- Cat.No. 产品名称 Information
-
GC40928
Trimethylamine N-oxide
三甲胺N-氧化物
A metabolite of choline, phosphatidylcholine, and L-carnitine
-
GC74921
PKA-IN-1
PKA-IN-1 是一种高效、选择性的 cyclic AMP 依赖性蛋白激酶 (PKA) 催化亚基 (cAK) 抑制剂, IC50 为0.03 μM。
-
GN10018
Baicalin
黄芩苷; Baicalein 7-O-β-D-glucuronide
A flavonoid with diverse biological activities
-
GD08281
Cadmium chloride monohydrate
氯化镉一水合物
-
GC16157
740 Y-P
740YPDGFR; PDGFR 740Y-P
PI 3-kinase activator,cell permeable
-
GC50506
Fluorescein-NAD+
Fluorescent NAD+; substrate for ADP-ribosylation for use in PARP assays
-
GC14433
7α,25-dihydroxy Cholesterol
7Α,25-二羟基胆固醇,7α,25-DHC
A GPR183 agonist
-
GC27378
FdUMP triethylammonium
2’-Deoxy-5-Fluorouridine 5’-phosphate triethylammonium
FdUMP (triethylammonium) 是 5-氟尿嘧啶 (5-FU) 的细胞内活性形式。5-FU 转运进入细胞后在多种酶的作用下转化为FdUMP。FdUMP 与胸苷酸合成酶 (thymidylate synthetase) 及其辅因子5,10-亚甲基四氢叶酸 (5,10-methylene tetrahydrofolate) 形成三元配合物抑制胸苷酸合成酶活性,进而导致 DNA 合成被抑制。
-
GC16201
Chlorhexidine digluconate (20% in water)
氯己定二葡糖酸盐
antiseptic
-
GC11183
A 77636 hydrochloride
Agonist of D1-like dopamine receptor,potent and selective
-
GC74063
BNN6
BNN6是一种热反应性NO供体。
-
GC65259
BC-1471
BC-1471, a small-molecule inhibitor of STAM-binding protein (STAMBP) deubiquitinase activity, decreases NACHT, LRR and PYD domains-containing protein 7 (NALP7) protein levels and suppresses IL-1β release after TLR agonism.
-
GC32791
BETd-260 (ZBC 260)
ZBC 260
BETd-260是基于PROTAC技术的一种有效的BET降解剂,在白血病细胞RS4;11中,降低BRD4蛋白活性,IC50值为30pM。
-
GB56466
5-DTAF
5-(4,6-二氯三嗪)氨基荧光素 5-(4,6-Dichlorotriazinyl)aminofluorescein 5-(4,6-二氯三嗪)氨基荧光素 100MG
-
GC10436
VPS34-IN1
Vacuolar Protein Sorting 34 Inhibitor 1, Vps34 Inhibitor 1
Vps34 inhibitor
-
GC11031
PX-478 2HCl
PX-478 is a selective inhibitor that suppresses constitutive and hypoxia-induced HIF-1α levels.
-
GC26550
MFN2 agonist-1
MFN2 agonist-1是一种小分子化合物,作为线粒体融合蛋白Mitofusin 2(MFN2)的激动剂,能够促进线粒体融合,在与线粒体功能障碍相关的疾病中具有潜在的治疗应用价值。
-
GC19186
GW4869
GW4869 is a noncompetitive neutral sphingomyelinase inhibitor with an IC50 of 1 uM.
-
GC27395
Dapirolizumab
Dapirolizumab 是一种针对 CD40 配体的单克隆抗体。Dapirolizumab 靶向 CD40L,阻断其与 CD40 受体的相互作用,并抑制适应性免疫激活。Dapirolizumab 可改善系统性红斑狼疮。
-
GC44867
SAICAR
Succino-AICAR
SAICAR is an intermediate in the de novo purine nucleotide synthesis pathway.
-
GC27394
Tyrode's Solution (calcium-free)
用于两栖类动物离体实验,肌体灌流、清洗组织。并维持离体组织的正常生理功能。
-
GC19000
BAY-588
BAY-588 is a glucose transporter inhibitor and derivative of BAY-876 .
-
GD13990
β-Glucan
β-葡聚糖
β-Glucan是由D-葡萄糖单体通过β-糖苷键连接而成的多糖。β-Glucan具有降胆固醇、降血糖、免疫调节、抗肿瘤、抗氧化和抗炎等功能。
-
GK10014
Protease Inhibitor Cocktail (EDTA-Free,100× in DMSO)
Protease inhibitor cocktail is used in cell lysates or tissue extracts to increase protein stability.
-
GC27393
2,4-Dichloropyridin-3-ol
2,4-二氯吡啶-3-醇
-
GC27384
7-Nitrobenzo[d]thiazol-2-amine
2-氨基-7-硝基苯并噻唑
-
GC27387
2,2'-(Propane-2,2-diyl)bis(4-phenyl-4,5-dihydrooxazole)
2,2'-(丙烷-2,2-二基)双(4-苯基-4,5-二氢恶唑)
-
GC27389
4-Phenylthiazole-5-carbaldehyde
4-苯基噻唑-5-甲醛
-
GC27392
3-Fluoro-2-isobutylpyridine
3-氟-2-异丁基吡啶
-
GC27390
4,7-Dichloropyrido[3,2-d]pyrimidine
4,7-二氯吡啶[3,2-d]嘧啶
-
GC27391
4-(Fluorosulfonyl)-2-methylbenzoic acid
4-(氟磺酰基)-2-甲基苯甲酸
-
GC27388
(5-(Methylsulfonyl)pyridin-3-yl)methanamine
(5-(甲基磺酰基)吡啶-3-基)甲胺
-
GC27386
2-Propyl-7H-purin-6-amine
2-丙基-7H-嘌呤-6-胺
-
GC27385
3-((4-Bromophenyl)amino)propanoic acid
3-((4-溴苯基)氨基)丙酸
-
GC27383
3-Methyl-4-(methylsulfonamido)benzoic acid
3-甲基-4-甲磺酰氨基苯甲酸
-
GC91483
DPPD-Q
C.I. 56000,2,5-Dianilino-1,4-benzoquinone,2,5-Dianilino-p-benzoquinone,2,5-Dianilino-para-benzoquinone,N,N′-Diphenyl-1,4-phenylenediamine quinone,N,N′-Diphenyl-p-phenylenediamine quinone,N,N′-Diphenyl-para-phenylenediamine quinone,NSC 11
DPPD-Q is an oxidized derivative of the antioxidant and substituted p-phenylenediamine DPPD.
-
GC26406
BSA-FITC
BSA≈5mg/ml
-
GC66337
Anti-Mouse PD-L1 Antibody
Anti-Mouse PD-L1 Antibody(10F.9G2)是抗小鼠PD-L1(CD274/B7-H1)的IgG2b抗体抑制剂,宿主是大鼠(Rat)。
-
GC65353
Ezurpimtrostat hydrochloride
GNS561 hydrochloride
Ezurpimtrostat hydrochloride (compound 2-3) 是一种口服有效的抗纤维化剂。Ezurpimtrostat hydrochloride 能明显减轻 DEN (二乙基亚硝胺)肝硬化大鼠的肝纤维化。Ezurpimtrostat hydrochloride 可用于纤维化、癌症、自噬和CTSB、CTSL 和 CTSD 相关的疾病研究。
-
GA22068
H-Arg-Arg-OH
精氨酸二聚体
Arginine-containing dipeptides as RR and RF (G-1515) are used by nitric oxide synthase as substrates in place of Arg.
-
GC68952
ddATP trisodium
2',3'-Dideoxyadenosine 5'-triphosphate trisodium
ddATP trisodium 是一种用于分子生物学和生物化学的核苷酸类似物,主要用于 DNA 测序和聚合酶链反应(PCR)
-
GC65098
ARL67156 triethylamine
FPL 67156 triethylamine
ARL67156 (FPL 67156) triethylamine 是一种 ecto-ATPase 抑制剂。ARL67156 triethylamine 是竞争性 NTPDase1 (CD39),NTPDase3 和 NPP1 抑制剂,Ki 分别为 11,18 和 12 μM。ARL67156 triethylamine 可用于钙化性主动脉瓣疾病、哮喘等疾病的研究。
-
GK10001
Cell Counting Kit-8 (CCK-8)
Cell Counting Kit-8,简称CCK-8试剂盒或CCK8试剂盒,是一种基于WST-8而广泛应用于细胞活性和细胞毒性检测的快速、高灵敏度试剂盒。
-
GC27382
2,6-Difluoro-3-methylphenylboronic acid
2,6-二氟-3-甲基苯基硼酸
-
GP20168
EGF Human
Epidermal Growth Factor Human Recombinant
-
GC43305
Compound 48/80 (hydrochloride)
C48/80 trihydrochloride
Compound 48/80 trihydrochloride is a mixture of condensation products of N-methyl-p-methoxyphenethylamine with formaldehyde.
-
GC42033
1-Palmitoyl-2-oleoyl-sn-glycero-3-PC
2-油酰-1-棕榈锡甘油-3-磷酸胆碱,POPC
A synthetic phosphatidylcholine
-
GC63216
Tesirine
SG3249
Tesirine 是一种抗体药物偶联物(ADC)的吡咯苯并二氮杂卓(PBD)二聚体有效载荷。
-
GC27381
Gentamicin-Amphotericin B (500×), Sterile
庆大霉素-两性霉素 B (500×),无菌
庆大霉素-两性霉素 B (500×),无菌 (Gentamicin-Amphotericin B (500×), Sterile) 是已过滤除菌,可直接用于细胞培养的双抗溶液。含有庆大霉素 5 mg/mL,两性霉素 B 125 μg/mL,建议 500 倍稀释使用。
-
GB55224
3-Methyl-2-oxovaleric acid (sodium)
3-甲基-2-氧戊酸钠