PKC(蛋白激酶C)
PKC (protein kinase C) is a serine/threonine protein kinase that mediates insulin signaling, actin cytoskeleton, cell mobility, apoptosis and tumorigenesis etc.
- Cat.No. 产品名称 Information
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GC26065
WAY-354831
WAY-354831 exhibits antibacterial activity.
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GC26055
WAY-301398
WAY-301398 (6-methoxynaphthalene) can bind to protein kinase C (PKC).
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GC25662
N-Desmethyltamoxifen
N-Desmethyltamoxifen, the major metabolite of Tamoxifen in humans and a ten-fold more potent protein kinase C (PKC) inhibitor than Tamoxifen, also is a potent regulator of ceramide metabolism in human AML cells, limiting ceramide glycosylation, hydrolysis, and sphingosine phosphorylation.
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GC67686
PKCiota-IN-2 formic
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GC66006
Protein kinase inhibitor H-7
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GC65126
PKC-iota inhibitor 1
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GC64815
Aurothiomalate sodium
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GC64263
Kobophenol A
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GC63778
Myelin Basic Protein TFA
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GC63439
Sangivamycin
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GC63177
Ruboxistaurin
Ruboxistaurin (LY333531) HCl is a β-specific protein kinase C inhibitor. It competitively and reversibly inhibits PKCβ1 and PKCβ2 with IC50 values of 4.7 and 5.9 nM respectively.
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GC49269
Myr-ZIP
A PKMζ inhibitor
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GC62612
CC-90005
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GC62478
ζ-Stat
ζ-Stat (NSC37044) is a specific and atypical protein kinase Cζ (PKCζ) inhibitor, with an IC50 of 5 μM.
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GC61776
Ingenol 3,20-dibenzoate
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GC61585
Pep2m, myristoylated TFA
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GC50704
CRT 0066854 hydrochloride
A PKCι and PKCζ inhibitor
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GC60274
O-Desmethyl Midostaurin
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GC60037
A-3 hydrochloride
A-3 hydrochloride, a potent, cell-permeable, reversible, ATP-competitive non-selective antagonist of various kinases, againsts cAMP-dependent protein kinase (PKA) (Ki=4.3 ?M), casein kinase II (CK2) (Ki=5.1 ?M) and myosin light chain kinase (MLCK) (Ki=7.4 ?M), also inhibits Protein Kinase C (PKC) and casein kinase I (CK1) with Ki values of 47 ?M and 80 ?M, respectively.
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GC38931
N-Desmethyltamoxifen hydrochloride
N-Desmethyltamoxifen hydrochloride (N-Desmethyl tamoxifen HCl), the primary metabolite of tamoxifen, is an estrogen response modifer and protein kinase C inhibitor with IC50 of 25 ?M.
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GC38482
Desmethylglycitein
An active metabolite of daidzein
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GC38388
DCPLA-ME
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GC38186
Daphnoretin
A coumarin with diverse biological activities
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GC38085
Decursinol angelate
A pyranocoumarin with diverse biological activities
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GC45414
CRT0066854
A PKCι and PKCζ inhibitor
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GC37015
Protein Kinase C 19-36
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GC37014
Protein Kinase C 19-31
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GC36974
Procyanidin A1
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GC36833
p32 Inhibitor M36
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GC36282
Hypocrellin A
A perylenequinoid with diverse biological activities
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GC35530
BJE6-106
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GC44729
Prostratin
An HIV re-activator
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GC44655
PKCε Inhibitor Peptide
An inhibitor of PKCε translocation
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GC43993
K252b
A cell-impermeable kinase inhibitor
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GC43286
CMPD101
A GRK2 and GRK3 inhibitor
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GC43105
C8 Ceramide (d18:1.8:0)
A cell-permeable ceramide analog
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GC42747
Afuresertib (hydrochloride)
A pan-Akt inhibitor
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GC40770
L-erythro Sphingosine (d18:1)
A bioactive sphingolipid
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GC32870
Ingenol ((-)-Ingenol)
A PKC activator
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GC32811
LXS196
A PKC inhibitor
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GC32714
Mitoxantrone (mitozantrone)
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GC31959
AS2521780
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GC31912
VTX-27
A PKCθ inhibitor
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GC31892
Decursin ((+)-Decursin)
A phytochemical with diverse biological activities
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GC31711
PKC-IN-1
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GC31656
Ingenol Mebutate (Ingenol 3-angelate)
A natural cytotoxic diterpene ester
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GC30545
Malantide
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GC30200
PKC-theta inhibitor
PKC-theta inhibitor (compound 20) inhibits PKC-θ with an IC50 of 18 nM.
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GC18521
Cercosporin
A cytotoxic phytotoxin
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GC18354
Bisindolylmaleimide X (hydrochloride)
A PKC inhibitor