Endocrinology and Hormones(内分泌和激素)

Endocrinology and Hormones

The endocrine system is an information signaling system that coordinates most bodily functions. It senses environmental changes and secretes corresponding hormones to coordinate metabolism, maintain homeostasis, and regulate growth and development.read more

Products for Endocrinology and Hormones

Cat.No. 产品名称 Information
GC17856 RU 58668 Pure antiestrogen that downregulates estrogen receptor expression
GC13546 Dynorphin A
强啡肽A
An endogenous opioid receptor agonist
GC15975 α-Estradiol
α-雌二醇; Alfatradiol; Epiestradiol; Epiestrol
A weak estrogen with neuroprotective effects
GC13189 Cyprodime hydrochloride
μ-opioid receptor antagonist
GC18003 (R,R)-THC (R,R)-THC 是 ERα 激动剂和 ERβ 拮抗剂，对 ERα 和 ERβ 的 Kis 分别为 9.0 nM 和 3.6 nM。
GC10803 DAMGO
L-酪氨酰-D-丙氨酰甘氨酰-N-(2-羟基乙基)-NALPHA-甲基-L-苯丙氨酰胺

A μ-opioid receptor agonist
GC15885 (±)-U-50488 hydrochloride
(±)-Trans-(1R,2R)-U-50488 hydrochloride
An Analytical Reference Material
GC12598 AGN 194310
VTP-194310
AGN 194310 (VTP-194310) 是一种高亲和力、有效和选择性的视黄酸受体 (RARs) 泛拮抗剂，对 RARα、RARβ、RARγ 的 Kd 值分别为 3 nM、2 nM、5 nM。
GC13664 AM580
4-[(5,6,7,8-四氢-5,5,8,8-四甲基-2-萘基)甲酰氨基]苯甲酸,CD336; NSC608001; Ro 40-6055
A selective RARα agonist
GC17983 Taltirelin
他替瑞林; TA-0910
Taltirelin (TA0910) 是促甲状腺素释放激素受体 (TRH-R) 的超级激动剂，IC50 为 910 nM，EC50 为 36 nM，可刺激细胞溶质 Ca2+ 浓度（Ca2+ 释放）的增加。
GC11781 Medroxyprogesterone
甲羟孕酮; 17α-Hydroxy-6α-methylprogesterone; U8840
A progesterone receptor agonist
GC13303 Etonogestrel
依托孕烯,3-Oxodesogestrel; 3-keto-Desogestrel
A steroidal progestin
GC15366 Clomiphene citrate
枸橼酸氯米芬; Clomifene citrate
A selective estrogen receptor modulator
GC12974 Medroxyprogesterone acetate
醋酸甲羟孕酮; Medroxyprogesterone 17-acetate; Farlutin
Medroxyprogesterone acetate（MPA）是一种人工合成的孕激素。
GC10702 Trimebutine
曲美布汀
An opioid receptor agonist
GC11436 Ethisterone
炔孕酮,Pregneninolone; 17α-Ethynyltestosterone
A synthetic progestin
GC12815 Formestane
福美司坦
An Analytical Reference Standard
GC11885 Sevelamer HCl
盐酸司维拉姆
Sevelamer HCl 是一种磷酸盐结合药物，用于治疗慢性肾病患者的高磷血症；由与环氧氯丙烷交联的聚烯丙胺组成。
GC14273 TTNPB (Arotinoid Acid)
Ro 13-7410; Arotinoid acid; AGN191183
A potent, selective RAR agonist
GC15001 Tiratricol
替拉曲可,3,3',5-Triiodothyroacetic acid
A thyroid hormone receptor agonist
GC12516 Spironolactone
螺内酯; SC9420
An Analytical Reference Standard
GC11822 Erteberel (LY500307)
芬克罗酮,LY500307
A potent and selective agonist of ERβ
GC12409 Liothyronine Sodium
三碘代甲状腺素钠盐
Liothyronine sodium 是一种强效的甲状腺激素受体TRα和TRβ激动剂，其 Ki 值为 2.33nM。
GC15324 Hexestrol
4,4'-(1,2-二乙基亚乙基)二苯酚
A synthetic non-steroidal estrogen receptor ligand
GC12126 Flutamide
氟他胺; SCH 13521
An androgen receptor antagonist and a prodrug form of 2-hydroxy flutamide
GC12000 Ethynodiol diacetate
双醋炔诺醇,Ethynodiol acetate
A synthetic progestogen
GC12182 Estriol
雌三醇; Oestriol
An estradiol metabolite produced during pregnancy
GC11796 Estradiol valerate
戊酸雌二醇,β-Estradiol 17-valerate
A synthetic estrogen
GC10139 Estradiol Cypionate
环戊丙酸雌二醇
A synthetic estrogen
GC16292 Equol
(±)-雌马酚
An estrogen receptor agonist
GC13072 Epiandrosterone
表雄酮; 3β-Androsterone; trans-Androsterone; iso-Androsterone
An Analytical Reference Standard
GC10245 Bazedoxifene HCl
盐酸巴多昔芬,TSE-424 hydrochloride
Bazedoxifene HCl (TSE-424 hydrochloride) 是一种具有口服活性、可渗透 BBB 的非甾体选择性雌激素受体调节剂 (SERM)，对 ERα 的 IC50 分别为 23 nM 和 99 nM；和ERβ，分别。盐酸巴多昔芬可用于骨质疏松症的研究。 Bazedoxifene HCl 作为 IL-6/GP130 蛋白质-蛋白质相互作用的抑制剂。 Bazedoxifene HCl 可用于胰腺癌的研究。
GC12434 AZD1981 A DP₂/CRTH₂ receptor antagonist
GC13297 Altrenogest
四烯雌酮,Allyltrenbolone; RU2267
A synthetic progestin
GC14704 Levonorgestrel
左炔诺孕酮; D-Norgestrel
A synthetic progestin
GC16433 Aminoglutethimide
氨鲁米特,DL-Aminoglutethimide
An aromatase inhibitor
GC12379 Drospirenone
屈螺酮,Dihydrospirorenone
A synthetic progestogen
GC10017 Gestodene
孕二烯酮; SHB 331; WL 70
A progestin
GC17113 Acitretin sodium
阿维A钠; Ro 10-1670 sodium
A retinoid
GC14379 Adapalene sodium salt
阿达帕林钠; CD 271 sodium salt
An RARβ and RARγ agonist
GC15578 Dienogest
地诺孕素; STS 557
A synthetic progestin and PR agonist
GC13835 Toremifene Citrate
枸橼酸托瑞米芬; Z-Toremifene citrate; NK 622; FC-1157a
A selective estrogen receptor modulator
GC17985 Chenodeoxycholic Acid
鹅去氧胆酸
A primary bile acid
GC10760 XL335
3-(3,4-二氟苯甲酰基)-1,2,3,6-四氢-1,1-二甲基氮杂卓[4,5-B]吲哚-5-甲酸1-甲基乙基酯,FXR-450; XL335; WAY-362450
A potent and selective FXR agonist
GC10975 GW4064
3-(2,6-二氯苯基)-4-(3'-羧基-2-氯二苯乙烯-4-基)氧甲基-5-异丙基异恶唑
GW4064作为合成的FXR激动剂，用于治疗胆汁淤积性肝病、代谢综合征和酒精性肝病。
GC11268 L-Thyroxine
L-甲状腺素,Levothyroxine; T4
A synthetic form of thyroxine
GC11016 Meptazinol HCl
盐酸美普他酚
μ1 阿片受体的部分激动剂
GC11677 Ulipristal acetate
醋酸乌利司他; CDB-2914
A selective progesterone receptor modulator
GC14304 Palovarotene
4-[(1E)-2-[5,6,7,8-四氢-5,5,8,8-四甲基-3-(1H-吡唑-1-基甲基)-2-萘基]乙烯基]苯甲酸,R 667; Ro 3300074
A RARγ agonist
GC11070 Dehydroepiandrosterone (DHEA)
脱氢表雄酮; Prasterone; Dehydroisoandrosterone; Dehydroepiandrosterone
脱氢表雄酮 (DHEA) 及其硫酸酯 DHEAS 共同代表了人体内最丰富的类固醇激素。