ROR(维甲酸相关孤儿受体)

ROR (RAR-related orphan receptor) is a nuclear receptor family of intracellular transcription factors and appears to bind as monomers to hormone response elements.

Cat.No. 产品名称 Information
GC68411 RORγt Inverse agonist 10
GC66327 Zilovertamab
GC65953 RORγt inverse agonist 23
GC65155 S18-000003 S18-000003, a potent, selective and orally active inhibitor of retinoic acid receptor-related orphan receptor-gamma-t (RORγt), with an IC50 of <30 μM towards human RORγt in competitive binding assays.
GC63458 Cedirogant Cedirogant (ABBV-157) is an orally active RORγt inverse agonist, can be used for psoriasis research.
GC63436 Bevurogant
Bevurogant 是一种类视黄醇相关孤儿受体-γt ( RORγt) 拮抗剂。Bevurogant 可用于慢性炎症性疾病的研究。
GC62623 RORγt Inverse agonist 6
GC62520 TMP780
GC62349 RORγt inverse agonist 13
GC47687 ML-209 An RORγt antagonist
GC47182 Dehydrolithocholic Acid A major metabolite of lithocholic acid
GC50389 XY 018 XY 018 是一种有效的 ROR-γ-选择性拮抗剂。
GC39299 TMP920
GC37944 XY101
GC37557 RORγt Inverse agonist 3
GC37556 ROR agonist-1
GC35214 A-9758
GC34710 PF-06747711
GC33882 GNE-6468
GC32713 Cintirorgon (LYC-55716) A ROR? agonist
GC32044 L 601920-0 (Methyl-3β-hydroxycholenate)
GC31880 AZD-0284
GC31871 GNE-0946
GC31533 Vimirogant (VTP-43742)
GC31163 TMP778
TMP778 is a selective inhibitor of RORγt with an IC50 of 5 nM in the Fluorescence Resonance Energy Transfer (FRET) assay and an IC50 of 17 nM in the RORγ assay.
GC18591 GSK805 An RORγt inverse agonist
GC14054 SR 0987 An agonist of RORγt
GC13905 GSK2981278 An inverse agonist of RORγ
GC10644 Neoruscogenin A bioavailable agonist of RORα
GC14418 SR 1555 (hydrochloride) inverse agonist of RORγ
GC14284 SR 2211 Selective inverse agonist of RORγ
GC15009 SR 1001 An RORα and γ inverse agonist
GC12877 SR3335 A selective inverse agonist of RORα
GC16392 SR1078 A selective RORα/RORγ agonist
GN10325 Nobiletin A flavonoid with diverse biological activities