Topoisomerase(拓扑异构酶)
Topoisomerase are enzymes that regulate the overwinding or underwinding of DNA.
Products for Topoisomerase
- Cat.No. 产品名称 Information
- GC10354 Daunorubicin HCl Antitumor antibiotic used in the treatment of acute myeloid leukemias
- GC10734 Beta-Lapachone An anti-cancer quinone
- GC16084 Teniposide A topoisomerase II poison
- GC12292 Ofloxacin A fluoroquinolone antibiotic
- GC11114 Moxifloxacin HCl A fluoroquinolone antibiotic
- GC11619 Dexrazoxane HCl (ICRF-187, ADR-529) Topoisomerase IIα inhibitor and intracellular ion chelator
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GC11473
Irinotecan
伊立替康 ((+)-Irinotecan) 是一种拓扑异构酶 I 抑制剂,通过与拓扑异构酶 I-DNA 复合物结合来阻止 DNA 链的重新连接。
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GC10686
Epirubicin HCl
An anthracycline antitumor antibiotic
- GC11019 Amonafide A DNA-intercalating topoisomerase II poison
- GC14969 Idarubicin HCl Antitumor antibiotic used in treatment of leukemia
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GC15617
Etoposide
An inhibitor of topoisomerase II
- GC15548 Ellagic acid Polyphenolic antioxidant
- GC14102 Genistein An isoflavonoid phytoestrogen
- GC14376 Gatifloxacin A fluoroquinolone antibiotic
- GC15439 Camptothecin A DNA enzyme topoisomerase I inhibitor
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GC17567
Doxorubicin (Adriamycin) HCl
An anthracycline antitumor antibiotic
- GC15644 Amrubicin Amrubicin (SM-5887) 是一种 DNA 拓扑异构酶 II 抑制剂,用于癌症研究。
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GC16994
Doxorubicin
多柔比星 (Hydroxydaunorubicin) 是一种具有细胞毒性的蒽环类抗生素,是一种抗癌化疗药物。
- GC14022 Voreloxin Hydrochloride Voreloxin Hydrochloride 是一流的拓扑异构酶 II 抑制剂,可嵌入 DNA 并诱导位点选择性 DNA DSB、G2 停滞和细胞凋亡。
- GC13544 Voreloxin An inhibitor of topoisomerase II
- GC11298 TH-302 A hypoxia-activated anticancer agent
- GC15853 Genz-644282 An inhibitor of topoisomerase I
- GC15250 DOXO-EMCH Prodrug of doxorubicin
- GC17412 Deferasirox Fe3+ chelate Deferasirox Fe3+ Chelate 是从专利 WO2003053986 中提取的铁螯合剂。
- GC11175 Daun02 Daun02 是拓扑异构酶抑制剂柔红霉素的前药。
- GC10480 Betulinic acid A plant triterpenoid similar to bile acids
- GC17271 4'-Demethylepipodophyllotoxin An inhibitor of tubulin polymerization
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GN10523
Berberine Sulfate
硫酸小檗碱是一种从中草药黄连中分离出来的生物碱,作为一种抗生素。
- GN10449 SN-38 (NK012) A potent inhibitor of DNA topoisomerase I
- GN10035 9-Methoxycamptothecin 9-Methoxycamptothecin (MCPT) 分离自 Nothapodytes foetida,通过抑制拓扑异构酶具有抗肿瘤活性。 9-Methoxycamptothecin (MCPT) 在癌症中诱导强烈的 G2/M 期阻滞和细胞凋亡。
- GN10416 Podophyllotoxin A lignan with diverse biological activities
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GN10208
Berberine hydrochloride
盐酸小檗碱是来源于毛茛科药用植物黄连的一种异喹啉类生物碱,具有抗肿瘤、抗炎、降血糖等多种药理活性。
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GN10221
Berberine
小檗碱(Natural Yellow 18)是一种从中草药黄连中分离出来的生物碱,作为一种抗生素。