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Topoisomerase(拓扑异构酶)

Topoisomerase are enzymes that regulate the overwinding or underwinding of DNA.

Products for  Topoisomerase

  1. Cat.No. 产品名称 Information
  2. GC10354 Daunorubicin HCl Antitumor antibiotic used in the treatment of acute myeloid leukemias
  3. GC10734 Beta-Lapachone An anti-cancer quinone
  4. GC16084 Teniposide A topoisomerase II poison
  5. GC12292 Ofloxacin A fluoroquinolone antibiotic
  6. GC11114 Moxifloxacin HCl A fluoroquinolone antibiotic
  7. GC11619 Dexrazoxane HCl (ICRF-187, ADR-529) Topoisomerase IIα inhibitor and intracellular ion chelator
  8. GC11473 Irinotecan

    伊立替康 ((+)-Irinotecan) 是一种拓扑异构酶 I 抑制剂,通过与拓扑异构酶 I-DNA 复合物结合来阻止 DNA 链的重新连接。

  9. GC10686 Epirubicin HCl

    An anthracycline antitumor antibiotic

  10. GC11019 Amonafide A DNA-intercalating topoisomerase II poison
  11. GC14969 Idarubicin HCl Antitumor antibiotic used in treatment of leukemia
  12. GC15617 Etoposide

    An inhibitor of topoisomerase II

  13. GC15548 Ellagic acid Polyphenolic antioxidant
  14. GC14102 Genistein An isoflavonoid phytoestrogen
  15. GC14376 Gatifloxacin A fluoroquinolone antibiotic
  16. GC15439 Camptothecin A DNA enzyme topoisomerase I inhibitor
  17. GC17567 Doxorubicin (Adriamycin) HCl

    An anthracycline antitumor antibiotic

  18. GC15644 Amrubicin Amrubicin (SM-5887) 是一种 DNA 拓扑异构酶 II 抑制剂,用于癌症研究。
  19. GC16994 Doxorubicin

    多柔比星 (Hydroxydaunorubicin) 是一种具有细胞毒性的蒽环类抗生素,是一种抗癌化疗药物。

  20. GC14022 Voreloxin Hydrochloride Voreloxin Hydrochloride 是一流的拓扑异构酶 II 抑制剂,可嵌入 DNA 并诱导位点选择性 DNA DSB、G2 停滞和细胞凋亡。
  21. GC13544 Voreloxin An inhibitor of topoisomerase II
  22. GC11298 TH-302 A hypoxia-activated anticancer agent
  23. GC15853 Genz-644282 An inhibitor of topoisomerase I
  24. GC15250 DOXO-EMCH Prodrug of doxorubicin
  25. GC17412 Deferasirox Fe3+ chelate Deferasirox Fe3+ Chelate 是从专利 WO2003053986 中提取的铁螯合剂。
  26. GC11175 Daun02 Daun02 是拓扑异构酶抑制剂柔红霉素的前药。
  27. GC10480 Betulinic acid A plant triterpenoid similar to bile acids
  28. GC17271 4'-Demethylepipodophyllotoxin An inhibitor of tubulin polymerization
  29. GN10523 Berberine Sulfate

    硫酸小檗碱是一种从中草药黄连中分离出来的生物碱,作为一种抗生素。

  30. GN10449 SN-38 (NK012) A potent inhibitor of DNA topoisomerase I
  31. GN10035 9-Methoxycamptothecin 9-Methoxycamptothecin (MCPT) 分离自 Nothapodytes foetida,通过抑制拓扑异构酶具有抗肿瘤活性。 9-Methoxycamptothecin (MCPT) 在癌症中诱导强烈的 G2/M 期阻滞和细胞凋亡。
  32. GN10416 Podophyllotoxin A lignan with diverse biological activities
  33. GN10208 Berberine hydrochloride

    盐酸小檗碱是来源于毛茛科药用植物黄连的一种异喹啉类生物碱,具有抗肿瘤、抗炎、降血糖等多种药理活性。

  34. GN10221 Berberine

    小檗碱(Natural Yellow 18)是一种从中草药黄连中分离出来的生物碱,作为一种抗生素。

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