mAChR(毒蕈碱型乙酰胆碱受体)
mAChRs (muscarinic acetylcholine receptors) are acetylcholine receptors that form G protein-receptor complexes in the cell membranes of certainneurons and other cells. They play several roles, including acting as the main end-receptor stimulated by acetylcholine released from postganglionic fibersin the parasympathetic nervous system. mAChRs are named as such because they are more sensitive to muscarine than to nicotine. Their counterparts are nicotinic acetylcholine receptors (nAChRs), receptor ion channels that are also important in the autonomic nervous system. Many drugs and other substances (for example pilocarpineand scopolamine) manipulate these two distinct receptors by acting as selective agonists or antagonists. Acetylcholine (ACh) is a neurotransmitter found extensively in the brain and the autonomic ganglia.
Products for mAChR
- Cat.No. 产品名称 Information
- GC15029 Glycopyrrolate A muscarinic acetylcholine receptor antagonist
- GC16059 Tarafenacin D-tartrate Tarafenacin D-tartrate (SVT-40776 D-tartrate) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM),选择性是 M2 受体的约 200 倍。
- GC13618 Tarafenacin Tarafenacin(SVT-40776) 是一种高度选择性的 M3 毒蕈碱受体拮抗剂 (Ki= 0.19 nM),选择性比 M2 受体高约 200 倍。
- GC17760 Clozapine An atypical antipsychotic
- GC14096 Aclidinium Bromide A muscarinic acetylcholine receptor antagonist
- GC16819 VU0152100 A muscarinic M4 receptor positive allosteric modulator
-
GC10621
Biperiden HCl
A muscarinic acetylcholine receptor antagonist
- GC10264 Arecoline hydrobromide Muscarinic acetylcholine receptor agonist
- GC12717 Ipratropium Bromide A muscarinic receptor antagonist
- GC16635 Diphemanil Methylsulfate An anticholinergic agent
- GC14113 Oxybutynin An antagonist of muscarinic acetylcholine receptors
- GC16526 Atropine A non-selective muscarinic acetylcholine receptor antagonist
- GC17779 Levetiracetam An antiepileptic compound
- GC11831 Umeclidinium bromide A muscarinic acetylcholine receptor antagonist
- GC12554 Tiotropium Bromide A muscarinic receptor antagonist
- GC16073 Dronedarone An antiarrhythmic agent
-
GC10822
Clozapine N-oxide (CNO)
clozapine和受体DREADD激动剂的代谢产物
- GC17157 Cevimeline hydrochloride hemihydrate Cevimeline hydrochloride hemihydrate (SNI-2011) 是乙酰胆碱的奎宁环衍生物,是一种选择性和口服活性的毒蕈碱 M1 和 M3 受体激动剂。
- GC14215 Cevimeline A muscarinic receptor agonist
- GN10542 Scopolamine butylbromide An antispasmodic agent