- Cat.No. 产品名称 Information
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GC13345
NXY-059
4-[[(1,1-二甲基乙基)氧化亚氨基]甲基]-1,3-苯二磺酸二钠,NXY-059
Free radical trapping agent
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GC11594
RG7388
RG 7388; RG-7388; ldasanutlin; Ro 5503781
MDM2 antagonist, oral, selective
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GC15359
SL-327
Selective MEK1/2 inhibitor
-
GC37722
TAK-448 acetate
MVT-602 acetate
TAK-448 acetate (MVT-602 acetate) 是一种有效的 KISS1R 激动剂,IC50 值为 460 pM,EC50 值为 632 pM。
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GC19156
TAS-120
TAS-120
A novel, potent and highly selective FGFR inhibitor
-
GC10108
WAY-100635
WAY 100635; WAY100635
5-HT1A receptor antagonist,potent and selective
-
GC13922
ZK 93423 hydrochloride
GABAA receptor agonist
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GC90155
1-Palmitoyl-2-Oleoyl-sn-glycero-3-PE
1-Palmitoyl-2-Oleoyl-sn-glycero-3-Phosphatidylethanolamine, 1-Palmitoyl-2-Oleoyl-sn-glycero-3-Phosphoethanolamine, 16:0-18:1 PE, PE(16:0/18:1), 1,2-POPE
一种磷脂
-
GN10231
Fraxin
秦皮甙,Fraxetol 8-glucoside; Fraxoside
A coumarin glycoside
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GC31648
4-Octyl Itaconate
4-辛基衣康酸
4-Octyl Itaconate (4-OI) is a cell-permeable itaconate derivative. Itaconate and 4-Octyl Itaconate had similar thiol reactivity, making 4-Octyl Itaconate a suitable itaconate surrogate to study its biological function.
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GK10002
SYBR Green qPCR Master Mix
The Super Hot-Start SYBR Green qPCR Master Mix is a ready-to-use qPCR cocktail.
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GC20228
α-Amyrin
α-香树脂醇
α-香树脂醇是一种五环三萜类化合物。
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GC27475
3-Methoxy-2-methylbenzoic acid
3-甲氧基邻甲基苯甲酸; 2-甲基间茴香酸; AKOS005259940; BCP19993; SCHEMBL311839; AM84144; SY020989; DTXSID00427374; EN300-299886;,3-methoxy-2-methylbenzoic acid; 3-methoxy-2-methyl-benzoic Acid; 2-methyl-3-methoxyl-benzoic acid; A8005; AC-3996; FT-0615969
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GA23423
Pyr-Arg-Thr-Lys-Arg-AMC
Pyr-Arg-Thr-Lys-Arg-AMC也称为pERTKR-AMC,是一种含有AMC(7-氨基-4-甲基香豆素)的五肽荧光底物。
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GC64436
PROTAC BRD4 Degrader-9
PROTAC BRD4 Degrader-9 (compound 8a) 是一种有效的由von Hippel-Lindau配体和BRD4配体相连的PROTAC。PROTAC BRD4 Degrader-9 可与 STEAP1 和 CLL1 抗体偶联从而降解 PC3 前列腺癌细胞中的 BRD4 蛋白,DC50 值分别为 0.86 nM 和 7.6 nM。
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GC68230
MitoSOX Red
MitoSOX Red是一种靶向线粒体的活细胞荧光探针,最大激发光/发射光为510/580 nm。
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GC19445
Azoxymethane
偶氮甲烷; AOM
偶氮甲烷作为一种结肠致癌物,可导致DNA加合物的形成。偶氮甲烷(AOM)导致O(6)-甲基鸟嘌呤加合物的形成,从而导致G->A跃迁。.
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GC27474
Isophoronediamine (cis- and trans- mixture)(IPDA)
异佛尔酮双胺; 1-氨基-3-氨基甲基-3,3,5-三甲基环己烷 (顺反混合物); 5-氨基-1,3,3-三甲基环己甲胺,顺式和反式的混合物; 1-amino-3,3,5-trimethyl-5-aminomethyl cyclohexane; IPDA
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GC37754
Teglicar
替格列卡
Teglicar 是选择性和可逆性的肉毒碱棕榈酰转移酶 1 (L-CPT1) 肝异构体抑制剂,可减少酮生成和葡萄糖生成,降低糖异生,改善葡萄糖稳态。Teglicar 具有潜在的抗高血糖特性。
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GD20454
Propionic Acid-d5
丙酸-d5
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GC71808
CMP-sialic acid synthetase (NmCSS)
CMP-sialic acid synthetase (NmCSS)是一种参与碳水化合物和含唾液酸的糖复合物生物合成的必需酶。
-
GC31535
3-Methyl-L-histidine
3-甲基-L-组氨酸
An amino acid
-
GC26573
ZINC00640089
ZINC00640089 是一种特异性的脂质运载蛋白-2 (LCN2) 抑制剂。
-
GC17242
(-)-epigallocatechin
(-)-表没食子儿茶素; Epigallocatechin; L-Epigallocatechin
green tea epicatechin
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GC32791
BETd-260 (ZBC 260)
ZBC 260
BETd-260是基于PROTAC技术的一种有效的BET降解剂,在白血病细胞RS4;11中,降低BRD4蛋白活性,IC50值为30pM。
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GC74063
BNN6
BNN6是一种热响应型一氧化氮供体,可有效地与光热疗法(PTT)相结合。
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GC62921
D-Allose
D-阿洛糖
D-Allose是一种超低热量的醛己糖,在冷冻过程中对细胞存活具有冷冻保护功能。
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GC35980
Emricasan
恩利卡生; PF 03491390; IDN-6556
A pan-caspase inhibitor
-
GC26684
Gadoterate meglumine
多它灵
Gadoterate meglumine是一种非特异性的顺磁性钆复合物,用作磁共振成像(MRI)的造影增强剂。
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GA10633
HOBt (anhydrous)
1-羟基苯并三唑(HOBT)
Racemization inhibitor
-
GC12581
K145
SphK2 inhibitor
-
GC36372
K145 hydrochloride
3-(2-氨基乙基)-5-[3-(4-丁氧基苯基)亚丙基]-2,4-噻唑烷二酮盐酸盐
A selective SPHK2 inhibitor
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GC19794
Phosphatidylserine
丝氨酸磷脂;二酰甘油酰磷酸丝氨酸;PS
磷脂酰丝氨酸
-
GC40998
Pinostrobin
球松素
A flavonoid with diverse biological activities
-
GC62724
R243
R243是一种CCR8受体抑制剂,R243可抑制由CCL1(CCR8的内源性配体)引发的信号通路。
-
GC12344
TAPI-1
TAPI
TACE/ADAM17 inhibitor
-
GC27473
4-Amino-3-chloropyridine
4-氨基-3-氯吡啶; 4-Pyridinamine, 3-chloro-; SCHEMBL322241; 3-chloro-4-pyridinylamine; Pyridine, 4-amino-3-chloro-; cid_581853; 4-amino-3-chloropyridine, AldrichCPR; AM20070176; 4-Amino-3-chloropyridine; A4339; 3-chloranylpyridin-4-amine; Eugenol BP; 3-Chloro-4
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GC19322
Pilocarpine
毛果芸香碱
Analytical standard
-
GC27472
4-Amino-3-ethylbenzonitrile
4-氨基-3-乙基苯甲腈; EN300-208814; Z1201617894; 4-Amino-3-ethylbenzonitrile; 4-Amino-3-ethyl-benzonitrile; MFCD00041431; DTXSID30370682; A811180; DS-1636; AMY8917; AKOS006230026; AC-5204; FT-0601004; 4-azanyl-3-ethyl-benzenecarbonitrile; 3-ethyl-4-aminobenzonitr
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GC27471
2-Amino-5-chlorobenzaldehyde
2-氨基-5-氯苯甲醛; 5-氯邻氨基苯甲醛; 4-氯-2-甲酰苯胺; FT-0600665; FT-0659888; EN300-98057; 2-Amino-5-chlorobenzaldehyde; 2-amino-5-chlorobenz-aldehyde; 2-amino-5-chlorobenzaldehyde, AldrichCPR; J-507929; KUIFMGITZFDQMP-UHFFFAOYSA-N; MFCD02093936; DTXSID40378770; 3-chloro-6
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GP20673
Insulin Human
Insulin Human Recombinant
-
GC61006
LS-102
LS102是一种选择性的E3连接酶synoviolin(Syvn1)抑制剂。LS-102抑制Syvn1自泛素化,IC50约为35μM,有研究类风湿关节炎的潜力。
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GC30506
Rhod-2 AM
Rhod-2 Acetoxymethyl ester
Rhod-2 AM是Rhod-2的乙酰甲酯衍生物,可透过细胞膜,通过其乳糖酶切割产生具有不透过膜的Rhod-2,可用来检测细胞或组织Ca2+水平。激发波长为552nm,发射波长为581nm。
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GC48385
SM-102
Lipid H
SM-102 is a synthetic ionizable amino lipid that has been widely used to combine with other lipids to form lipid nanoparticles.
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GB57125
Barium titanium oxide
钛酸钡 氧化钡钛
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GC30806
Cyclo(his-pro) (Cyclo(histidyl-proline))
环(组氨酰-脯氨酰),Cyclo(histidyl-proline); Histidylproline diketopiperazine
A cyclic neuropeptide and metabolite of TRH
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GC10829
Heparin
肝素
injectable anticoagulant
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GC16533
Oligomycin Complex
寡霉素
寡霉素复合物(Oligomycin complex)由寡霉素A、B和C的混合物组成。
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GD20561
Ruthenium(IV) oxide
氧化钌
-
GC39810
CID44216842
Cdc42-IN-1
CID44216842 (Cdc42-IN-1) is a potent Cdc42-selective guanine nucleotide binding lead inhibitor with EC50s of 1.0 μM and 1.2 μM for Cdc42WT and Cdc42Q61L mutant in GTP binding assay, respectively.