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Home >> Signaling Pathways >> Ubiquitination/ Proteasome

Ubiquitination/ Proteasome(泛素化/蛋白酶体)

  1. Cat.No. 产品名称 Information
  2. GC11669 Tamoxifen Citrate

    他莫昔芬柠檬酸盐; ICI 46474; (Z)-Tamoxifen Citrate; trans-Tamoxifen Citrate

     A selective estrogen receptor modulator
  3. GC16233 Tacrolimus (FK506)

    他克莫司; FK506; Fujimycin; FR900506

     他克莫司 (FK506) 是一种具有强效免疫抑制作用的大环内酯类抗生素，从筑波链霉菌中分离出来，以前曾用于预防人类同种异体移植和治疗自身免疫性疾病。
  4. GC13350 Raloxifene HCl

    盐酸雷洛昔芬; Keoxifene hydrochloride; LY156758; LY139481 hydrochloride

     A selective estrogen receptor modulator
  5. GC11637 Mifepristone

    米非司酮; RU486; RU 38486

     Mifepristone (RU486）是一种口服有效的孕酮（PR）受体和糖皮质激素受体（GR）拮抗剂，用作堕胎药物，体外实验中IC50值分别为0.2nM和2.6nM。
  6. GC11688 Megestrol Acetate

    醋酸甲地孕酮

     A synthetic progestogen
  7. GC17865 Lomustine

    洛莫司汀; CCNU; NSC 79037

     A DNA alkylating agent
  8. GC14961 Cytarabine hydrochloride

    盐酸阿糖胞苷; Cytosine β-D-arabinofuranoside hydrochloride; Cytosine Arabinoside hydrochloride; Ara-C hydrochloride

     A nucleoside analog and prodrug form of ara-CTP
  9. GC11747 Amsacrine hydrochloride

    盐酸胺苯吖啶,m-AMSA hydrochloride; acridinyl anisidide hydrochloride

     A topoisomerase II poison
  10. GC12326 Amsacrine

    安吖啶; m-AMSA; acridinyl anisidide

     A topoisomerase II poison
  11. GC10580 AICAR phosphate

    5-氨基-1-核糖基咪唑-4-甲酰胺磷酸盐,Acadesine phosphate; AICA Riboside phosphate

    An activator of AMPK
  12. GC14292 Apatinib Mesylate

    阿帕替尼

    A selective VEGFR2 inhibitor
  13. GC11006 Montelukast Sodium

    孟鲁司特钠; MK0476

     A CysLT1 receptor antagonist
  14. GC10722 SR-3677

    N-[2-[2-(二甲基氨基)乙氧基]-4-(1H-吡唑-4-基)苯基]-2,3-二氢-1,4-苯并二恶烷-2-甲酰胺

     A ROCK1 and ROCK2 inhibitor
  15. GC10982 YM201636

    6-氨基-N-[3-[4-(4-吗啉基)吡啶并[3',2':4,5]呋喃并[3,2-D]嘧啶-2-基]苯基]-3-吡啶甲酰胺

     Inhibitor of PIKfyve
  16. GC12828 Daunorubicin

    柔红霉素; Daunomycin; RP 13057; Rubidomycin

    Daunorubicin (Daunomycin) 是一种拓扑异构酶 II 抑制剂，具有有效的抗肿瘤活性。
  17. GC10354 Daunorubicin HCl

    盐酸柔红霉素; Daunomycin hydrochloride; RP 13057 hydrochloride; Rubidomycin hydrochloride

     Antitumor antibiotic used in the treatment of acute myeloid leukemias
  18. GC13858 Torin 2

    9-(6-氨基-3-吡啶基)-1-[3-(三氟甲基)苯基]苯并[H]-1,6-萘啶-2(1H)-酮

     Selective inhibitor of mTOR
  19. GC13223 Aliskiren Hemifumarate

    阿利克仑半富马酸盐; CGP 60536 hemifumarate; CGP60536B hemifumarate; SPP 100 hemifumarate

     A nonpeptide renin inhibitor
  20. GC17868 TWS119 A GSK3β inhibitor
  21. GC11424 Valproic acid

    丙戊酸; VPA; 2-Propylpentanoic Acid

     A class I HDAC inhibitor
  22. GC12389 Efavirenz

    依法韦仑; DMP 266; EFV; L-743726

     A non-nucleoside reverse transcriptase inhibitor
  23. GC13468 BI-D1870 An inhibitor of RSK1-4
  24. GC14071 OSI-027

    反式-4-[4-氨基-5-(7-甲氧基-1H-吲哚-2-基)咪唑并[5,1-F][1,2,4]三嗪-7-基]环己烷羧酸,ASP7486

     Dual mTORC1/mTORC2 inhibitor
  25. GC13001 SB 203580 hydrochloride

    SB 203580 hydrochloride; RWJ 64809 hydrochloride

     A water soluble p38 MAPK inhibitor
  26. GC17651 Sunitinib

    舒尼替尼; SU 11248

     舒尼替尼Sunitinib（SU 11248）是一种具口服活性的多靶点受体酪氨酸激酶抑制剂，对血管内皮生长因子受体（VEGFR2）和血小板衍生生长因子受体（PDGFRβ）的IC50分别为80nM和2nM。
  27. GC10198 Memantine hydrochloride

    盐酸美金刚; D-145 hydrochloride

     An NMDA receptor antagonist
  28. GC17243 Dorsomorphin (Compound C)

    6-[4-[2-(1-哌啶基)乙氧基]苯基]-3-(4-吡啶基)吡唑并[1,5-A]嘧啶,Compound C

     Dorsomorphin（Compound C）是一种细胞渗透的AMPK抑制剂。
  29. GC10789 XCT790

    3-[4-[[2,4-二(三氟甲基)苄基]氧基]-3-甲氧基苯基]-2-氰基-N-(5-三氟甲基-[1,3,4]噻二唑-2-基)丙烯酰胺

     A selective inverse agonist of ERRα
  30. GC10734 Beta-Lapachone

    3,4-二氢-2,2-二甲基-2H-萘并[1,2-B]吡喃-5,6-二酮,ARQ-501; NSC-26326

     An anti-cancer quinone
  31. GC11068 GSK2656157 A PERK inhibitor
  32. GC17250 NMS-873

    VCP Inhibitor III

     A selective inhibitor of VCP/p97
  33. GC11375 UNC1999 A selective, cell-permeable EZH2 inhibitor
  34. GC15771 PYR-41 An irreversible inhibitor of ubiquitin-activating enzyme
  35. GC12560 Dorsomorphin (Compound C) 2HCl

    BML-275 2HCl,Compound C 2HCl

    IC50:Dorsomorphin 以剂量依赖性方式抑制 BMP4 诱导的 BMP 反应性 SMAD 磷酸化（半数最大抑制浓度 (IC50) =0.47 mM）。
  36. GC15725 PTC-209 PTC-209 是一种小分子化合物，可选择性抑制 BMI-1，在 HT1080 细胞中的 IC50 为 0.5μM，是一种很有前途的抗癌药物在体外，PTC-209 以 0.1 到 10μM 之间的剂量处理人结直肠癌细胞，以剂量依赖性方式降低 BMI-1 蛋白水平，同时减少细胞生长。
  37. GC13793 NH125 An antibacterial imidazole
  38. GC11932 NSC697923 A selective inhibitor of Ubc13
  39. GC13136 (S)-Crizotinib An MTH1 inhibitor
  40. GC17737 PD 169316

    4-[4-(4-氟苯基)-2-(4-硝基苯基)-1H-咪唑-5-基]吡啶

     A specific p38 MAPK inhibitor
  41. GC16543 TAK-715

    N-(4-(2-乙基-4-(3-甲基苯基)噻唑-5-基)吡啶-2-基)苯甲酰胺

     An inhibitor of p38α MAPK
  42. GC17508 VX-702

    6-[(氨基羰基)(2,6-二氟苯基)氨基]-2-(2,4-二氟苯基)-3-吡啶甲酰胺

     An inhibitor of p38 MAP kinases
  43. GC12926 VX-745

    VX-745

     A p38α MAPK inhibitor
  44. GC10048 MNS

    3,4-亚甲二氧-beta-硝基苯乙烯,NSC 170724; 5-(2-Nitrovinyl)benzodioxole

     An inhibitor of Src, Syk, and platelet aggregation
  45. GC13559 Cilengitide

    西仑吉肽; EMD 121974

     An integrin αVβ3 receptor antagonist
  46. GC17716 Oxaliplatin

    奥沙利铂

    奥沙利铂（Oxaliplatin）是一种用于治疗癌症的细胞毒性化疗药物。
  47. GC16425 Flavopiridol hydrochloride

    (-)-2-(2-氯苯基)-5,7-二羟基-8-[(3S,4R)-3-羟基-1-甲基-4-哌啶基]-4H-1-苯并吡喃-4-酮盐酸盐,Alvocidib Hydrochloride; L86-8275 Hydrochloride; HMR-1275 Hydrochloride

     An inhibitor of cyclin-dependent kinases
  48. GC15741 LY2603618

    LY2603618; IC-83

     A Chk1 inhibitor
  49. GC11229 IOWH-032

    3-(3,5-二溴-4-羟基苯基)-N-(4-苯氧基苄基)-1,2,4-恶二唑-5-甲酰胺

     A modulator of CFTR
  50. GC17519 Concanamycin A

    刀豆素A; Antibiotic X 4357B; Folimycin; X 4357B

     Concanamycin A 是液泡型 ATP 酶 (V-ATPase) 的特异性抑制剂，IC50 值为 10 nM 。
  51. GC15015 (±)-Bay K 8644

    1,4-二氢-2,6-二甲基-5-硝基-4-(2-[三氟甲基]苯基)吡啶-3-羧酸甲酯,SQ 28,873

     A Ca2+ channel activator

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