5-HT Receptor(5-羟色胺受体)
5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.
Products for 5-HT Receptor
- Cat.No. 产品名称 Information
- GC12383 SB 258585 hydrochloride A selective 5-HT6 receptor antagonist
- GC13883 Ritanserin A potent 5-HT2A receptor antagonist
- GC15135 Ro 60-0175 fumarate A 5-HT2 receptor agonist
- GC14030 Altanserin hydrochloride 5-HT2A receptor antagonist
- GC11980 WAY 161503 hydrochloride A 5-HT2C receptor agonist
- GC17343 Zacopride hydrochloride Zacopride hydrochloride 是一种高效的 5-HT3 受体拮抗剂,对 5-HT3 和 5-HT4 受体的 Kis 分别为 0.38 和 373 nM。
- GC17706 R-96544 hydrochloride 5-HT2 receptor antagonist
- GC10310 SB 206553 hydrochloride A 5-HT2C and 5-HT2B receptor antagonist
- GC15248 GR 125487 sulfamate 5-HT4 receptor antagonist
- GC14516 Mesulergine hydrochloride 5-HT2A and 2C receptor antagonist
- GC13607 LY 215840 5-HT2/5-HT7 receptor antagonist
- GC17140 GR 127935 hydrochloride A 5-HT1B and 5-HT1D receptor antagonist
- GC13298 NAS-181 NAS181 是一种有效的、选择性的大鼠 5-HT1B 受体拮抗剂,Ki 为 47 nM。
- GC16556 SB 221284 SB 221284 是一种选择性 5-HT2C/2B 受体拮抗剂,对 5-HT2A、5-HT2B 和 5-HT2C 受体的 pKi 值分别为 6.4、7.9 和 8.6。
- GC14347 SB 228357 SB 228357 是一种选择性、有效的口服活性 5-HT2C/2B 受体拮抗剂,5-HT2A、5-HT2B 和 5-HT2C 的 pKi 值分别为 6.9、8.0 和 9.0。
- GC12803 SB 204741 A 5-HT2B receptor antagonist
- GC11624 GR 113808 A 5-HT4 antagonist
- GC16653 CP 94253 hydrochloride A 5-HT1B receptor agonist
- GC12735 SDZ SER 082 fumarate 5-HT2B/2C receptor antagonist
- GC15551 SB 216641 hydrochloride A 5-HT1B receptor antagonist
- GC13438 SB 224289 hydrochloride A 5-HT1B receptor inverse agonist
- GC15630 SR 57227 hydrochloride A 5-HT3 receptor agonist
- GC11231 BW 723C86 hydrochloride A selective HT2B receptor agonist
- GC17524 GR 55562 dihydrochloride 5-HT1B (5-HT1Dβ) silent antagonist
- GC10068 CP 93129 dihydrochloride A 5-HT1B receptor agonist
- GC15979 RS 16566 dihydrochloride (R)-zacopride 结合位点的配体
- GC16553 N-Desmethylclozapine An active metabolite of clozapine
- GC14696 RS 67506 hydrochloride potent and selective 5-HT4 partial agonist
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GC15137
RS 56812 hydrochloride
5-HT3 partial agonist
- GC17745 MK 212 hydrochloride A 5-HT2C receptor agonist
- GC11119 MDL 11,939 A potent 5-HT2A receptor antagonist
- GC14959 2-[1-(4-Piperonyl)piperazinyl]benzothiazole 5-HT4 receptor
- GC16861 RS 23597-190 hydrochloride 5-HT4 receptor antagonist
- GC15569 3-AQC 5-HT3 antagonist
- GC10357 Metergoline A serotonin receptor antagonist
- GC11577 α-Methyl-5-hydroxytryptamine maleate A 5-HT receptor agonist
- GC15235 NAN-190 hydrobromide A 5-HT1A receptor mixed antagonist and partial agonist
- GC14724 Methylergometrine maleate 5-HT1/5-HT2 receptor antagonist
- GC16040 4F 4PP oxalate A 5-HT2A receptor antagonist
- GC16135 Cinanserin hydrochloride A 5-HT receptor antagonist
- GC14814 5-Carboxamidotryptamine maleate 5-HT1 agonist
- GC10401 SB 204070 Potent and selective 5-HT4 receptor antagonist
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GC16031
1-(3-Chlorophenyl)piperazine (hydrochloride)
An Analytical Reference Standard
- GC14149 WAY 208466 dihydrochloride A selective 5-HT6 receptor agonist
- GC14105 Alprenolol hydrochloride A non-selective β-AR and 5-HT receptor antagonist
- GC15011 PNU 109291 5-HT1D receptor agonist
- GC17854 PNU 142633 PNU 142633 是一种高亲和力、选择性和口服活性的 5-HT1D 受体激动剂,对人 5-HT1D 受体和人 5-HT1B 受体的 Kis 分别为 6 nM 和 \u003e 18 000 nM。
- GC11416 Spiperone hydrochloride Spiperone hydrochloride (Spiroperidol hydrochloride) 是一种选择性多巴胺 D2 受体(D2、D3、D4、D1 和 D5 受体的 Ki 值分别为 0.06 nM、0.6 nM、0.08 nM、~350 nM、~3500 nM)和 5-HT2A /5-HT1A 受体 (Kis of 1 nM/49 nM) 拮抗剂。
- GC17734 Pindolol A β1- and β2-AR antagonist
- GC16876 1-Phenylbiguanide hydrochloride 5-HT3 receptor agonist