinoid
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GC42769
all-trans Retinoyl β-D-Glucuronide
A metabolite of all-trans retinoic acid
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GC49393
all-trans-13,14-Dihydroretinol
A metabolite of all-trans retinoic acid
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GC18482
all-trans-5,6-epoxy Retinoic Acid
An agonist of RAR isoforms
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GC13664
AM580
A selective RARα agonist
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GC63932
Amsilarotene
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GC19035
AR7
A RARα antagonist
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GC46892
ATRA-BA Hybrid
A prodrug form of all-trans retinoic acid and butyric acid
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GC10037
Bexarotene
An RXR agonist
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GC46923
Bexarotene-d4
A neuropeptide with diverse biological activities
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GC60076
Bigelovin
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GC11504
BMS 195614
A neutral RARα-selective antagonist
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GC49654
BMS 270394
A RARγ agonist
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GC10656
BMS 453
An RARβ agonist, RARα/γ antagonist
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GC15648
BMS 493
A pan-RAR inverse agonist
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GC14185
BMS 753
A synthetic retinoid and RARα agonist
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GC17382
BMS 961
A RAR? agonist
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GC46104
Butyric Acid-d7
An internal standard for the quantification of sodium butyrate
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GC11794
CD 1530
A selective RARγ agonist
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GC10080
CD 2314
CD 2314 是一种有效的选择性 RARβ 受体激动剂,在 S91 黑色素瘤细胞中的 Kd 为 195 nM。
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GC12072
CD 2665
A selective RARβ and RARγ antagonist
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GC17730
CD 3254
A selective RXR agonist
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GC11464
CD 437
A selective RARγ agonist
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GC11053
Ch 55
An RAR agonist
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GC11676
EC 23
A synthetic retinoid
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GC12577
ER 50891
ER-50891 是一种有效的视黄酸受体 α(RARα) 拮抗剂。 ER-50891 显着减弱 ATRA 对 BMP 2 诱导的成骨细胞生成的抑制作用。
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GC17143
Fenretinide
A synthetic retinoic acid derivative