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5-HT Receptor(5-羟色胺受体)

5-HT receptor (5-hydroxytryptamine receptors) is a group of GPCRs (G protein-coupled receptors) and LGICs (ligand-gated ion channels) found in the central and peripheral nervous systems.

Products for  5-HT Receptor

  1. Cat.No. 产品名称 Information
  2. GC12383 SB 258585 hydrochloride A selective 5-HT6 receptor antagonist
  3. GC13883 Ritanserin A potent 5-HT2A receptor antagonist
  4. GC15135 Ro 60-0175 fumarate A 5-HT2 receptor agonist
  5. GC14030 Altanserin hydrochloride 5-HT2A receptor antagonist
  6. GC11980 WAY 161503 hydrochloride A 5-HT2C receptor agonist
  7. GC17343 Zacopride hydrochloride Zacopride hydrochloride 是一种高效的 5-HT3 受体拮抗剂,对 5-HT3 和 5-HT4 受体的 Kis 分别为 0.38 和 373 nM。
  8. GC17706 R-96544 hydrochloride 5-HT2 receptor antagonist
  9. GC10310 SB 206553 hydrochloride A 5-HT2C and 5-HT2B receptor antagonist
  10. GC15248 GR 125487 sulfamate 5-HT4 receptor antagonist
  11. GC14516 Mesulergine hydrochloride 5-HT2A and 2C receptor antagonist
  12. GC13607 LY 215840 5-HT2/5-HT7 receptor antagonist
  13. GC17140 GR 127935 hydrochloride A 5-HT1B and 5-HT1D receptor antagonist
  14. GC13298 NAS-181 NAS181 是一种有效的、选择性的大鼠 5-HT1B 受体拮抗剂,Ki 为 47 nM。
  15. GC16556 SB 221284 SB 221284 是一种选择性 5-HT2C/2B 受体拮抗剂,对 5-HT2A、5-HT2B 和 5-HT2C 受体的 pKi 值分别为 6.4、7.9 和 8.6。
  16. GC14347 SB 228357 SB 228357 是一种选择性、有效的口服活性 5-HT2C/2B 受体拮抗剂,5-HT2A、5-HT2B 和 5-HT2C 的 pKi 值分别为 6.9、8.0 和 9.0。
  17. GC12803 SB 204741 A 5-HT2B receptor antagonist
  18. GC11624 GR 113808 A 5-HT4 antagonist
  19. GC16653 CP 94253 hydrochloride A 5-HT1B receptor agonist
  20. GC12735 SDZ SER 082 fumarate 5-HT2B/2C receptor antagonist
  21. GC15551 SB 216641 hydrochloride A 5-HT1B receptor antagonist
  22. GC13438 SB 224289 hydrochloride A 5-HT1B receptor inverse agonist
  23. GC15630 SR 57227 hydrochloride A 5-HT3 receptor agonist
  24. GC11231 BW 723C86 hydrochloride A selective HT2B receptor agonist
  25. GC17524 GR 55562 dihydrochloride 5-HT1B (5-HT1Dβ) silent antagonist
  26. GC10068 CP 93129 dihydrochloride A 5-HT1B receptor agonist
  27. GC15979 RS 16566 dihydrochloride (R)-zacopride 结合位点的配体
  28. GC16553 N-Desmethylclozapine An active metabolite of clozapine
  29. GC14696 RS 67506 hydrochloride potent and selective 5-HT4 partial agonist
  30. GC15137 RS 56812 hydrochloride

    5-HT3 partial agonist

  31. GC17745 MK 212 hydrochloride A 5-HT2C receptor agonist
  32. GC11119 MDL 11,939 A potent 5-HT2A receptor antagonist
  33. GC14959 2-[1-(4-Piperonyl)piperazinyl]benzothiazole 5-HT4 receptor
  34. GC16861 RS 23597-190 hydrochloride 5-HT4 receptor antagonist
  35. GC15569 3-AQC 5-HT3 antagonist
  36. GC10357 Metergoline A serotonin receptor antagonist
  37. GC11577 α-Methyl-5-hydroxytryptamine maleate A 5-HT receptor agonist
  38. GC15235 NAN-190 hydrobromide A 5-HT1A receptor mixed antagonist and partial agonist
  39. GC14724 Methylergometrine maleate 5-HT1/5-HT2 receptor antagonist
  40. GC16040 4F 4PP oxalate A 5-HT2A receptor antagonist
  41. GC16135 Cinanserin hydrochloride A 5-HT receptor antagonist
  42. GC14814 5-Carboxamidotryptamine maleate 5-HT1 agonist
  43. GC10401 SB 204070 Potent and selective 5-HT4 receptor antagonist
  44. GC16031 1-(3-Chlorophenyl)piperazine (hydrochloride)

    An Analytical Reference Standard

  45. GC14149 WAY 208466 dihydrochloride A selective 5-HT6 receptor agonist
  46. GC14105 Alprenolol hydrochloride A non-selective β-AR and 5-HT receptor antagonist
  47. GC15011 PNU 109291 5-HT1D receptor agonist
  48. GC17854 PNU 142633 PNU 142633 是一种高亲和力、选择性和口服活性的 5-HT1D 受体激动剂,对人 5-HT1D 受体和人 5-HT1B 受体的 Kis 分别为 6 nM 和 \u003e 18 000 nM。
  49. GC11416 Spiperone hydrochloride Spiperone hydrochloride (Spiroperidol hydrochloride) 是一种选择性多巴胺 D2 受体(D2、D3、D4、D1 和 D5 受体的 Ki 值分别为 0.06 nM、0.6 nM、0.08 nM、~350 nM、~3500 nM)和 5-HT2A /5-HT1A 受体 (Kis of 1 nM/49 nM) 拮抗剂。
  50. GC17734 Pindolol A β1- and β2-AR antagonist
  51. GC16876 1-Phenylbiguanide hydrochloride 5-HT3 receptor agonist

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