Search Site
  • 0
    My Cart

    Click Here to Find How Many Items You Have Added:)

qq在线咨询
Home >> Signaling Pathways >> GPCR/G protein >> 5-HT Receptor

5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

Products for  5-HT Receptor

  1. Cat.No. 产品名称 Information
  2. GC31014 Irindalone (Lu 21-098) Irindalone (Lu 21-098) 是一种新型血清素 5-HT2 拮抗剂。
  3. GC31011 FK1052 hydrochloride FK1052 hydrochloride ((±)-FK1052) 是 Fabesetron hydrochloride 的消旋体，是一种有效的 5-HT3 和 5-HT4 受体双重拮抗剂。
  4. GC30999 Pimethixene (Pimetixene) Pimethixene (Pimetixene) 是抗组胺药和抗血清素能化合物，用作抗偏头痛剂。
  5. GC30989 Bromperidol (R-11333)

    An Analytical Reference Standard
  6. GC30982 Eltoprazine (DU 28853) Eltoprazine (DU 28853)(DU28853) 是一种安定或抗侵袭剂，可作为 5-HT1A 和 5-HT1B 受体的激动剂和 5-HT2C 受体的拮抗剂。
  7. GC30980 Pardoprunox hydrochloride (SLV-308 hydrochloride) A dopamine D2 and D3 receptor partial agonist and 5-HT1A agonist
  8. GC30972 Lidanserin (ZK-33839) Lidanserin (ZK-33839) (ZK-33839) 作为 5-HT2A 和 α1-肾上腺素能受体拮抗剂起作用。
  9. GC30964 Vabicaserin hydrochloride (SCA 136) Vabicaserin hydrochloride (SCA 136) 是一种 5-羟色胺 2C (5-HT2C) 受体选择性激动剂，EC50 为 8 nM。
  10. GC30953 Phenylbiguanide (N-Phenylbiguanide) 1-Phenylbiguanide (Phenylbiguanide, PBG, N-Phenylbiguanide) is a 5-hydroxytryptamine3 (5-HT3) receptor agonist with EC50 of 3.0 μM.
  11. GC30939 Eptapirone (F 11440) A potent and selective 5-HT1A receptor agonist
  12. GC30926 Lurasidone (SM-13496) An atypical antipsychotic
  13. GC30910 Eucalyptol (1,8-Cineole) Eucalyptol是5-HT3受体,钾通道,TNF-α和IL-1β的抑制剂。
  14. GC30907 AVN-492 A 5-HT6 receptor antagonist
  15. GC30888 8-OH-DPAT (8-Hydroxy-DPAT)

    8-OH-DPAT, at a pIC50 of 8.19, exhibits robust and specific agonistic activity on 5-HT1A receptors, indicating high selectivity.
  16. GC30880 LP-211 An agonist of 5-HT7 receptors
  17. GC30826 Temanogrel (APD791) Temanogrel (APD791) 是一种高度选择性的 5-HT2A 受体拮抗剂，Ki 为 4.9 nM。
  18. GC30797 lumateperone Tosylate (ITI-007)

    An atypical antipsychotic
  19. GC30796 Nelotanserin (APD125) Nelotanserin (APD125) 是一种有效的 5-HT2A 反向激动剂、中度有效的 5-HT2C 部分反向激动剂和弱 5-HT2B 反向激动剂，在 IP 积累试验中 IC50 分别为 1.7、79、791 nM。
  20. GC30787 Sertindole (Lu 23-174) An atypical antipsychotic
  21. GC30762 Harmine (Telepathine) A unique regulator of PPARγ expression
  22. GC30681 Revexepride Revexepride是一种高度选择性的5-HT4receptor激动剂，也是潜在的CYP3A4enzyme诱导剂，可用于治疗胃食管返流疾病。
  23. GC30446 MHP 133 MHP133是一种多靶点抑制剂，可以抑制AChE的活性，KKi值为69μM;同时抑制毒蕈碱M1和M2受体，5HT4受体和咪唑I2受体。
  24. GC30413 Dolasetron Mesylate (MDL-73147EF) A 5-HT3 receptor antagonist
  25. GC30412 Dolasetron (MDL-73147) A 5-HT3 receptor antagonist
  26. GC30352 Lintopride

    Lintopride是5HT4拮抗剂，对5HT3有轻微拮抗作用。
  27. GC30314 5-HT4 antagonist 1 5-HT4antagonist1是一个5-HT4受体拮抗剂，其pKi值为9.6。
  28. GC30280 Chlorpromazine D6 hydrochloride An internal standard for the quantification of chlorpromazine
  29. GC30273 Tedatioxetine hydrobromide (Lu AA 24530 hydrobromide) Tedatioxetine (Lu AA24530) hydrobromide 可作为 5-HT2A、5-HT2C、5-HT3 和 α；1A-肾上腺素受体拮抗剂，可作为 5-羟色胺和去甲肾上腺素 (NE) 的首选三重再摄取抑制剂 (TRI)。
  30. GC30206 Roluperidone (CYR-101) A dual antagonist of 5-HT2A and σ2 receptors
  31. GC30198 Dolasetron Mesylate hydrate A 5-HT3 receptor antagonist
  32. GC19389 YL0919 YL0919 (YL0919) 是一种具有双重活性的口服抗抑郁药，作为高度选择性的 5-HT 摄取阻滞剂和有效的 5-HT1Areceptor 激动剂 (Ki=0.19 nM)。
  33. GC19354 TG6-10-1 A potent EP2 receptor antagonist
  34. GC19294 Piboserod A selective, potent 5-HT4 receptor antagonist
  35. GC19176 GSK163090 GSK163090 是一种有效的、选择性的和具有口服活性的 5-HT1A/1B/1D 受体拮抗剂，pKi 值分别为 9.4/8.5/9.7。
  36. GC18244 Eltoprazine (hydrochloride) A partial agonist of 5-HT1A, 5-HT1B, and 5-HT2B receptors
  37. GC17488 Trimipramine (maleate) A tricyclic antidepressant
  38. GC14940 5-Methoxytryptamine
  39. GC12587 1-(1-Naphthyl) piperazine (hydrochloride) A serotonin receptor antagonist
  40. GC11100 Flibanserin A 5-HT1A receptor agonist and 5-HT2A receptor antagonist
  41. GC12293 Perphenazine A typical antipsychotic
  42. GC10743 Cyclobenzaprine HCl An Analytical Reference Material
  43. GC11844 Pimavanserin A 5-HT2A inverse agonist
  44. GC13390 DOB hydrochloride An Analytical Reference Standard
  45. GC11338 Org 37684 Org 37684 是一种高效的 5-HT2C 受体激动剂 (pEC50\u003d8.17)。
  46. GC17044 LP 20 hydrochloride ligand of the 5-HT7 receptor
  47. GC17857 PU 02 A selective 5-HT3 receptor antagonist
  48. GC10535 S 32212 hydrochloride An inverse agonist of 5-HT2C receptors
  49. GC11516 DV 7028 hydrochloride 5-HT2A receptor antagonist
  50. GC10495 EMD 281014 hydrochloride 5-HT2A antagonist
  51. GC16807 AT 1015 Long-acting 5-HT2A antagonist

Items 201 to 250 of 463 total

per page
  2. 3
  3. 4
  4. 5
  5. 6
  6. 7

Set Descending Direction